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Solid-phase synthesis and structure-activity relationships of novel biarylethers as melanin-concentrating hormone receptor-1 antagonists. [electronic resource] by
- Ma, Vu
- Bannon, Anthony W
- Baumgartner, Jamie
- Hale, Clarence
- Hsieh, Faye
- Hulme, Christopher
- Rorrer, Kirk
- Salon, John
- van Staden, Carlo
- Tempest, Paul
Producer: 20061102
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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Design of novel histone deacetylase inhibitors. [electronic resource] by
- Siliphaivanh, Phieng
- Harrington, Paul
- Witter, David J
- Otte, Karin
- Tempest, Paul
- Kattar, Sam
- Kral, Astrid M
- Fleming, Judith C
- Deshmukh, Sujal V
- Harsch, Andreas
- Secrist, Paul J
- Miller, Thomas A
Producer: 20071121
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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5.
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Use of molecular modeling aided design to dial out hERG liability in adenosine A(2A) receptor antagonists. [electronic resource] by
- Deng, Qiaolin
- Lim, Yeon-Hee
- Anand, Rajan
- Yu, Younong
- Kim, Jae-hun
- Zhou, Wei
- Zheng, Junying
- Tempest, Paul
- Levorse, Dorothy
- Zhang, Xiaoping
- Greene, Scott
- Mullins, Deborra
- Culberson, Chris
- Sherborne, Brad
- Parker, Eric M
- Stamford, Andrew
- Ali, Amjad
Producer: 20160308
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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Thiophene carboxamide inhibitors of JAK2 as potential treatments for myleoproliferative neoplasms. [electronic resource] by
- Haidle, Andrew M
- Zabierek, Anna A
- Childers, Kaleen K
- Rosenstein, Craig
- Mathur, Anjili
- Altman, Michael D
- Chan, Grace
- Xu, Lin
- Bachman, Eric
- Mo, Jan-Rung
- Bouthillette, Melaney
- Rush, Thomas
- Tempest, Paul
- Marshall, C Gary
- Young, Jonathan R
Producer: 20141020
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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Parallel medicinal chemistry approaches to selective HDAC1/HDAC2 inhibitor (SHI-1:2) optimization. [electronic resource] by
- Kattar, Solomon D
- Surdi, Laura M
- Zabierek, Anna
- Methot, Joey L
- Middleton, Richard E
- Hughes, Bethany
- Szewczak, Alexander A
- Dahlberg, William K
- Kral, Astrid M
- Ozerova, Nicole
- Fleming, Judith C
- Wang, Hongmei
- Secrist, Paul
- Harsch, Andreas
- Hamill, Julie E
- Cruz, Jonathan C
- Kenific, Candia M
- Chenard, Melissa
- Miller, Thomas A
- Berk, Scott C
- Tempest, Paul
Producer: 20090310
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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Evolution of a highly selective and potent 2-(pyridin-2-yl)-1,3,5-triazine Tie-2 kinase inhibitor. [electronic resource] by
- Hodous, Brian L
- Geuns-Meyer, Stephanie D
- Hughes, Paul E
- Albrecht, Brian K
- Bellon, Steve
- Bready, James
- Caenepeel, Sean
- Cee, Victor J
- Chaffee, Stuart C
- Coxon, Angela
- Emery, Maurice
- Fretland, Jenne
- Gallant, Paul
- Gu, Yan
- Hoffman, Doug
- Johnson, Rebecca E
- Kendall, Richard
- Kim, Joseph L
- Long, Alexander M
- Morrison, Michael
- Olivieri, Philip R
- Patel, Vinod F
- Polverino, Anthony
- Rose, Paul
- Tempest, Paul
- Wang, Ling
- Whittington, Douglas A
- Zhao, Huilin
Producer: 20070327
In:
Journal of medicinal chemistry vol. 50
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Lead optimization of 4,4-biaryl piperidine amides as γ-secretase inhibitors. [electronic resource] by
- Close, Joshua
- Heidebrecht, Richard
- Hendrix, John
- Li, Chaomin
- Munoz, Ben
- Surdi, Laura
- Kattar, Solomon
- Tempest, Paul
- Moses, Paul
- Geng, Xiaoliu
- Hughes, Bethany
- Smotrov, Nadya
- Moxham, Chris
- Chapnick, Jennifer
- Kariv, Ilona
- Nikov, George
- Burke, Julie Elizabeth
- Deshmukh, Sujal
- Jeliazkova-Mecheva, Valentina
- Leach, John Kevin
- Diaz, Damaris
- Xu, Lin
- Yang, Ziping
- Kwei, Gloria
- Moy, Lily
- Shah, Sanjiv
- Tanga, Flobert
- Kenefic, Candia
- Savage, Dan
- Shearman, Mark
- Ball, Richard G
- McNevin, Michael J
- Markarewicz, Amanda
- Miller, Thomas
Producer: 20121011
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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