Discovery and SAR of cinnolines/quinolines as liver X receptor (LXR) agonists with binding selectivity for LXRbeta. [electronic resource]
Producer: 20090630Description: 3519-27 p. digitalISSN:- 1464-3391
- ATP Binding Cassette Transporter 1
- ATP-Binding Cassette Transporters -- metabolism
- Animals
- Cell Line
- Computer Simulation
- DNA-Binding Proteins -- agonists
- Drug Discovery
- Heterocyclic Compounds, 2-Ring -- chemistry
- Humans
- Liver X Receptors
- Mice
- Orphan Nuclear Receptors
- Quinolines -- chemical synthesis
- Receptors, Cytoplasmic and Nuclear -- agonists
- Sterol Regulatory Element Binding Protein 1 -- metabolism
- Structure-Activity Relationship
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Publication Type: Journal Article
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