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Covalent Inhibition of the Histamine H [electronic resource] by
- Wágner, Gábor
- Mocking, Tamara A M
- Kooistra, Albert J
- Slynko, Inna
- Ábrányi-Balogh, Péter
- Keserű, György M
- Wijtmans, Maikel
- Vischer, Henry F
- de Esch, Iwan J P
- Leurs, Rob
Producer: 20200505
In:
Molecules (Basel, Switzerland) vol. 24
Availability: No items available.
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4.
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Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: hit-to-lead optimization. [electronic resource] by
- Nógrádi, Katalin
- Wágner, Gábor
- Domány, György
- Bobok, Amrita
- Magdó, Ildikó
- Kiss, Béla
- Kolok, Sándor
- Fónagy, Katalin
- Gyertyán, István
- Háda, Viktor
- Kóti, János
- Gál, Krisztina
- Farkas, Sándor
- Keserű, György M
- Greiner, István
- Szombathelyi, Zsolt
Producer: 20150306
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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5.
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Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Lead optimization. [electronic resource] by
- Nógrádi, Katalin
- Wágner, Gábor
- Domány, György
- Bobok, Amrita
- Magdó, Ildikó
- Kolok, Sándor
- Mikó-Bakk, Mónika L
- Vastag, Mónika
- Sághy, Katalin
- Gyertyán, István
- Kóti, János
- Gál, Krisztina
- Farkas, Sándor
- Keserű, György M
- Greiner, István
- Szombathelyi, Zsolt
Producer: 20151221
In:
Bioorganic & medicinal chemistry letters vol. 25
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Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs. [electronic resource] by
- Wágner, Gábor
- Wéber, Csaba
- Nyéki, Olga
- Nógrádi, Katalin
- Bielik, Attila
- Molnár, László
- Bobok, Amrita
- Horváth, Attila
- Kiss, Béla
- Kolok, Sándor
- Nagy, József
- Kurkó, Dalma
- Gál, Krisztina
- Greiner, István
- Szombathelyi, Zsolt
- Keseru, György M
- Domány, György
Producer: 20100913
In:
Bioorganic & medicinal chemistry letters vol. 20
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4-Aryl-3-arylsulfonyl-quinolines as negative allosteric modulators of metabotropic GluR5 receptors: From HTS hit to development candidate. [electronic resource] by
- Galambos, János
- Domány, György
- Nógrádi, Katalin
- Wágner, Gábor
- Keserű, György M
- Bobok, Amrita
- Kolok, Sándor
- Mikó-Bakk, Mónika L
- Vastag, Mónika
- Sághy, Katalin
- Kóti, János
- Szakács, Zoltán
- Béni, Zoltán
- Gál, Krisztina
- Szombathelyi, Zsolt
- Greiner, István
Producer: 20160930
In:
Bioorganic & medicinal chemistry letters vol. 26
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8.
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4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H [electronic resource] by
- Wágner, Gábor
- Mocking, Tamara A M
- Arimont, Marta
- Provensi, Gustavo
- Rani, Barbara
- Silva-Marques, Bruna
- Latacz, Gniewomir
- Da Costa Pereira, Daniel
- Karatzidou, Christina
- Vischer, Henry F
- Wijtmans, Maikel
- Kieć-Kononowicz, Katarzyna
- de Esch, Iwan J P
- Leurs, Rob
Producer: 20200622
In:
Journal of medicinal chemistry vol. 62
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Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu [electronic resource] by
- Galambos, János
- Bielik, Attila
- Wágner, Gábor
- Domány, György
- Kóti, János
- Béni, Zoltán
- Szigetvári, Áron
- Sánta, Zsuzsanna
- Orgován, Zoltán
- Bobok, Amrita
- Kiss, Béla
- Mikó-Bakk, Mónika L
- Vastag, Mónika
- Sághy, Katalin
- Krasavin, Mikhail
- Gál, Krisztina
- Greiner, István
- Szombathelyi, Zsolt
- Keserű, György M
Producer: 20170913
In:
European journal of medicinal chemistry vol. 133
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10.
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Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists. [electronic resource] by
- Galambos, János
- Wágner, Gábor
- Nógrádi, Katalin
- Bielik, Attila
- Molnár, László
- Bobok, Amrita
- Horváth, Attila
- Kiss, Béla
- Kolok, Sándor
- Nagy, József
- Kurkó, Dalma
- Bakk, Mónika L
- Vastag, Mónika
- Sághy, Katalin
- Gyertyán, István
- Gál, Krisztina
- Greiner, István
- Szombathelyi, Zsolt
- Keseru, György M
- Domány, György
Producer: 20101123
In:
Bioorganic & medicinal chemistry letters vol. 20
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11.
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Discovery and Preclinical Characterization of 3-((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications. [electronic resource] by
- Galambos, János
- Bielik, Attila
- Krasavin, Mikhail
- Orgován, Zoltán
- Domány, György
- Nógrádi, Katalin
- Wágner, Gábor
- Balogh, György T
- Béni, Zoltán
- Kóti, János
- Szakács, Zoltán
- Bobok, Amrita
- Kolok, Sándor
- Mikó-Bakk, Mónika L
- Vastag, Mónika
- Sághy, Katalin
- Laszy, Judit
- Halász, Attila Sándor
- Balázs, Ottilia
- Gál, Krisztina
- Greiner, István
- Szombathelyi, Zsolt
- Keserű, György M
Producer: 20170619
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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