Results
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Synthesis and evaluation of potent and selective beta3 adrenergic receptor agonists containing heterobiaryl carboxylic acids. [electronic resource] by
- Shearer, Barry G
- Chao, Esther Y
- Uehling, David E
- Deaton, David N
- Cowan, Conrad
- Sherman, Bryan W
- Milliken, Tula
- Faison, Walter
- Brown, Kathleen
- Adkison, Kimberly K
- Lee, Frank
Producer: 20071121
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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3.
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Dual EGFR/ErbB-2 inhibitors from novel pyrrolidinyl-acetylenic thieno[3,2-d]pyrimidines. [electronic resource] by
- Hubbard, Robert D
- Dickerson, Scott H
- Emerson, Holly K
- Griffin, Robert J
- Reno, Michael J
- Hornberger, Keith R
- Rusnak, David W
- Wood, Edgar R
- Uehling, David E
- Waterson, Alex G
Producer: 20091229
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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4.
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Identification of RSK and TTK as Modulators of Blood Vessel Morphogenesis Using an Embryonic Stem Cell-Based Vascular Differentiation Assay. [electronic resource] by
- Hammoud, Lamis
- Adams, Jessica R
- Loch, Amanda J
- Marcellus, Richard C
- Uehling, David E
- Aman, Ahmed
- Fladd, Christopher
- McKee, Trevor D
- Jo, Christine E B
- Al-Awar, Rima
- Egan, Sean E
- Rossant, Janet
Producer: 20171121
In:
Stem cell reports vol. 7
Availability: No items available.
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5.
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Synthesis and evaluation of potent and selective beta(3) adrenergic receptor agonists containing acylsulfonamide, sulfonylsulfonamide, and sulfonylurea carboxylic acid isosteres. [electronic resource] by
- Uehling, David E
- Donaldson, Kelly H
- Deaton, David N
- Hyman, Clifton E
- Sugg, Elizabeth E
- Barrett, David G
- Hughes, Robert G
- Reitter, Barbara
- Adkison, Kim K
- Lancaster, Mary E
- Lee, Frank
- Hart, Robert
- Paulik, Mark A
- Sherman, Bryan W
- True, Timothy
- Cowan, Conrad
Producer: 20020219
In:
Journal of medicinal chemistry vol. 45
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6.
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Alkynyl pyrimidines as dual EGFR/ErbB2 kinase inhibitors. [electronic resource] by
- Waterson, Alex G
- Stevens, Kirk L
- Reno, Michael J
- Zhang, Yue-Mei
- Boros, Eric E
- Bouvier, Frederic
- Rastagar, Abdullah
- Uehling, David E
- Dickerson, Scott H
- Reep, Bryan
- McDonald, Octerloney B
- Wood, Edgar R
- Rusnak, David W
- Alligood, Krystal J
- Rudolph, Sharon K
Producer: 20060626
In:
Bioorganic & medicinal chemistry letters vol. 16
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7.
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Dabrafenib; preclinical characterization, increased efficacy when combined with trametinib, while BRAF/MEK tool combination reduced skin lesions. [electronic resource] by
- King, Alastair J
- Arnone, Marc R
- Bleam, Maureen R
- Moss, Katherine G
- Yang, Jingsong
- Fedorowicz, Kelly E
- Smitheman, Kimberly N
- Erhardt, Joseph A
- Hughes-Earle, Angela
- Kane-Carson, Laurie S
- Sinnamon, Robert H
- Qi, Hongwei
- Rheault, Tara R
- Uehling, David E
- Laquerre, Sylvie G
Producer: 20140207
In:
PloS one vol. 8
Availability: No items available.
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8.
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Development of potent B-RafV600E inhibitors containing an arylsulfonamide headgroup. [electronic resource] by
- Stellwagen, John C
- Adjabeng, George M
- Arnone, Marc R
- Dickerson, Scott H
- Han, Chao
- Hornberger, Keith R
- King, Alastair J
- Mook, Robert A
- Petrov, Kimberly G
- Rheault, Tara R
- Rominger, Cynthia M
- Rossanese, Olivia W
- Smitheman, Kimberly N
- Waterson, Alex G
- Uehling, David E
Producer: 20111122
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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9.
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Thienopyrimidine-based dual EGFR/ErbB-2 inhibitors. [electronic resource] by
- Rheault, Tara R
- Caferro, Thomas R
- Dickerson, Scott H
- Donaldson, Kelly H
- Gaul, Michael D
- Goetz, Aaron S
- Mullin, Robert J
- McDonald, Octerloney B
- Petrov, Kimberly G
- Rusnak, David W
- Shewchuk, Lisa M
- Spehar, Glenn M
- Truesdale, Anne T
- Vanderwall, Dana E
- Wood, Edgar R
- Uehling, David E
Producer: 20100706
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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10.
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Biarylaniline phenethanolamines as potent and selective beta3 adrenergic receptor agonists. [electronic resource] by
- Uehling, David E
- Shearer, Barry G
- Donaldson, Kelly H
- Chao, Esther Y
- Deaton, David N
- Adkison, Kim K
- Brown, Kathleen K
- Cariello, Neal F
- Faison, Walter L
- Lancaster, Mary E
- Lin, Jasmine
- Hart, Robert
- Milliken, Tula O
- Paulik, Mark A
- Sherman, Bryan W
- Sugg, Elizabeth E
- Cowan, Conrad
Producer: 20060606
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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11.
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Synthesis and evaluation of aniline headgroups for alkynyl thienopyrimidine dual EGFR/ErbB-2 kinase inhibitors. [electronic resource] by
- Waterson, Alex G
- Petrov, Kimberly G
- Hornberger, Keith R
- Hubbard, Robert D
- Sammond, Douglas M
- Smith, Stephon C
- Dickson, Hamilton D
- Caferro, Thomas R
- Hinkle, Kevin W
- Stevens, Kirk L
- Dickerson, Scott H
- Rusnak, David W
- Spehar, Glenn M
- Wood, Edgar R
- Griffin, Robert J
- Uehling, David E
Producer: 20090828
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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12.
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Discovery of Dabrafenib: A Selective Inhibitor of Raf Kinases with Antitumor Activity against B-Raf-Driven Tumors. [electronic resource] by
- Rheault, Tara R
- Stellwagen, John C
- Adjabeng, George M
- Hornberger, Keith R
- Petrov, Kimberly G
- Waterson, Alex G
- Dickerson, Scott H
- Mook, Robert A
- Laquerre, Sylvie G
- King, Alastair J
- Rossanese, Olivia W
- Arnone, Marc R
- Smitheman, Kimberly N
- Kane-Carson, Laurie S
- Han, Chao
- Moorthy, Ganesh S
- Moss, Katherine G
- Uehling, David E
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
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13.
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Synthesis and stereochemical effects of pyrrolidinyl-acetylenic thieno[3,2-d]pyrimidines as EGFR and ErbB-2 inhibitors. [electronic resource] by
- Stevens, Kirk L
- Alligood, Krystal J
- Alberti, Jennifer G Badiang
- Caferro, Thomas R
- Chamberlain, Stanley D
- Dickerson, Scott H
- Dickson, Hamilton D
- Emerson, Holly K
- Griffin, Robert J
- Hubbard, Robert D
- Keith, Barry R
- Mullin, Robert J
- Petrov, Kimberly G
- Gerding, Roseanne M
- Reno, Michael J
- Rheault, Tara R
- Rusnak, David W
- Sammond, Douglas M
- Smith, Stephon C
- Uehling, David E
- Waterson, Alex G
- Wood, Edgar R
Producer: 20090128
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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14.
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Discovery and optimization of imidazo[1,2-a]pyridine inhibitors of insulin-like growth factor-1 receptor (IGF-1R). [electronic resource] by
- Emmitte, Kyle A
- Wilson, Brian J
- Baum, Erich W
- Emerson, Holly K
- Kuntz, Kevin W
- Nailor, Kristen E
- Salovich, James M
- Smith, Stephon C
- Cheung, Mui
- Gerding, Roseanne M
- Stevens, Kirk L
- Uehling, David E
- Mook, Robert A
- Moorthy, Ganesh S
- Dickerson, Scott H
- Hassell, Anne M
- Leesnitzer, M Anthony
- Shewchuk, Lisa M
- Groy, Arthur
- Rowand, Jason L
- Anderson, Kelly
- Atkins, Charity L
- Yang, Jingsong
- Sabbatini, Peter
- Kumar, Rakesh
Producer: 20100706
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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15.
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6-Ethynylthieno[3,2-d]- and 6-ethynylthieno[2,3-d]pyrimidin-4-anilines as tunable covalent modifiers of ErbB kinases. [electronic resource] by
- Wood, Edgar R
- Shewchuk, Lisa M
- Ellis, Byron
- Brignola, Perry
- Brashear, Ronald L
- Caferro, Thomas R
- Dickerson, Scott H
- Dickson, Hamilton D
- Donaldson, Kelly H
- Gaul, Michael
- Griffin, Robert J
- Hassell, Anne M
- Keith, Barry
- Mullin, Robert
- Petrov, Kimberly G
- Reno, Michael J
- Rusnak, David W
- Tadepalli, Sarva M
- Ulrich, John C
- Wagner, Craig D
- Vanderwall, Dana E
- Waterson, Alex G
- Williams, Jon D
- White, Wendy L
- Uehling, David E
Producer: 20080429
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 105
Availability: No items available.
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