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Discovery of Small Molecule RIP1 Kinase Inhibitors for the Treatment of Pathologies Associated with Necroptosis. [electronic resource] by
- Harris, Philip A
- Bandyopadhyay, Deepak
- Berger, Scott B
- Campobasso, Nino
- Capriotti, Carol A
- Cox, Julie A
- Dare, Lauren
- Finger, Joshua N
- Hoffman, Sandra J
- Kahler, Kirsten M
- Lehr, Ruth
- Lich, John D
- Nagilla, Rakesh
- Nolte, Robert T
- Ouellette, Michael T
- Pao, Christina S
- Schaeffer, Michelle C
- Smallwood, Angela
- Sun, Helen H
- Swift, Barbara A
- Totoritis, Rachel D
- Ward, Paris
- Marquis, Robert W
- Bertin, John
- Gough, Peter J
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 4
Availability: No items available.
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DNA-Encoded Library Screening Identifies Benzo[b][1,4]oxazepin-4-ones as Highly Potent and Monoselective Receptor Interacting Protein 1 Kinase Inhibitors. [electronic resource] by
- Harris, Philip A
- King, Bryan W
- Bandyopadhyay, Deepak
- Berger, Scott B
- Campobasso, Nino
- Capriotti, Carol A
- Cox, Julie A
- Dare, Lauren
- Dong, Xiaoyang
- Finger, Joshua N
- Grady, LaShadric C
- Hoffman, Sandra J
- Jeong, Jae U
- Kang, James
- Kasparcova, Viera
- Lakdawala, Ami S
- Lehr, Ruth
- McNulty, Dean E
- Nagilla, Rakesh
- Ouellette, Michael T
- Pao, Christina S
- Rendina, Alan R
- Schaeffer, Michelle C
- Summerfield, Jennifer D
- Swift, Barbara A
- Totoritis, Rachel D
- Ward, Paris
- Zhang, Aming
- Zhang, Daohua
- Marquis, Robert W
- Bertin, John
- Gough, Peter J
Producer: 20160816
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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The Identification and Pharmacological Characterization of 6-(tert-Butylsulfonyl)-N-(5-fluoro-1H-indazol-3-yl)quinolin-4-amine (GSK583), a Highly Potent and Selective Inhibitor of RIP2 Kinase. [electronic resource] by
- Haile, Pamela A
- Votta, Bartholomew J
- Marquis, Robert W
- Bury, Michael J
- Mehlmann, John F
- Singhaus, Robert
- Charnley, Adam K
- Lakdawala, Ami S
- Convery, Máire A
- Lipshutz, David B
- Desai, Biva M
- Swift, Barbara
- Capriotti, Carol A
- Berger, Scott B
- Mahajan, Mukesh K
- Reilly, Michael A
- Rivera, Elizabeth J
- Sun, Helen H
- Nagilla, Rakesh
- Beal, Allison M
- Finger, Joshua N
- Cook, Michael N
- King, Bryan W
- Ouellette, Michael T
- Totoritis, Rachel D
- Pierdomenico, Maria
- Negroni, Anna
- Stronati, Laura
- Cucchiara, Salvatore
- Ziółkowski, Bartłomiej
- Vossenkämper, Anna
- MacDonald, Thomas T
- Gough, Peter J
- Bertin, John
- Casillas, Linda N
Producer: 20170529
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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5.
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Identification of Quinoline-Based RIP2 Kinase Inhibitors with an Improved Therapeutic Index to the hERG Ion Channel. [electronic resource] by
- Haile, Pamela A
- Casillas, Linda N
- Bury, Michael J
- Mehlmann, John F
- Singhaus, Robert
- Charnley, Adam K
- Hughes, Terry V
- DeMartino, Michael P
- Wang, Gren Z
- Romano, Joseph J
- Dong, Xiaoyang
- Plotnikov, Nikolay V
- Lakdawala, Ami S
- Convery, Maire A
- Votta, Bartholomew J
- Lipshutz, David B
- Desai, Biva M
- Swift, Barbara
- Capriotti, Carol A
- Berger, Scott B
- Mahajan, Mukesh K
- Reilly, Michael A
- Rivera, Elizabeth J
- Sun, Helen H
- Nagilla, Rakesh
- LePage, Carol
- Ouellette, Michael T
- Totoritis, Rachel D
- Donovan, Brian T
- Brown, Barry S
- Chaudhary, Khuram W
- Gough, Peter J
- Bertin, John
- Marquis, Robert W
Publication details: ACS medicinal chemistry letters Oct 2018
In:
ACS medicinal chemistry letters vol. 9
Availability: No items available.
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6.
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Discovery of a First-in-Class Receptor Interacting Protein 1 (RIP1) Kinase Specific Clinical Candidate (GSK2982772) for the Treatment of Inflammatory Diseases. [electronic resource] by
- Harris, Philip A
- Berger, Scott B
- Jeong, Jae U
- Nagilla, Rakesh
- Bandyopadhyay, Deepak
- Campobasso, Nino
- Capriotti, Carol A
- Cox, Julie A
- Dare, Lauren
- Dong, Xiaoyang
- Eidam, Patrick M
- Finger, Joshua N
- Hoffman, Sandra J
- Kang, James
- Kasparcova, Viera
- King, Bryan W
- Lehr, Ruth
- Lan, Yunfeng
- Leister, Lara K
- Lich, John D
- MacDonald, Thomas T
- Miller, Nathan A
- Ouellette, Michael T
- Pao, Christina S
- Rahman, Attiq
- Reilly, Michael A
- Rendina, Alan R
- Rivera, Elizabeth J
- Schaeffer, Michelle C
- Sehon, Clark A
- Singhaus, Robert R
- Sun, Helen H
- Swift, Barbara A
- Totoritis, Rachel D
- Vossenkämper, Anna
- Ward, Paris
- Wisnoski, David D
- Zhang, Daohua
- Marquis, Robert W
- Gough, Peter J
- Bertin, John
Producer: 20170616
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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