Results
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1.
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Discovery of Pyridones As Oral AMPK Direct Activators. [electronic resource] by
- Mirguet, Olivier
- Sautet, Stéphane
- Clément, Catherine-Anne
- Toum, Jérôme
- Donche, Frédéric
- Marques, Celine
- Rondet, Emilie
- Pizzonero, Mathieu
- Beaufils, Benjamin
- Dudit, Yann
- Huet, Pascal
- Trottet, Lionel
- Grondin, Pascal
- Brusq, Jean-Marie
- Boursier, Eric
- Saintillan, Yannick
- Nicodeme, Edwige
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
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2.
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From ApoA1 upregulation to BET family bromodomain inhibition: discovery of I-BET151. [electronic resource] by
- Mirguet, Olivier
- Lamotte, Yann
- Donche, Frédéric
- Toum, Jérôme
- Gellibert, Françoise
- Bouillot, Anne
- Gosmini, Romain
- Nguyen, Van-Loc
- Delannée, Delphine
- Seal, Jonathan
- Blandel, Florence
- Boullay, Anne-Bénédicte
- Boursier, Eric
- Martin, Sandrine
- Brusq, Jean-Marie
- Krysa, Gael
- Riou, Alizon
- Tellier, Rémi
- Costaz, Agnès
- Huet, Pascal
- Dudit, Yann
- Trottet, Lionel
- Kirilovsky, Jorge
- Nicodeme, Edwige
Producer: 20120918
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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3.
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Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains. [electronic resource] by
- Mirguet, Olivier
- Gosmini, Romain
- Toum, Jérôme
- Clément, Catherine A
- Barnathan, Mélanie
- Brusq, Jean-Marie
- Mordaunt, Jacqueline E
- Grimes, Richard M
- Crowe, Miriam
- Pineau, Olivier
- Ajakane, Myriam
- Daugan, Alain
- Jeffrey, Phillip
- Cutler, Leanne
- Haynes, Andrea C
- Smithers, Nicholas N
- Chung, Chun-wa
- Bamborough, Paul
- Uings, Iain J
- Lewis, Antonia
- Witherington, Jason
- Parr, Nigel
- Prinjha, Rab K
- Nicodème, Edwige
Producer: 20131223
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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4.
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The discovery of I-BET726 (GSK1324726A), a potent tetrahydroquinoline ApoA1 up-regulator and selective BET bromodomain inhibitor. [electronic resource] by
- Gosmini, Romain
- Nguyen, Van Loc
- Toum, Jérôme
- Simon, Christophe
- Brusq, Jean-Marie G
- Krysa, Gael
- Mirguet, Olivier
- Riou-Eymard, Alizon M
- Boursier, Eric V
- Trottet, Lionel
- Bamborough, Paul
- Clark, Hugh
- Chung, Chun-wa
- Cutler, Leanne
- Demont, Emmanuel H
- Kaur, Rejbinder
- Lewis, Antonia J
- Schilling, Mark B
- Soden, Peter E
- Taylor, Simon
- Walker, Ann L
- Walker, Matthew D
- Prinjha, Rab K
- Nicodème, Edwige
Producer: 20141218
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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5.
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Substituted 2-[(4-aminomethyl)phenoxy]-2-methylpropionic acid PPARalpha agonists. 1. Discovery of a novel series of potent HDLc raising agents. [electronic resource] by
- Sierra, Michael L
- Beneton, Véronique
- Boullay, Anne-Bénédict
- Boyer, Thierry
- Brewster, Andrew G
- Donche, Frédéric
- Forest, Marie-Claire
- Fouchet, Marie-Hélène
- Gellibert, Françoise J
- Grillot, Didier A
- Lambert, Millard H
- Laroze, Alain
- Le Grumelec, Christelle
- Linget, Jean Michel
- Montana, Valerie G
- Nguyen, Van-Loc
- Nicodème, Edwige
- Patel, Vipul
- Penfornis, Annie
- Pineau, Olivier
- Pohin, Danig
- Potvain, Florent
- Poulain, Géraldine
- Ruault, Cécile Bertho
- Saunders, Michael
- Toum, Jérôme
- Xu, H Eric
- Xu, Robert X
- Pianetti, Pascal M
Producer: 20070327
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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6.
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Discovery and characterization of small molecule inhibitors of the BET family bromodomains. [electronic resource] by
- Chung, Chun-Wa
- Coste, Herve
- White, Julia H
- Mirguet, Olivier
- Wilde, Jonathan
- Gosmini, Romain L
- Delves, Chris
- Magny, Sylvie M
- Woodward, Robert
- Hughes, Stephen A
- Boursier, Eric V
- Flynn, Helen
- Bouillot, Anne M
- Bamborough, Paul
- Brusq, Jean-Marie G
- Gellibert, Francoise J
- Jones, Emma J
- Riou, Alizon M
- Homes, Paul
- Martin, Sandrine L
- Uings, Iain J
- Toum, Jerome
- Clement, Catherine A
- Boullay, Anne-Benedicte
- Grimley, Rachel L
- Blandel, Florence M
- Prinjha, Rab K
- Lee, Kevin
- Kirilovsky, Jorge
- Nicodeme, Edwige
Producer: 20110817
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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