Discovery and Structure-Activity-Relationship Study of N-Alkyl-5-hydroxypyrimidinone Carboxamides as Novel Antitubercular Agents Targeting Decaprenylphosphoryl-β-d-ribose 2'-Oxidase. [electronic resource]
Producer: 20190930Description: 9952-9965 p. digitalISSN:- 1520-4804
- Alkylation
- Animals
- Antitubercular Agents -- chemistry
- Drug Design
- Female
- High-Throughput Screening Assays
- Mice
- Microbial Sensitivity Tests
- Molecular Docking Simulation
- Molecular Targeted Therapy
- Mycobacterium tuberculosis -- drug effects
- Oxidoreductases -- chemistry
- Protein Conformation
- Pyrimidinones -- chemistry
- Structure-Activity Relationship
- Tissue Distribution
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Publication Type: Journal Article; Research Support, N.I.H., Intramural; Research Support, Non-U.S. Gov't
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