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Synthesis and structure-activity relationships of 1,2,3,4-tetrahydropyrido[2,3-b]pyrazines as potent and selective inhibitors of the anaplastic lymphoma kinase. [electronic resource] by
- Milkiewicz, Karen L
- Weinberg, Linda R
- Albom, Mark S
- Angeles, Thelma S
- Cheng, Mangeng
- Ghose, Arup K
- Roemmele, Renee C
- Theroff, Jay P
- Underiner, Ted L
- Zificsak, Craig A
- Dorsey, Bruce D
Producer: 20101014
In:
Bioorganic & medicinal chemistry vol. 18
Availability: No items available.
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4.
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Design, synthesis, and biological evaluation of sulfonyl acrylonitriles as novel inhibitors of cancer metastasis and spread. [electronic resource] by
- Shen, Yi
- Zificsak, Craig A
- Shea, Jill E
- Lao, Xuegang
- Bollt, Oana
- Li, Xiufen
- Lisko, Joseph G
- Theroff, Jay P
- Scaife, Courtney L
- Ator, Mark A
- Ruggeri, Bruce A
- Dorsey, Bruce D
- Kuwada, Scott K
Producer: 20150414
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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5.
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Methanesulfonamido-cyclohexylamine derivatives of 2,4-diaminopyrimidine as potent ALK inhibitors. [electronic resource] by
- Zificsak, Craig A
- Theroff, Jay P
- Aimone, Lisa D
- Angeles, Thelma S
- Albom, Mark S
- Cheng, Mangeng
- Mesaros, Eugen F
- Ott, Gregory R
- Quail, Matthew R
- Underiner, Ted L
- Wan, Weihua
- Dorsey, Bruce D
Producer: 20111122
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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Structure-activity relationship and pharmacokinetic profile of 5-ketopyrazole factor Xa inhibitors. [electronic resource] by
- Varnes, Jeffrey G
- Wacker, Dean A
- Pinto, Donald J P
- Orwat, Michael J
- Theroff, Jay P
- Wells, Brian
- Galemo, Robert A
- Luettgen, Joseph M
- Knabb, Robert M
- Bai, Steven
- He, Kan
- Lam, Patrick Y S
- Wexler, Ruth R
Producer: 20080527
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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Fused bicyclic derivatives of 2,4-diaminopyrimidine as c-Met inhibitors. [electronic resource] by
- Weinberg, Linda R
- Albom, Mark S
- Angeles, Thelma S
- Husten, Jean
- Lisko, Joseph G
- McHugh, Robert J
- Milkiewicz, Karen L
- Murthy, Seetha
- Ott, Gregory R
- Theroff, Jay P
- Tripathy, Rabindranath
- Underiner, Ted L
- Zificsak, Craig A
- Dorsey, Bruce D
Producer: 20110414
In:
Bioorganic & medicinal chemistry letters vol. 21
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Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor. [electronic resource] by
- Palmer, Wylie S
- Poncet-Montange, Guillaume
- Liu, Gang
- Petrocchi, Alessia
- Reyna, Naphtali
- Subramanian, Govindan
- Theroff, Jay
- Yau, Anne
- Kost-Alimova, Maria
- Bardenhagen, Jennifer P
- Leo, Elisabetta
- Shepard, Hannah E
- Tieu, Trang N
- Shi, Xi
- Zhan, Yanai
- Zhao, Shuping
- Barton, Michelle C
- Draetta, Giulio
- Toniatti, Carlo
- Jones, Philip
- Geck Do, Mary
- Andersen, Jannik N
Producer: 20160726
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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9.
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Optimization of a novel kinase inhibitor scaffold for the dual inhibition of JAK2 and FAK kinases. [electronic resource] by
- Zificsak, Craig A
- Gingrich, Diane E
- Breslin, Henry J
- Dunn, Derek D
- Milkiewicz, Karen L
- Theroff, Jay P
- Thieu, Tho V
- Underiner, Ted L
- Weinberg, Linda R
- Aimone, Lisa D
- Albom, Mark S
- Mason, Jennifer L
- Saville, Lisa
- Husten, Jean
- Angeles, Thelma S
- Finn, James P
- Jan, Mahfuza
- O'Kane, Teresa M
- Dobrzanski, Pawel
- Dorsey, Bruce D
Producer: 20120803
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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10.
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2,4-Diaminopyrimidine inhibitors of c-Met kinase bearing benzoxazepine anilines. [electronic resource] by
- Zificsak, Craig A
- Theroff, Jay P
- Aimone, Lisa D
- Albom, Mark S
- Angeles, Thelma S
- Brown, Rebecca A
- Galinis, Deborah
- Grobelny, Jennifer V
- Herbertz, Torsten
- Husten, Jean
- Kocsis, Laura S
- LoSardo, Christine
- Miknyoczki, Sheila J
- Murthy, Seetha
- Rolon-Steele, Damaris
- Underiner, Ted L
- Wells-Knecht, Kevin J
- Worrell, Candace S
- Zeigler, Kelli S
- Dorsey, Bruce D
Producer: 20110425
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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11.
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An inhibitor of oxidative phosphorylation exploits cancer vulnerability. [electronic resource] by
- Molina, Jennifer R
- Sun, Yuting
- Protopopova, Marina
- Gera, Sonal
- Bandi, Madhavi
- Bristow, Christopher
- McAfoos, Timothy
- Morlacchi, Pietro
- Ackroyd, Jeffrey
- Agip, Ahmed-Noor A
- Al-Atrash, Gheath
- Asara, John
- Bardenhagen, Jennifer
- Carrillo, Caroline C
- Carroll, Christopher
- Chang, Edward
- Ciurea, Stefan
- Cross, Jason B
- Czako, Barbara
- Deem, Angela
- Daver, Naval
- de Groot, John Frederick
- Dong, Jian-Wen
- Feng, Ningping
- Gao, Guang
- Gay, Jason
- Do, Mary Geck
- Greer, Jennifer
- Giuliani, Virginia
- Han, Jing
- Han, Lina
- Henry, Verlene K
- Hirst, Judy
- Huang, Sha
- Jiang, Yongying
- Kang, Zhijun
- Khor, Tin
- Konoplev, Sergej
- Lin, Yu-Hsi
- Liu, Gang
- Lodi, Alessia
- Lofton, Timothy
- Ma, Helen
- Mahendra, Mikhila
- Matre, Polina
- Mullinax, Robert
- Peoples, Michael
- Petrocchi, Alessia
- Rodriguez-Canale, Jaime
- Serreli, Riccardo
- Shi, Thomas
- Smith, Melinda
- Tabe, Yoko
- Theroff, Jay
- Tiziani, Stefano
- Xu, Quanyun
- Zhang, Qi
- Muller, Florian
- DePinho, Ronald A
- Toniatti, Carlo
- Draetta, Giulio F
- Heffernan, Timothy P
- Konopleva, Marina
- Jones, Philip
- Di Francesco, M Emilia
- Marszalek, Joseph R
Producer: 20190510
In:
Nature medicine vol. 24
Availability: No items available.
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