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Pharmacologic and genetic approaches define human pancreatic β cell mitogenic targets of DYRK1A inhibitors. [electronic resource] by
- Ackeifi, Courtney
- Swartz, Ethan
- Kumar, Kunal
- Liu, Hongtao
- Chalada, Suebsuwong
- Karakose, Esra
- Scott, Donald K
- Garcia-Ocaña, Adolfo
- Sanchez, Roberto
- DeVita, Robert J
- Stewart, Andrew F
- Wang, Peng
Producer: 20210510
In:
JCI insight vol. 5
Availability: No items available.
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Synthesis and Biological Validation of a Harmine-Based, Central Nervous System (CNS)-Avoidant, Selective, Human β-Cell Regenerative Dual-Specificity Tyrosine Phosphorylation-Regulated Kinase A (DYRK1A) Inhibitor. [electronic resource] by
- Kumar, Kunal
- Wang, Peng
- Wilson, Jessica
- Zlatanic, Viktor
- Berrouet, Cecilia
- Khamrui, Susmita
- Secor, Cody
- Swartz, Ethan A
- Lazarus, Michael
- Sanchez, Roberto
- Stewart, Andrew F
- Garcia-Ocana, Adolfo
- DeVita, Robert J
Producer: 20200902
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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Combined Inhibition of DYRK1A, SMAD, and Trithorax Pathways Synergizes to Induce Robust Replication in Adult Human Beta Cells. [electronic resource] by
- Wang, Peng
- Karakose, Esra
- Liu, Hongtao
- Swartz, Ethan
- Ackeifi, Courtney
- Zlatanic, Viktor
- Wilson, Jessica
- González, Bryan J
- Bender, Aaron
- Takane, Karen K
- Ye, Lillian
- Harb, George
- Pagliuca, Felicia
- Homann, Dirk
- Egli, Dieter
- Argmann, Carmen
- Scott, Donald K
- Garcia-Ocaña, Adolfo
- Stewart, Andrew F
Producer: 20200511
In:
Cell metabolism vol. 29
Availability: No items available.
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GLP-1 receptor agonists synergize with DYRK1A inhibitors to potentiate functional human β cell regeneration. [electronic resource] by
- Ackeifi, Courtney
- Wang, Peng
- Karakose, Esra
- Manning Fox, Jocelyn E
- González, Bryan J
- Liu, Hongtao
- Wilson, Jessica
- Swartz, Ethan
- Berrouet, Cecilia
- Li, Yansui
- Kumar, Kunal
- MacDonald, Patrick E
- Sanchez, Roberto
- Thorens, Bernard
- DeVita, Robert
- Homann, Dirk
- Egli, Dieter
- Scott, Donald K
- Garcia-Ocaña, Adolfo
- Stewart, Andrew F
Producer: 20210623
In:
Science translational medicine vol. 12
Availability: No items available.
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