Results
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1.
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Identification of potent pyrazolo[4,3-h]quinazoline-3-carboxamides as multi-cyclin-dependent kinase inhibitors. [electronic resource] by
- Traquandi, Gabriella
- Ciomei, Marina
- Ballinari, Dario
- Casale, Elena
- Colombo, Nicoletta
- Croci, Valter
- Fiorentini, Francesco
- Isacchi, Antonella
- Longo, Antonio
- Mercurio, Ciro
- Panzeri, Achille
- Pastori, Wilma
- Pevarello, Paolo
- Volpi, Daniele
- Roussel, Patrick
- Vulpetti, Anna
- Brasca, Maria Gabriella
Producer: 20100401
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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2.
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Optimization of diarylthiazole B-raf inhibitors: identification of a compound endowed with high oral antitumor activity, mitigated hERG inhibition, and low paradoxical effect. [electronic resource] by
- Pulici, Maurizio
- Traquandi, Gabriella
- Marchionni, Chiara
- Modugno, Michele
- Lupi, Rosita
- Amboldi, Nadia
- Casale, Elena
- Colombo, Nicoletta
- Corti, Luca
- Fasolini, Marina
- Gasparri, Fabio
- Pastori, Wilma
- Scolaro, Alessandra
- Donati, Daniele
- Felder, Eduard
- Galvani, Arturo
- Isacchi, Antonella
- Pesenti, Enrico
- Ciomei, Marina
Producer: 20150929
In:
ChemMedChem vol. 10
Availability: No items available.
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3.
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Identification of N,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide (PHA-848125), a potent, orally available cyclin dependent kinase inhibitor. [electronic resource] by
- Brasca, Maria Gabriella
- Amboldi, Nadia
- Ballinari, Dario
- Cameron, Alexander
- Casale, Elena
- Cervi, Giovanni
- Colombo, Maristella
- Colotta, Francesco
- Croci, Valter
- D'Alessio, Roberto
- Fiorentini, Francesco
- Isacchi, Antonella
- Mercurio, Ciro
- Moretti, Walter
- Panzeri, Achille
- Pastori, Wilma
- Pevarello, Paolo
- Quartieri, Francesca
- Roletto, Fulvia
- Traquandi, Gabriella
- Vianello, Paola
- Vulpetti, Anna
- Ciomei, Marina
Producer: 20100701
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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4.
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3-Aminopyrazole inhibitors of CDK2/cyclin A as antitumor agents. 2. Lead optimization. [electronic resource] by
- Pevarello, Paolo
- Brasca, Maria Gabriella
- Orsini, Paolo
- Traquandi, Gabriella
- Longo, Antonio
- Nesi, Marcella
- Orzi, Fabrizio
- Piutti, Claudia
- Sansonna, Pietro
- Varasi, Mario
- Cameron, Alexander
- Vulpetti, Anna
- Roletto, Fulvia
- Alzani, Rachele
- Ciomei, Marina
- Albanese, Clara
- Pastori, Wilma
- Marsiglio, Aurelio
- Pesenti, Enrico
- Fiorentini, Francesco
- Bischoff, Jim R
- Mercurio, Ciro
Producer: 20050524
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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5.
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3-Aminopyrazole inhibitors of CDK2/cyclin A as antitumor agents. 1. Lead finding. [electronic resource] by
- Pevarello, Paolo
- Brasca, Maria Gabriella
- Amici, Raffaella
- Orsini, Paolo
- Traquandi, Gabriella
- Corti, Luca
- Piutti, Claudia
- Sansonna, Pietro
- Villa, Manuela
- Pierce, Betsy S
- Pulici, Maurizio
- Giordano, Patrizia
- Martina, Katia
- Fritzen, Edward L
- Nugent, Richard A
- Casale, Elena
- Cameron, Alexander
- Ciomei, Marina
- Roletto, Fulvia
- Isacchi, Antonella
- Fogliatto, GianPaolo
- Pesenti, Enrico
- Pastori, Wilma
- Marsiglio, Aurelio
- Leach, Karen L
- Clare, Paula M
- Fiorentini, Francesco
- Varasi, Mario
- Vulpetti, Anna
- Warpehoski, Martha A
Producer: 20040709
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
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