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Discovery of substituted-2,4-dimethyl-(naphthalene-4-carbonyl)amino-benzoic acid as potent and selective EP4 antagonists. [electronic resource] by
- Blanco, Maria-Jesus
- Vetman, Tatiana
- Chandrasekhar, Srinivasan
- Fisher, Matthew J
- Harvey, Anita
- Mudra, Daniel
- Wang, Xu-Shan
- Yu, Xiao-Peng
- Schiffler, Matthew A
- Warshawsky, Alan M
Producer: 20160726
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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4.
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Discovery of potent aryl-substituted 3-[(3-methylpyridine-2-carbonyl) amino]-2,4-dimethyl-benzoic acid EP4 antagonists with improved pharmacokinetic profile. [electronic resource] by
- Blanco, Maria-Jesus
- Vetman, Tatiana
- Chandrasekhar, Srinivasan
- Fisher, Matthew J
- Harvey, Anita
- Chambers, Mark
- Lin, Chaohua
- Mudra, Daniel
- Oskins, Jennifer
- Wang, Xu-Shan
- Yu, Xiao-Peng
- Warshawsky, Alan M
Producer: 20161013
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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5.
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Identification and biological activity of 6-alkyl-substituted 3-methyl-pyridine-2-carbonyl amino dimethyl-benzoic acid EP4 antagonists. [electronic resource] by
- Blanco, Maria-Jesus
- Vetman, Tatiana
- Chandrasekhar, Srinivasan
- Fisher, Matthew J
- Harvey, Anita
- Kuklish, Steven L
- Chambers, Mark
- Lin, Chaohua
- Mudra, Daniel
- Oskins, Jennifer
- Wang, Xu-Shan
- Yu, Xiao-Peng
- Warshawsky, Alan M
Producer: 20161219
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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6.
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Tetrahydroisoquinoline PPARgamma agonists: design of novel, highly selective non-TZD antihyperglycemic agents. [electronic resource] by
- Henry, James R
- Li, Yihong
- Warshawsky, Alan M
- Brozinick, Joseph T
- Hawkins, Eric D
- Misener, Elizabeth A
- Briere, Daniel A
- Montrose-Rafizadeh, Chahrzad
- Zink, Richard W
- Yumibe, Nathan P
- Ajamie, Rose T
- Wilken, Brad
- Devanarayan, Viswanath
Producer: 20070216
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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7.
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Analgesic and anti-inflammatory properties of novel, selective, and potent EP4 receptor antagonists. [electronic resource] by
- Chandrasekhar, Srinivasan
- Yu, Xiao-Peng
- Harvey, Anita K
- Oskins, Jennifer L
- Lin, Chaohua
- Wang, Xushan
- Blanco, Maria-Jesus
- Fisher, Matthew J
- Kuklish, Steven L
- Schiffler, Matthew A
- Vetman, Tatiana
- Warshawsky, Alan M
- York, Jeremy S
- Bendele, Alison M
- Chambers, Mark G
Publication details: Pharmacology research & perspectives 06 2017
In:
Pharmacology research & perspectives vol. 5
Availability: No items available.
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8.
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Design and synthesis of novel and potent amide linked PPARgamma/delta dual agonists. [electronic resource] by
- Shi, Qing
- Canada, Emily J
- Xu, Yanping
- Warshawsky, Alan M
- Etgen, Garret J
- Broderick, Carol L
- Clutinger, Cathleen K
- Irwin, Lynnie A
- Laurila, Michael E
- Montrose-Rafizadeh, Chahrzad
- Oldham, Brian A
- Wang, Minmin
- Winneroski, Leonard L
- Xie, Chaoyu
- York, Jeremy S
- Yumibe, Nathan P
- Zink, Richard W
- Mantlo, Nathan
Producer: 20080303
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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9.
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Synthesis and evaluation of aminomethyl dihydrocinnamates as a new class of PPAR ligands. [electronic resource] by
- Warshawsky, Alan M
- Alt, Charles A
- Brozinick, Joseph T
- Harkness, Allen R
- Hawkins, Eric D
- Henry, James R
- Matthews, Donald P
- Miller, Anne R
- Misener, Elizabeth A
- Montrose-Rafizadeh, Chahrzad
- Rhodes, Gary A
- Shen, Quanrong
- Vance, Jennifer A
- Udodong, Uko E
- Wang, Minmin
- Zhang, Tony Y
- Zink, Richard W
Producer: 20070216
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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10.
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Characterization of 3,3-dimethyl substituted N-aryl piperidines as potent microsomal prostaglandin E synthase-1 inhibitors. [electronic resource] by
- Kuklish, Steven L
- Antonysamy, Stephen
- Bhattachar, Shobha N
- Chandrasekhar, Srinivasan
- Fisher, Matthew J
- Fretland, Adrian J
- Gooding, Karen
- Harvey, Anita
- Hughes, Norman E
- Luz, John G
- Manninen, Peter R
- McGee, James E
- Navarro, Antonio
- Norman, Bryan H
- Partridge, Katherine M
- Quimby, Steven J
- Schiffler, Matthew A
- Sloan, Ashley V
- Warshawsky, Alan M
- York, Jeremy S
- Yu, Xiao-Peng
Producer: 20170717
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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11.
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Discovery and characterization of [(cyclopentyl)ethyl]benzoic acid inhibitors of microsomal prostaglandin E synthase-1. [electronic resource] by
- Partridge, Katherine M
- Antonysamy, Stephen
- Bhattachar, Shobha N
- Chandrasekhar, Srinivasan
- Fisher, Matthew J
- Fretland, Adrian
- Gooding, Karen
- Harvey, Anita
- Hughes, Norman E
- Kuklish, Steven L
- Luz, John G
- Manninen, Peter R
- McGee, James E
- Mudra, Daniel R
- Navarro, Antonio
- Norman, Bryan H
- Quimby, Steven J
- Schiffler, Matthew A
- Sloan, Ashley V
- Warshawsky, Alan M
- Weller, Jennifer M
- York, Jeremy S
- Yu, Xiao-Peng
Producer: 20170926
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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12.
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Discovery of LY3104607: A Potent and Selective G Protein-Coupled Receptor 40 (GPR40) Agonist with Optimized Pharmacokinetic Properties to Support Once Daily Oral Treatment in Patients with Type 2 Diabetes Mellitus. [electronic resource] by
- Hamdouchi, Chafiq
- Maiti, Pranab
- Warshawsky, Alan M
- DeBaillie, Amy C
- Otto, Keith A
- Wilbur, Kelly L
- Kahl, Steven D
- Patel Lewis, Anjana
- Cardona, Guemalli R
- Zink, Richard W
- Chen, Keyue
- Cr, Siddaramaiah
- Lineswala, Jayana P
- Neathery, Grace L
- Bouaichi, Cecilia
- Diseroad, Benjamin A
- Campbell, Alison N
- Sweetana, Stephanie A
- Adams, Lisa A
- Cabrera, Over
- Ma, Xiaosu
- Yumibe, Nathan P
- Montrose-Rafizadeh, Chahrzad
- Chen, Yanyun
- Miller, Anne Reifel
Producer: 20190218
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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13.
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2-Alkoxydihydrocinnamates as PPAR agonists. Activity modulation by the incorporation of phenoxy substituents. [electronic resource] by
- Martín, José A
- Brooks, Dawn A
- Prieto, Lourdes
- González, Rosario
- Torrado, Alicia
- Rojo, Isabel
- López de Uralde, Beatriz
- Lamas, Carlos
- Ferritto, Rafael
- Dolores Martín-Ortega, María
- Agejas, Javier
- Parra, Francisco
- Rizzo, John R
- Rhodes, Gary A
- Robey, Roger L
- Alt, Charles A
- Wendel, Samuel R
- Zhang, Tony Y
- Reifel-Miller, Anne
- Montrose-Rafizadeh, Chahrzad
- Brozinick, Joseph T
- Hawkins, Eric
- Misener, Elizabeth A
- Briere, Daniel A
- Ardecky, Robert
- Fraser, James D
- Warshawsky, Alan M
Producer: 20050502
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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