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Quinoline-3-carboxamide containing sulfones as liver X receptor (LXR) agonists with binding selectivity for LXRbeta and low blood-brain penetration. [electronic resource] by
- Hu, Baihua
- Bernotas, Ron
- Unwalla, Rayomand
- Collini, Michael
- Quinet, Elaine
- Feingold, Irene
- Goos-Nilsson, Annika
- Wilhelmsson, Anna
- Nambi, Ponnal
- Evans, Mark
- Wrobel, Jay
Producer: 20100420
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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11.
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4-(3-aryloxyaryl)quinoline alcohols are liver X receptor agonists. [electronic resource] by
- Bernotas, Ronald C
- Kaufman, David H
- Singhaus, Robert R
- Ullrich, John
- Unwalla, Rayomand
- Quinet, Elaine
- Nambi, Ponnal
- Wilhelmsson, Anna
- Goos-Nilsson, Annika
- Wrobel, Jay
Producer: 20100212
In:
Bioorganic & medicinal chemistry vol. 17
Availability: No items available.
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12.
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Carboxylic acid based quinolines as liver X receptor modulators that have LXRbeta receptor binding selectivity. [electronic resource] by
- Hu, Baihua
- Quinet, Elaine
- Unwalla, Rayomand
- Collini, Mike
- Jetter, James
- Dooley, Rebecca
- Andraka, Diane
- Nogle, Lisa
- Savio, Dawn
- Halpern, Anita
- Goos-Nilsson, Annika
- Wilhelmsson, Anna
- Nambi, Ponnal
- Wrobel, Jay
Producer: 20080212
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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13.
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Biarylether amide quinolines as liver X receptor agonists. [electronic resource] by
- Bernotas, Ronald C
- Singhaus, Robert R
- Kaufman, David H
- Ullrich, John
- Fletcher, Horace
- Quinet, Elaine
- Nambi, Ponnal
- Unwalla, Rayomand
- Wilhelmsson, Anna
- Goos-Nilsson, Annika
- Farnegardh, Mathias
- Wrobel, Jay
Producer: 20090916
In:
Bioorganic & medicinal chemistry vol. 17
Availability: No items available.
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14.
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Identification of phenylsulfone-substituted quinoxaline (WYE-672) as a tissue selective liver X-receptor (LXR) agonist. [electronic resource] by
- Hu, Baihua
- Unwalla, Rayomand J
- Goljer, Igor
- Jetter, James W
- Quinet, Elaine M
- Berrodin, Thomas J
- Basso, Michael D
- Feingold, Irene B
- Nilsson, Annika Goos
- Wilhelmsson, Anna
- Evans, Mark J
- Wrobel, Jay E
Producer: 20100514
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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15.
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4-(3-Aryloxyaryl)quinoline sulfones are potent liver X receptor agonists. [electronic resource] by
- Bernotas, Ronald C
- Singhaus, Robert R
- Kaufman, David H
- Travins, Jeremy M
- Ullrich, John W
- Unwalla, Rayomand
- Quinet, Elaine
- Evans, Mark
- Nambi, Ponnal
- Olland, Andrea
- Kauppi, Björn
- Wilhelmsson, Anna
- Goos-Nilsson, Annika
- Wrobel, Jay
Producer: 20100506
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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16.
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Synthesis of 4-(3-biaryl)quinoline sulfones as potent liver X receptor agonists. [electronic resource] by
- Ullrich, John W
- Morris, Robert
- Bernotas, Ronald C
- Travins, Jeremy M
- Jetter, James
- Unwalla, Rayomand
- Quinet, Elaine
- Nambi, Ponnal
- Feingold, Irene
- Huselton, Christine
- Enroth, Christofer
- Wilhelmsson, Anna
- Goos-Nilsson, Annika
- Wrobel, Jay
Producer: 20100727
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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17.
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Discovery of (2S,4R)-1-(2-aminoacetyl)-4-benzamidopyrrolidine-2-carboxylic acid hydrochloride (GAP-134)13, an orally active small molecule gap-junction modifier for the treatment of atrial fibrillation. [electronic resource] by
- Butera, John A
- Larsen, Bjarne Due
- Hennan, James K
- Kerns, Edward
- Di, Li
- Alimardanov, Asaf
- Swillo, Robert E
- Morgan, Gwen A
- Liu, Kun
- Wang, Qiang
- Rossman, Eric I
- Unwalla, Rayomand
- McDonald, Leonard
- Huselton, Christine
- Petersen, Jørgen S
Producer: 20090709
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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18.
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Molecular and pharmacological properties of a potent and selective novel nonsteroidal progesterone receptor agonist tanaproget. [electronic resource] by
- Zhang, Zhiming
- Olland, Andrea M
- Zhu, Yuan
- Cohen, Jeff
- Berrodin, Tom
- Chippari, Susan
- Appavu, Chandrasekaran
- Li, Shen
- Wilhem, James
- Chopra, Raj
- Fensome, Andrew
- Zhang, Puwen
- Wrobel, Jay
- Unwalla, Rayomand J
- Lyttle, C Richard
- Winneker, Richard C
Producer: 20051012
In:
The Journal of biological chemistry vol. 280
Availability: No items available.
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19.
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Structure-based design of estrogen receptor-beta selective ligands. [electronic resource] by
- Manas, Eric S
- Unwalla, Rayomand J
- Xu, Zhang B
- Malamas, Michael S
- Miller, Chris P
- Harris, Heather A
- Hsiao, Chulai
- Akopian, Tatos
- Hum, Wah-Tung
- Malakian, Karl
- Wolfrom, Scott
- Bapat, Ashok
- Bhat, Ramesh A
- Stahl, Mark L
- Somers, William S
- Alvarez, Juan C
Producer: 20050113
In:
Journal of the American Chemical Society vol. 126
Availability: No items available.
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20.
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Further modification on phenyl acetic acid based quinolines as liver X receptor modulators. [electronic resource] by
- Hu, Baihua
- Jetter, James
- Kaufman, David
- Singhaus, Robert
- Bernotas, Ronald
- Unwalla, Rayomand
- Quinet, Elaine
- Savio, Dawn
- Halpern, Anita
- Basso, Michael
- Keith, James
- Clerin, Valerie
- Chen, Liang
- Liu, Qiang-Yuan
- Feingold, Irene
- Huselton, Christine
- Azam, Farooq
- Goos-Nilsson, Annika
- Wilhelmsson, Anna
- Nambi, Ponnal
- Wrobel, Jay
Producer: 20070627
In:
Bioorganic & medicinal chemistry vol. 15
Availability: No items available.
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