Discovery of 2-aryl-8-hydroxy (or methoxy)-isoquinolin-1(2H)-ones as novel EGFR inhibitor by scaffold hopping. [electronic resource]
Producer: 20140514Description: 6956-64 p. digitalISSN:- 1464-3391
- Antineoplastic Agents -- chemistry
- Binding Sites
- Cell Line, Tumor
- Cell Proliferation -- drug effects
- Drug Evaluation, Preclinical
- ErbB Receptors -- antagonists & inhibitors
- Humans
- Isoquinolines -- chemistry
- Molecular Docking Simulation
- Protein Binding -- drug effects
- Protein Kinase Inhibitors -- chemistry
- Protein Structure, Tertiary
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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