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Establishment of a secondary screening assay for P/Q-type calcium channel blockers. [electronic resource] by
- Hermann, David
- Mezler, Mario
- Swensen, Andrew M
- Bruehl, Claus
- Obergrußerger, Ali
- Wicke, Karsten
- Schoemaker, Hans
- Gross, Gerhard
- Draguhn, Andreas
- Nimmrich, Volker
Producer: 20131118
In:
Combinatorial chemistry & high throughput screening vol. 16
Availability: No items available.
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Development and validation of a fluorescence-based HTS assay for the identification of P/Q-type calcium channel blockers. [electronic resource] by
- Mezler, Mario
- Hermann, David
- Swensen, Andrew M
- Draguhn, Andreas
- Terstappen, Georg C
- Gross, Gerhard
- Schoemaker, Hans
- Freiberg, Gail
- Pratt, Steve
- Gopalakrishnan, Sujatha M
- Nimmrich, Volker
Producer: 20120813
In:
Combinatorial chemistry & high throughput screening vol. 15
Availability: No items available.
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9.
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A high-capacity membrane potential FRET-based assay for the sodium-coupled glucose co-transporter SGLT1. [electronic resource] by
- Weinglass, Adam B
- Swensen, Andrew M
- Liu, Jessica
- Schmalhofer, William
- Thomas, Anu
- Williams, Brande
- Ross, Leila
- Hashizume, Kristina
- Kohler, Martin
- Kaczorowski, Gregory J
- Garcia, Maria L
Producer: 20080709
In:
Assay and drug development technologies vol. 6
Availability: No items available.
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10.
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An automated electrophysiological assay for differentiating Ca(v)2.2 inhibitors based on state dependence and kinetics. [electronic resource] by
- Swensen, Andrew M
- Niforatos, Wende
- Vortherms, Timothy A
- Perner, Richard J
- Li, Tao
- Schrimpf, Michael R
- Scott, Victoria E
- Lee, Lance
- Jarvis, Michael F
- McGaraughty, Steve
Producer: 20130516
In:
Assay and drug development technologies vol. 10
Availability: No items available.
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11.
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A high-throughput assay for evaluating state dependence and subtype selectivity of Cav2 calcium channel inhibitors. [electronic resource] by
- Dai, Ge
- Haedo, Rodolfo J
- Warren, Vivien A
- Ratliff, Kevin S
- Bugianesi, Randal M
- Rush, Alison
- Williams, Mark E
- Herrington, James
- Smith, McHardy M
- McManus, Owen B
- Swensen, Andrew M
Producer: 20080709
In:
Assay and drug development technologies vol. 6
Availability: No items available.
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Discovery of 4-[(2R,4R)-4-({[1-(2,2-Difluoro-1,3-benzodioxol-5-yl)cyclopropyl]carbonyl}amino)-7-(difluoromethoxy)-3,4-dihydro-2H-chromen-2-yl]benzoic Acid (ABBV/GLPG-2222), a Potent Cystic Fibrosis Transmembrane Conductance Regulator (CFTR) Corrector for the Treatment of Cystic Fibrosis. [electronic resource] by
- Wang, Xueqing
- Liu, Bo
- Searle, Xenia
- Yeung, Clinton
- Bogdan, Andrew
- Greszler, Stephen
- Singh, Ashvani
- Fan, Yihong
- Swensen, Andrew M
- Vortherms, Timothy
- Balut, Corina
- Jia, Ying
- Desino, Kelly
- Gao, Wenqing
- Yong, Hong
- Tse, Chris
- Kym, Philip
Producer: 20190415
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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Identification and Characterization of Novel CFTR Potentiators. [electronic resource] by
- Gees, Maarten
- Musch, Sara
- Van der Plas, Steven
- Wesse, Anne-Sophie
- Vandevelde, Ann
- Verdonck, Katleen
- Mammoliti, Oscar
- Hwang, Tzyh-Chang
- Sonck, Kathleen
- Stouten, Pieter
- Swensen, Andrew M
- Jans, Mia
- Van der Schueren, Jan
- Nelles, Luc
- Andrews, Martin
- Conrath, Katja
Publication details: Frontiers in pharmacology 2018
In:
Frontiers in pharmacology vol. 9
Availability: No items available.
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14.
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Comparative analysis of inactivated-state block of N-type (Ca(v)2.2) calcium channels. [electronic resource] by
- Vortherms, Timothy A
- Swensen, Andrew M
- Niforatos, Wende
- Limberis, James T
- Neelands, Torben R
- Janis, Richard S
- Thimmapaya, Rama
- Donnelly-Roberts, Diana L
- Namovic, Marian T
- Zhang, Di
- Brent Putman, C
- Martin, Ruth L
- Surowy, Carol S
- Jarvis, Michael F
- Scott, Victoria E
Producer: 20111011
In:
Inflammation research : official journal of the European Histamine Research Society ... [et al.] vol. 60
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Synthesis and SAR of 4-aminocyclopentapyrrolidines as orally active N-type calcium channel inhibitors for inflammatory and neuropathic pain. [electronic resource] by
- Beebe, Xenia
- Yeung, Clinton M
- Darczak, Daria
- Shekhar, Shashank
- Vortherms, Timothy A
- Miller, Loan
- Milicic, Ivan
- Swensen, Andrew M
- Zhu, Chang Z
- Banfor, Patricia
- Wetter, Jill M
- Marsh, Kennan C
- Jarvis, Michael F
- Scott, Victoria E
- Schrimpf, Michael R
- Lee, Chih-Hung
Producer: 20140415
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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16.
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Characterization of the substituted N-triazole oxindole TROX-1, a small-molecule, state-dependent inhibitor of Ca(V)2 calcium channels. [electronic resource] by
- Swensen, Andrew M
- Herrington, James
- Bugianesi, Randal M
- Dai, Ge
- Haedo, Rodolfo J
- Ratliff, Kevin S
- Smith, McHardy M
- Warren, Vivien A
- Arneric, Stephen P
- Eduljee, Cyrus
- Parker, David
- Snutch, Terrance P
- Hoyt, Scott B
- London, Clare
- Duffy, Joseph L
- Kaczorowski, Gregory J
- McManus, Owen B
Producer: 20120411
In:
Molecular pharmacology vol. 81
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17.
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A-1048400 is a novel, orally active, state-dependent neuronal calcium channel blocker that produces dose-dependent antinociception without altering hemodynamic function in rats. [electronic resource] by
- Scott, Victoria E
- Vortherms, Timothy A
- Niforatos, Wende
- Swensen, Andrew M
- Neelands, Torben
- Milicic, Ivan
- Banfor, Patricia N
- King, Andrew
- Zhong, Chengmin
- Simler, Gricelda
- Zhan, Cenchen
- Bratcher, Natalie
- Boyce-Rustay, Janel M
- Zhu, Chang Z
- Bhatia, Pramila
- Doherty, George
- Mack, Helmut
- Stewart, Andrew O
- Jarvis, Michael F
Producer: 20120214
In:
Biochemical pharmacology vol. 83
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18.
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Biological Characterization of F508delCFTR Protein Processing by the CFTR Corrector ABBV-2222/GLPG2222. [electronic resource] by
- Singh, Ashvani K
- Fan, Yihong
- Balut, Corina
- Alani, Sara
- Manelli, Arlene M
- Swensen, Andrew M
- Jia, Ying
- Neelands, Torben R
- Vortherms, Timothy A
- Liu, Bo
- Searle, Xenia B
- Wang, Xueqing
- Gao, Wenqing
- Hwang, Tzyh-Chang
- Ren, Hong Y
- Cyr, Douglas
- Kym, Philip R
- Conrath, Katja
- Tse, Chris
Producer: 20200713
In:
The Journal of pharmacology and experimental therapeutics vol. 372
Availability: No items available.
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19.
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Pharmacologic inhibition of the renal outer medullary potassium channel causes diuresis and natriuresis in the absence of kaliuresis. [electronic resource] by
- Garcia, Maria L
- Priest, Birgit T
- Alonso-Galicia, Magdalena
- Zhou, Xiaoyan
- Felix, John P
- Brochu, Richard M
- Bailey, Timothy
- Thomas-Fowlkes, Brande
- Liu, Jessica
- Swensen, Andrew
- Pai, Lee-Yuh
- Xiao, Jianying
- Hernandez, Melba
- Hoagland, Kimberly
- Owens, Karen
- Tang, Haifeng
- de Jesus, Reynalda K
- Roy, Sophie
- Kaczorowski, Gregory J
- Pasternak, Alexander
Producer: 20140210
In:
The Journal of pharmacology and experimental therapeutics vol. 348
Availability: No items available.
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20.
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Discovery of ABBV/GLPG-3221, a Potent Corrector of CFTR for the Treatment of Cystic Fibrosis. [electronic resource] by
- Scanio, Marc J C
- Searle, Xenia B
- Liu, Bo
- Koenig, John R
- Altenbach, Robert
- Gfesser, Gregory A
- Bogdan, Andrew
- Greszler, Stephen
- Zhao, Gang
- Singh, Ashvani
- Fan, Yihong
- Swensen, Andrew M
- Vortherms, Timothy
- Manelli, Arlene
- Balut, Corina
- Jia, Ying
- Gao, Wenqing
- Yong, Hong
- Schrimpf, Michael
- Tse, Chris
- Kym, Philip
- Wang, Xueqing
Publication details: ACS medicinal chemistry letters Nov 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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