Results
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1.
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A calcineurin antifungal strategy with analogs of FK506. [electronic resource] by
- Nambu, Mitchell
- Covel, Jonathan A
- Kapoor, Mili
- Li, Xiaoming
- Moloney, Molly K
- Numa, Mehdi M
- Soltow, Quinlyn A
- Trzoss, Michael
- Webb, Peter
- Webb, Robert R
- Mutz, Mitchell
Producer: 20171219
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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2.
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Solubilized phenyl-pyrazole ureas as potent, selective 5-HT(2A) inverse-agonists and their application as antiplatelet agents. [electronic resource] by
- Dosa, Peter I
- Strah-Pleynet, Sonja
- Jayakumar, Honnappa
- Casper, Martin
- Decaire, Marc
- Xiong, Yifeng
- Lehmann, Juerg
- Choi, Karoline
- Elwell, Katie
- Wong, Amy
- Webb, Robert R
- Adams, John W
- Ramirez, Juan
- Richman, Jeremy G
- Thomsen, William
- Semple, Graeme
- Teegarden, Bradley R
Producer: 20091123
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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3.
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Design, synthesis and in vitro evaluation of potent, novel, small molecule inhibitors of plasminogen activator inhibitor-1. [electronic resource] by
- Folkes, Adrian
- Brown, S David
- Canne, Lynne E
- Chan, Jocelyn
- Engelhardt, Erin
- Epshteyn, Sergey
- Faint, Richard
- Golec, Julian
- Hanel, Art
- Kearney, Patrick
- Leahy, James W
- Mac, Morrison
- Matthews, David
- Prisbylla, Michael P
- Sanderson, Jason
- Simon, Reyna J
- Tesfai, Zerom
- Vicker, Nigel
- Wang, Shouming
- Webb, Robert R
- Charlton, Peter
Producer: 20020917
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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4.
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Discovery and SAR of new benzazepines as potent and selective 5-HT(2C) receptor agonists for the treatment of obesity. [electronic resource] by
- Smith, Brian M
- Smith, Jeffrey M
- Tsai, James H
- Schultz, Jeffrey A
- Gilson, Charles A
- Estrada, Scott A
- Chen, Rita R
- Park, Douglas M
- Prieto, Emily B
- Gallardo, Charlemagne S
- Sengupta, Dipanjan
- Thomsen, William J
- Saldana, Hazel R
- Whelan, Kevin T
- Menzaghi, Frederique
- Webb, Robert R
- Beeley, Nigel R A
Producer: 20050705
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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5.
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Discovery and structure-activity relationship of 3-methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): a highly selective 5-hydroxytryptamine2A receptor inverse agonist for the treatment of arterial thrombosis. [electronic resource] by
- Xiong, Yifeng
- Teegarden, Bradley R
- Choi, Jin-Sun Karoline
- Strah-Pleynet, Sonja
- Decaire, Marc
- Jayakumar, Honnappa
- Dosa, Peter I
- Casper, Martin D
- Pham, Lan
- Feichtinger, Konrad
- Ullman, Brett
- Adams, John
- Yuskin, Diane
- Frazer, John
- Morgan, Michael
- Sadeque, Abu
- Chen, Weichao
- Webb, Robert R
- Connolly, Daniel T
- Semple, Graeme
- Al-Shamma, Hussien
Producer: 20100701
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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6.
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A new family of H3 receptor antagonists based on the natural product Conessine. [electronic resource] by
- Santora, Vincent J
- Covel, Jonathan A
- Hayashi, Rena
- Hofilena, Brian J
- Ibarra, Jason B
- Pulley, Michelle D
- Weinhouse, Michael I
- Sengupta, Dipanjan
- Duffield, Jonathan J
- Semple, Graeme
- Webb, Robert R
- Sage, Carleton
- Ren, Albert
- Pereira, Guilherme
- Knudsen, Jens
- Edwards, Jeffrey E
- Suarez, Marissa
- Frazer, John
- Thomsen, William
- Hauser, Erin
- Whelan, Kevin
- Grottick, Andrew J
Producer: 20080512
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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7.
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Discovery of 1-[3-(4-bromo-2-methyl-2h-pyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea (nelotanserin) and related 5-hydroxytryptamine2A inverse agonists for the treatment of insomnia. [electronic resource] by
- Teegarden, Bradley R
- Li, Hongmei
- Jayakumar, Honnappa
- Strah-Pleynet, Sonja
- Dosa, Peter I
- Selaya, Susan D
- Kato, Naomi
- Elwell, Katie H
- Davidson, Jarrod
- Cheng, Karen
- Saldana, Hazel
- Frazer, John M
- Whelan, Kevin
- Foster, Jonathan
- Espitia, Stephan
- Webb, Robert R
- Beeley, Nigel R A
- Thomsen, William
- Morairty, Stephen R
- Kilduff, Thomas S
- Al-Shamma, Hussien A
Producer: 20100401
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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8.
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Discovery and structure-activity relationship of (1R)-8-chloro-2,3,4,5-tetrahydro-1-methyl-1H-3-benzazepine (Lorcaserin), a selective serotonin 5-HT2C receptor agonist for the treatment of obesity. [electronic resource] by
- Smith, Brian M
- Smith, Jeffrey M
- Tsai, James H
- Schultz, Jeffrey A
- Gilson, Charles A
- Estrada, Scott A
- Chen, Rita R
- Park, Douglas M
- Prieto, Emily B
- Gallardo, Charlemagne S
- Sengupta, Dipanjan
- Dosa, Peter I
- Covel, Jon A
- Ren, Albert
- Webb, Robert R
- Beeley, Nigel R A
- Martin, Michael
- Morgan, Michael
- Espitia, Stephen
- Saldana, Hazel R
- Bjenning, Christina
- Whelan, Kevin T
- Grottick, Andrew J
- Menzaghi, Frederique
- Thomsen, William J
Producer: 20080417
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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