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Structure-activity relationship studies and discovery of a potent transient receptor potential vanilloid (TRPV1) antagonist 4-[3-chloro-5-[(1S)-1,2-dihydroxyethyl]-2-pyridyl]-N-[5-(trifluoromethyl)-2-pyridyl]-3,6-dihydro-2H-pyridine-1-carboxamide (V116517) as a clinical candidate for pain management. [electronic resource] by
- Tafesse, Laykea
- Kanemasa, Toshiyuki
- Kurose, Noriyuki
- Yu, Jianming
- Asaki, Toshiyuki
- Wu, Gang
- Iwamoto, Yuka
- Yamaguchi, Yoshitaka
- Ni, Chiyou
- Engel, John
- Tsuno, Naoki
- Patel, Aniket
- Zhou, Xiaoming
- Shintani, Takuya
- Brown, Kevin
- Hasegawa, Tsuyoshi
- Shet, Manjunath
- Iso, Yasuyoshi
- Kato, Akira
- Kyle, Donald J
Producer: 20150207
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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