Results
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[3H]A-81988, a potent, selective, competitive antagonist radioligand for angiotensin AT1 receptors. [electronic resource] by
- Hancock, A A
- Surber, B W
- Rotert, G
- Thomas, S
- Tasker, A S
- Sorensen, B K
- Vodenlich, A D
- Opgenorth, T J
- Kerkman, D J
- DeBernardis, J F
Producer: 19940712
In:
European journal of pharmacology vol. 267
Availability: No items available.
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4.
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Discovery of a series of cyclohexylethylamine-containing protein farnesyltransferase inhibitors exhibiting potent cellular activity. [electronic resource] by
- Henry, K J
- Wasicak, J
- Tasker, A S
- Cohen, J
- Ewing, P
- Mitten, M
- Larsen, J J
- Kalvin, D M
- Swenson, R
- Ng, S C
- Saeed, B
- Cherian, S
- Sham, H
- Rosenberg, S H
Producer: 19991217
In:
Journal of medicinal chemistry vol. 42
Availability: No items available.
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5.
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Pyrrolidine-3-carboxylic acids as endothelin antagonists. 4. Side chain conformational restriction leads to ET(B) selectivity. [electronic resource] by
- von Geldern, T W
- Tasker, A S
- Sorensen, B K
- Winn, M
- Szczepankiewicz, B G
- Dixon, D B
- Chiou, W J
- Wang, L
- Wessale, J L
- Adler, A
- Marsh, K C
- Nguyen, B
- Opgenorth, T J
Producer: 19991014
In:
Journal of medicinal chemistry vol. 42
Availability: No items available.
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6.
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Potent and selective non-benzodioxole-containing endothelin-A receptor antagonists. [electronic resource] by
- Tasker, A S
- Sorensen, B K
- Jae, H S
- Winn, M
- von Geldern, T W
- Dixon, D B
- Chiou, W J
- Dayton, B D
- Calzadila, S
- Hernandez, L
- Marsh, K C
- WuWong, J R
- Opgenorth, T J
Producer: 19970313
In:
Journal of medicinal chemistry vol. 40
Availability: No items available.
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7.
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Discovery of a series of pyrrolidine-based endothelin receptor antagonists with enhanced ET(A) receptor selectivity. [electronic resource] by
- Boyd, S A
- Mantei, R A
- Tasker, A S
- Liu, G
- Sorensen, B K
- Henry, K J
- von Geldern, T W
- Winn, M
- Wu-Wong, J R
- Chiou, W J
- Dixon, D B
- Hutchins, C W
- Marsh, K C
- Nguyen, B
- Opgenorth, T J
Producer: 19990909
In:
Bioorganic & medicinal chemistry vol. 7
Availability: No items available.
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8.
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2,4-Diarylpyrrolidine-3-carboxylic acids--potent ETA selective endothelin receptor antagonists. 1. Discovery of A-127722. [electronic resource] by
- Winn, M
- von Geldern, T W
- Opgenorth, T J
- Jae, H S
- Tasker, A S
- Boyd, S A
- Kester, J A
- Mantei, R A
- Bal, R
- Sorensen, B K
- Wu-Wong, J R
- Chiou, W J
- Dixon, D B
- Novosad, E I
- Hernandez, L
- Marsh, K C
Producer: 19960815
In:
Journal of medicinal chemistry vol. 39
Availability: No items available.
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9.
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Second-generation peptidomimetic inhibitors of protein farnesyltransferase demonstrating improved cellular potency and significant in vivo efficacy. [electronic resource] by
- O'Connor, S J
- Barr, K J
- Wang, L
- Sorensen, B K
- Tasker, A S
- Sham, H
- Ng, S C
- Cohen, J
- Devine, E
- Cherian, S
- Saeed, B
- Zhang, H
- Lee, J Y
- Warner, R
- Tahir, S
- Kovar, P
- Ewing, P
- Alder, J
- Mitten, M
- Leal, J
- Marsh, K
- Bauch, J
- Hoffman, D J
- Sebti, S M
- Rosenberg, S H
Producer: 19991014
In:
Journal of medicinal chemistry vol. 42
Availability: No items available.
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10.
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New antimitotic agents with activity in multi-drug-resistant cell lines and in vivo efficacy in murine tumor models. [electronic resource] by
- Szczepankiewicz, B G
- Liu, G
- Jae, H S
- Tasker, A S
- Gunawardana, I W
- von Geldern, T W
- Gwaltney, S L
- Wu-Wong, J R
- Gehrke, L
- Chiou, W J
- Credo, R B
- Alder, J D
- Nukkala, M A
- Zielinski, N A
- Jarvis, K
- Mollison, K W
- Frost, D J
- Bauch, J L
- Hui, Y H
- Claiborne, A K
- Li, Q
- Rosenberg, S H
Producer: 20020107
In:
Journal of medicinal chemistry vol. 44
Availability: No items available.
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