Discovery and structural characterization of a phospholamban-binding cyclic peptide and design of novel inhibitors of phospholamban. [electronic resource]
Producer: 20130924Description: 463-73 p. digitalISSN:- 1747-0285
- Amino Acid Sequence
- Animals
- Calcium -- metabolism
- Calcium-Binding Proteins -- antagonists & inhibitors
- Drug Design
- Drug Evaluation, Preclinical
- Guinea Pigs
- Heart -- drug effects
- Humans
- Models, Molecular
- Myocardium -- metabolism
- Peptide Library
- Peptides, Cyclic -- chemical synthesis
- Protein Binding
- Sarcoplasmic Reticulum Calcium-Transporting ATPases -- metabolism
- Small Molecule Libraries -- chemistry
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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