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SAR studies of 6-(arylamino)-4,4-disubstituted-1-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-ones as progesterone receptor antagonists. [electronic resource] by
- Kern, Jeffrey C
- Terefenko, Eugene A
- Fensome, Andrew
- Unwallla, Ray
- Wrobel, Jay
- Zhu, Yuan
- Cohen, Jeffrey
- Winneker, Richard
- Zhang, Zhiming
- Zhang, Puwen
Producer: 20070424
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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6.
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Synthesis and activity of novel 1- or 3-(3-amino-1-phenyl propyl)-1,3-dihydro-2H-benzimidazol-2-ones as selective norepinephrine reuptake inhibitors. [electronic resource] by
- Zhang, Puwen
- Terefenko, Eugene A
- McComas, Casey C
- Mahaney, Paige E
- Vu, An
- Trybulski, Eugene
- Koury, Elizabeth
- Johnston, Grace
- Bray, Jenifer
- Deecher, Darlene
Producer: 20090109
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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7.
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7-aryl 1,5-dihydro-benzo[e][1,4]oxazepin-2-ones and analogs as non-steroidal progesterone receptor antagonists. [electronic resource] by
- Zhang, Puwen
- Kern, Jeffrey C
- Terefenko, Eugene A
- Fensome, Andrew
- Unwalla, Ray
- Zhang, Zhiming
- Cohen, Jeffrey
- Berrodin, Thomas J
- Yudt, Matthew R
- Winneker, Richard C
- Wrobel, Jay
Producer: 20080805
In:
Bioorganic & medicinal chemistry vol. 16
Availability: No items available.
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8.
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1,5-Dihydro-benzo[e][1,4]oxazepin-2(1H)-ones containing a 7-(5'-cyanopyrrol-2-yl) group as nonsteroidal progesterone receptor modulators. [electronic resource] by
- Kern, Jeffrey C
- Terefenko, Eugene A
- Fensome, Andrew
- Unwalla, Ray
- Wrobel, Jay
- Cohen, Jeffrey
- Zhu, Yuan
- Berrodin, Thomas J
- Yudt, Matthew R
- Winneker, Richard C
- Zhang, Zhiming
- Zhang, Puwen
Producer: 20081014
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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9.
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3-(Arylamino)-3-phenylpropan-2-olamines as a new series of dual norepinephrine and serotonin reuptake inhibitors. [electronic resource] by
- Vu, An T
- Cohn, Stephen T
- Terefenko, Eugene A
- Moore, William J
- Zhang, Puwen
- Mahaney, Paige E
- Trybulski, Eugene J
- Goljer, Igor
- Dooley, Rebecca
- Bray, Jenifer A
- Johnston, Grace H
- Leiter, Jennifer
- Deecher, Darlene C
Producer: 20090821
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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10.
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1- or 3-(3-Amino-2-hydroxy-1-phenyl propyl)-1,3-dihydro-2H-benzimidazol-2-ones: potent, selective, and orally efficacious norepinephrine reuptake inhibitors. [electronic resource] by
- Zhang, Puwen
- Terefenko, Eugene A
- Bray, Jenifer
- Deecher, Darlene
- Fensome, Andrew
- Harrison, Jim
- Kim, Callain
- Koury, Elizabeth
- Mark, Lilly
- McComas, Casey C
- Mugford, Cheryl A
- Trybulski, Eugene J
- Vu, An T
- Whiteside, Garth T
- Mahaney, Paige E
Producer: 20091014
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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11.
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Structure-activity relationships of the 1-amino-3-(1H-indol-1-yl)-3-phenylpropan-2-ol series of monoamine reuptake inhibitors. [electronic resource] by
- Mahaney, Paige E
- Kim, Callain Y
- Coghlan, Richard D
- Cohn, Stephen T
- Heffernan, Gavin D
- Huselton, Christine A
- Terefenko, Eugene A
- Vu, An T
- Zhang, Puwen
- Burroughs, Kevin D
- Cosmi, Scott A
- Bray, Jenifer A
- Johnston, Grace H
- Deecher, Darlene C
- Trybulski, Eugene J
Producer: 20091130
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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12.
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Synthesis and structure-activity relationship of novel 6-aryl-1,4-dihydrobenzo[d][1,3]oxazine-2-thiones as progesterone receptor modulators leading to the potent and selective nonsteroidal progesterone receptor agonist tanaproget. [electronic resource] by
- Fensome, Andrew
- Bender, Reinhold
- Chopra, Rajiv
- Cohen, Jeff
- Collins, Mark A
- Hudak, Valerie
- Malakian, Karl
- Lockhead, Susan
- Olland, Andrea
- Svenson, Kristine
- Terefenko, Eugene A
- Unwalla, Ray J
- Wilhelm, James M
- Wolfrom, Scott
- Zhu, Yuan
- Zhang, Zhiming
- Zhang, Puwen
- Winneker, Richard C
- Wrobel, Jay
Producer: 20050927
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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13.
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Discovery of novel selective norepinephrine inhibitors: 1-(2-morpholin-2-ylethyl)-3-aryl-1,3-dihydro-2,1,3-benzothiadiazole 2,2-dioxides (WYE-114152). [electronic resource] by
- O'Neill, David J
- Adedoyin, Adedayo
- Bray, Jenifer A
- Deecher, Darlene C
- Fensome, Andrew
- Goldberg, Joel A
- Harrison, Jim
- Leventhal, Liza
- Mann, Charles
- Mark, Lilly
- Nogle, Lisa
- Sullivan, Nicole R
- Spangler, Taylor B
- Terefenko, Eugene A
- Trybulski, Eugene J
- Uveges, Albert J
- Vu, An
- Whiteside, Garth T
- Zhang, Puwen
Producer: 20111212
In:
Journal of medicinal chemistry vol. 54
Availability: No items available.
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