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Discovery of a Dual PRMT5-PRMT7 Inhibitor. [electronic resource] by
- Smil, David
- Eram, Mohammad S
- Li, Fengling
- Kennedy, Steven
- Szewczyk, Magdalena M
- Brown, Peter J
- Barsyte-Lovejoy, Dalia
- Arrowsmith, Cheryl H
- Vedadi, Masoud
- Schapira, Matthieu
Producer: 20150420
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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9.
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Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening. [electronic resource] by
- Ferreira de Freitas, Renato
- Eram, Mohammad S
- Smil, David
- Szewczyk, Magdalena M
- Kennedy, Steven
- Brown, Peter J
- Santhakumar, Vijayaratnam
- Barsyte-Lovejoy, Dalia
- Arrowsmith, Cheryl H
- Vedadi, Masoud
- Schapira, Matthieu
Producer: 20170609
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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10.
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Correction to Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening. [electronic resource] by
- Ferreira de Freitas, Renato
- Eram, Mohammad S
- Smil, David
- Szewczyk, Magdalena M
- Kennedy, Steven
- Brown, Peter J
- Santhakumar, Vijayaratnam
- Barsyte-Lovejoy, Dalia
- Arrowsmith, Cheryl H
- Vedadi, Masoud
- Schapira, Matthieu
Publication details: Journal of medicinal chemistry 08 2016
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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11.
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Sialidase down-regulation reduces non-HDL cholesterol, inhibits leukocyte transmigration, and attenuates atherosclerosis in ApoE knockout mice. [electronic resource] by
- White, Elizabeth J
- Gyulay, Gabriel
- Lhoták, Šárka
- Szewczyk, Magdalena M
- Chong, Taryne
- Fuller, Mark T
- Dadoo, Omid
- Fox-Robichaud, Alison E
- Austin, Richard C
- Trigatti, Bernardo L
- Igdoura, Suleiman A
Producer: 20190405
In:
The Journal of biological chemistry vol. 293
Availability: No items available.
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12.
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Characterization of inv(3) cell line OCI-AML-20 with stroma-dependent CD34 expression. [electronic resource] by
- Luciani, Genna M
- Xie, Lihua
- Dilworth, David
- Tierens, Anne
- Moskovitz, Yoni
- Murison, Alex
- Szewczyk, Magdalena M
- Mitchell, Amanda
- Lupien, Mathieu
- Shlush, Liran
- Dick, John E
- Arrowsmith, Cheryl H
- Barsyte-Lovejoy, Dalia
- Minden, Mark D
Producer: 20190326
In:
Experimental hematology vol. 69
Availability: No items available.
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13.
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Discovery of a Potent, Selective, and Cell-Active Dual Inhibitor of Protein Arginine Methyltransferase 4 and Protein Arginine Methyltransferase 6. [electronic resource] by
- Shen, Yudao
- Szewczyk, Magdalena M
- Eram, Mohammad S
- Smil, David
- Kaniskan, H Ümit
- de Freitas, Renato Ferreira
- Senisterra, Guillermo
- Li, Fengling
- Schapira, Matthieu
- Brown, Peter J
- Arrowsmith, Cheryl H
- Barsyte-Lovejoy, Dalia
- Liu, Jing
- Vedadi, Masoud
- Jin, Jian
Producer: 20170619
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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14.
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Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors. [electronic resource] by
- Dahlin, Jayme L
- Nelson, Kathryn M
- Strasser, Jessica M
- Barsyte-Lovejoy, Dalia
- Szewczyk, Magdalena M
- Organ, Shawna
- Cuellar, Matthew
- Singh, Gurpreet
- Shrimp, Jonathan H
- Nguyen, Nghi
- Meier, Jordan L
- Arrowsmith, Cheryl H
- Brown, Peter J
- Baell, Jonathan B
- Walters, Michael A
Producer: 20181001
In:
Nature communications vol. 8
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Discovery of a Potent Class I Protein Arginine Methyltransferase Fragment Inhibitor. [electronic resource] by
- Ferreira de Freitas, Renato
- Eram, Mohammad S
- Szewczyk, Magdalena M
- Steuber, Holger
- Smil, David
- Wu, Hong
- Li, Fengling
- Senisterra, Guillermo
- Dong, Aiping
- Brown, Peter J
- Hitchcock, Marion
- Moosmayer, Dieter
- Stegmann, Christian M
- Egner, Ursula
- Arrowsmith, Cheryl
- Barsyte-Lovejoy, Dalia
- Vedadi, Masoud
- Schapira, Matthieu
Producer: 20160712
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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16.
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LLY-283, a Potent and Selective Inhibitor of Arginine Methyltransferase 5, PRMT5, with Antitumor Activity. [electronic resource] by
- Bonday, Zahid Q
- Cortez, Guillermo S
- Grogan, Michael J
- Antonysamy, Stephen
- Weichert, Ken
- Bocchinfuso, Wayne P
- Li, Fengling
- Kennedy, Steven
- Li, Binghui
- Mader, Mary M
- Arrowsmith, Cheryl H
- Brown, Peter J
- Eram, Mohammad S
- Szewczyk, Magdalena M
- Barsyte-Lovejoy, Dalia
- Vedadi, Masoud
- Guccione, Ernesto
- Campbell, Robert M
Publication details: ACS medicinal chemistry letters Jul 2018
In:
ACS medicinal chemistry letters vol. 9
Availability: No items available.
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17.
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TP-064, a potent and selective small molecule inhibitor of PRMT4 for multiple myeloma. [electronic resource] by
- Nakayama, Kazuhide
- Szewczyk, Magdalena M
- Dela Sena, Carlo
- Wu, Hong
- Dong, Aiping
- Zeng, Hong
- Li, Fengling
- de Freitas, Renato Ferreira
- Eram, Mohammad S
- Schapira, Matthieu
- Baba, Yuji
- Kunitomo, Mihoko
- Cary, Douglas R
- Tawada, Michiko
- Ohashi, Akihiro
- Imaeda, Yasuhiro
- Saikatendu, Kumar Singh
- Grimshaw, Charles E
- Vedadi, Masoud
- Arrowsmith, Cheryl H
- Barsyte-Lovejoy, Dalia
- Kiba, Atsushi
- Tomita, Daisuke
- Brown, Peter J
Publication details: Oncotarget Apr 2018
In:
Oncotarget vol. 9
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18.
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Discovery of Potent and Selective Allosteric Inhibitors of Protein Arginine Methyltransferase 3 (PRMT3). [electronic resource] by
- Kaniskan, H Ümit
- Eram, Mohammad S
- Zhao, Kehao
- Szewczyk, Magdalena M
- Yang, Xiaobao
- Schmidt, Keith
- Luo, Xiao
- Xiao, Sean
- Dai, Miao
- He, Feng
- Zang, Irene
- Lin, Ying
- Li, Fengling
- Dobrovetsky, Elena
- Smil, David
- Min, Sun-Joon
- Lin-Jones, Jennifer
- Schapira, Matthieu
- Atadja, Peter
- Li, En
- Barsyte-Lovejoy, Dalia
- Arrowsmith, Cheryl H
- Brown, Peter J
- Liu, Feng
- Yu, Zhengtian
- Vedadi, Masoud
- Jin, Jian
Producer: 20190218
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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19.
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A potent, selective and cell-active allosteric inhibitor of protein arginine methyltransferase 3 (PRMT3). [electronic resource] by
- Kaniskan, H Ümit
- Szewczyk, Magdalena M
- Yu, Zhengtian
- Eram, Mohammad S
- Yang, Xiaobao
- Schmidt, Keith
- Luo, Xiao
- Dai, Miao
- He, Feng
- Zang, Irene
- Lin, Ying
- Kennedy, Steven
- Li, Fengling
- Dobrovetsky, Elena
- Dong, Aiping
- Smil, David
- Min, Sun-Joon
- Landon, Melissa
- Lin-Jones, Jennifer
- Huang, Xi-Ping
- Roth, Bryan L
- Schapira, Matthieu
- Atadja, Peter
- Barsyte-Lovejoy, Dalia
- Arrowsmith, Cheryl H
- Brown, Peter J
- Zhao, Kehao
- Jin, Jian
- Vedadi, Masoud
Producer: 20160112
In:
Angewandte Chemie (International ed. in English) vol. 54
Availability: No items available.
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20.
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Discovery of a chemical probe for PRDM9. [electronic resource] by
- Allali-Hassani, Abdellah
- Szewczyk, Magdalena M
- Ivanochko, Danton
- Organ, Shawna L
- Bok, Jabez
- Ho, Jessica Sook Yuin
- Gay, Florence P H
- Li, Fengling
- Blazer, Levi
- Eram, Mohammad S
- Halabelian, Levon
- Dilworth, David
- Luciani, Genna M
- Lima-Fernandes, Evelyne
- Wu, Qin
- Loppnau, Peter
- Palmer, Nathan
- Talib, S Zakiah A
- Brown, Peter J
- Schapira, Matthieu
- Kaldis, Philipp
- O'Hagan, Ronan C
- Guccione, Ernesto
- Barsyte-Lovejoy, Dalia
- Arrowsmith, Cheryl H
- Sanders, John M
- Kattar, Solomon D
- Bennett, D Jonathan
- Nicholson, Benjamin
- Vedadi, Masoud
Producer: 20200406
In:
Nature communications vol. 10
Availability: No items available.
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