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Kinetics of 5-HT2B receptor signaling: profound agonist-dependent effects on signaling onset and duration. [electronic resource] by
- Unett, David J
- Gatlin, Joel
- Anthony, Todd L
- Buzard, Daniel J
- Chang, Steve
- Chen, Chuan
- Chen, Xiaohua
- Dang, Huong T-M
- Frazer, John
- Le, Minh K
- Sadeque, Abu J M
- Xing, Charles
- Gaidarov, Ibragim
Producer: 20140123
In:
The Journal of pharmacology and experimental therapeutics vol. 347
Availability: No items available.
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5.
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Discovery of a lead series of potent benzodiazepine 5-HT [electronic resource] by
- Ren, Albert
- Zhu, Xiuwen
- Feichtinger, Konrad
- Lehman, Juerg
- Kasem, Michelle
- Schrader, Thomas O
- Wong, Amy
- Dang, Huong
- Le, Minh
- Frazer, John
- Unett, David J
- Grottick, Andrew J
- Whelan, Kevin T
- Morgan, Michael E
- Sage, Carleton R
- Semple, Graeme
Producer: 20210421
In:
Bioorganic & medicinal chemistry letters vol. 30
Availability: No items available.
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6.
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Discovery of a new series of potent prostacyclin receptor agonists with in vivo activity in rat. [electronic resource] by
- Tran, Thuy-Anh
- Shin, Young-Jun
- Kramer, Bryan
- Choi, Juyi
- Zou, Ning
- Vallar, Pureza
- Martens, Peter
- Boatman, P Douglas
- Adams, John W
- Ramirez, Juan
- Shi, Yunqing
- Morgan, Michael
- Unett, David J
- Chang, Steve
- Shu, Hsin-Hui
- Tung, Shiu-Feng
- Semple, Graeme
Producer: 20151215
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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7.
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Discovery of APD371: Identification of a Highly Potent and Selective CB [electronic resource] by
- Han, Sangdon
- Thoresen, Lars
- Jung, Jae-Kyu
- Zhu, Xiuwen
- Thatte, Jayant
- Solomon, Michelle
- Gaidarov, Ibragim
- Unett, David J
- Yoon, Woo Hyun
- Barden, Jeremy
- Sadeque, Abu
- Usmani, Amin
- Chen, Chuan
- Semple, Graeme
- Grottick, Andrew J
- Al-Shamma, Hussein
- Christopher, Ronald
- Jones, Robert M
Publication details: ACS medicinal chemistry letters Dec 2017
In:
ACS medicinal chemistry letters vol. 8
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Discovery of the first potent and orally efficacious agonist of the orphan G-protein coupled receptor 119. [electronic resource] by
- Semple, Graeme
- Fioravanti, Beatriz
- Pereira, Guillherme
- Calderon, Imelda
- Uy, Jane
- Choi, Karoline
- Xiong, Yifeng
- Ren, Albert
- Morgan, Michael
- Dave, Vibha
- Thomsen, William
- Unett, David J
- Xing, Charles
- Bossie, Stuart
- Carroll, Chris
- Chu, Zhi-Liang
- Grottick, Andrew J
- Hauser, Erin K
- Leonard, James
- Jones, Robert M
Producer: 20081024
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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9.
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Discovery and optimization of 5-fluoro-4,6-dialkoxypyrimidine GPR119 agonists. [electronic resource] by
- Buzard, Daniel J
- Kim, Sun Hee
- Lehmann, Juerg
- Han, Sangdon
- Calderon, Imelda
- Wong, Amy
- Kawasaki, Andrew
- Narayanan, Sanju
- Bhat, Rohit
- Gharbaoui, Tawfik
- Lopez, Luis
- Yue, Dawei
- Whelan, Kevin
- Al-Shamma, Hussien
- Unett, David J
- Shu, Hsin-Hui
- Tung, Shiu-Feng
- Chang, Steve
- Chuang, Ching-Fen
- Morgan, Michael
- Sadeque, Abu
- Chu, Zhi-Liang
- Leonard, James N
- Jones, Robert M
Producer: 20150330
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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10.
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Discovery of a novel trans-1,4-dioxycyclohexane GPR119 agonist series. [electronic resource] by
- Han, Sangdon
- Narayanan, Sanju
- Kim, Sun Hee
- Calderon, Imelda
- Zhu, Xiuwen
- Kawasaki, Andrew
- Yue, Dawei
- Lehmann, Juerg
- Wong, Amy
- Buzard, Daniel J
- Semple, Graeme
- Carroll, Chris
- Chu, Zhi-Liang
- Al-Sharmma, Hussein
- Shu, Hsin-Hui
- Tung, Shiu-Feng
- Unett, David J
- Behan, Dominic P
- Yoon, Woo Hyun
- Morgan, Michael
- Usmani, Khawja A
- Chen, Chuan
- Sadeque, Abu
- Leonard, James N
- Jones, Robert M
Producer: 20160308
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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11.
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Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxamides as potent and selective CB2 receptor agonists. [electronic resource] by
- Han, Sangdon
- Thoresen, Lars
- Zhu, Xiuwen
- Narayanan, Sanju
- Jung, Jae-Kyu
- Strah-Pleynet, Sonja
- Decaire, Marc
- Choi, Karoline
- Xiong, Yifeng
- Yue, Dawei
- Semple, Graeme
- Thatte, Jayant
- Solomon, Michelle
- Fu, Lixia
- Whelan, Kevin
- Al-Shamma, Hussien
- Gatlin, Joel
- Chen, Ruoping
- Dang, Huong
- Pride, Cameron
- Gaidarov, Ibragim
- Unett, David J
- Behan, Dominic P
- Sadeque, Abu
- Usmani, Khawja A
- Chen, Chuan
- Edwards, Jeffrey
- Morgan, Michael
- Jones, Robert M
Producer: 20150921
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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12.
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Discovery of 2-(((1r,4r)-4-(((4-Chlorophenyl)(phenyl)carbamoyl)oxy)methyl)cyclohexyl)methoxy)acetate (Ralinepag): An Orally Active Prostacyclin Receptor Agonist for the Treatment of Pulmonary Arterial Hypertension. [electronic resource] by
- Tran, Thuy-Anh
- Kramer, Bryan
- Shin, Young-Jun
- Vallar, Pureza
- Boatman, P Douglas
- Zou, Ning
- Sage, Carleton R
- Gharbaoui, Tawfik
- Krishnan, Ashwin
- Pal, Biman
- Shakya, Sagar R
- Garrido Montalban, Antonio
- Adams, John W
- Ramirez, Juan
- Behan, Dominic P
- Shifrina, Anna
- Blackburn, Anthony
- Leakakos, Tina
- Shi, Yunqing
- Morgan, Michael
- Sadeque, Abu
- Chen, Weichao
- Unett, David J
- Gaidarov, Ibragim
- Chen, Xiaohua
- Chang, Steve
- Shu, Hsin-Hui
- Tung, Shiu-Feng
- Semple, Graeme
Producer: 20170706
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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13.
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(7-Benzyloxy-2,3-dihydro-1H-pyrrolo[1,2-a]indol-1-yl)acetic Acids as S1P1 Functional Antagonists. [electronic resource] by
- Buzard, Daniel J
- Lopez, Luis
- Moody, Jeanne
- Kawasaki, Andrew
- Schrader, Thomas O
- Kasem, Michelle
- Johnson, Ben
- Zhu, Xiuwen
- Thoresen, Lars
- Kim, Sun Hee
- Gharbaoui, Tawfik
- Sengupta, Dipanjan
- Calvano, Lorene
- Krishnan, Ashwin
- Gao, Yinghong
- Semple, Graeme
- Edwards, Jeff
- Barden, Jeremy
- Morgan, Michael
- Usmani, Khawja
- Chen, Chuan
- Sadeque, Abu
- Chen, Weichao
- Christopher, Ronald J
- Thatte, Jayant
- Fu, Lixia
- Solomon, Michelle
- Whelan, Kevin
- Al-Shamma, Hussien
- Gatlin, Joel
- Gaidarov, Ibragim
- Anthony, Todd
- Le, Minh
- Unett, David J
- Stirn, Scott
- Blackburn, Anthony
- Behan, Dominic P
- Jones, Robert M
Producer: 20141217
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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14.
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Discovery of APD334: Design of a Clinical Stage Functional Antagonist of the Sphingosine-1-phosphate-1 Receptor. [electronic resource] by
- Buzard, Daniel J
- Kim, Sun Hee
- Lopez, Luis
- Kawasaki, Andrew
- Zhu, Xiuwen
- Moody, Jeanne
- Thoresen, Lars
- Calderon, Imelda
- Ullman, Brett
- Han, Sangdon
- Lehmann, Juerg
- Gharbaoui, Tawfik
- Sengupta, Dipanjan
- Calvano, Lorene
- Montalban, Antonio Garrido
- Ma, You-An
- Sage, Carleton
- Gao, Yinghong
- Semple, Graeme
- Edwards, Jeff
- Barden, Jeremy
- Morgan, Michael
- Chen, Weichao
- Usmani, Khawja
- Chen, Chuan
- Sadeque, Abu
- Christopher, Ronald J
- Thatte, Jayant
- Fu, Lixia
- Solomon, Michelle
- Mills, David
- Whelan, Kevin
- Al-Shamma, Hussien
- Gatlin, Joel
- Le, Minh
- Gaidarov, Ibragim
- Anthony, Todd
- Unett, David J
- Blackburn, Anthony
- Rueter, Jaimie
- Stirn, Scott
- Behan, Dominic P
- Jones, Robert M
Producer: 20141217
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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