Results
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1.
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Structure-based design of nonpeptide inhibitors of interleukin-1beta converting enzyme (ICE, caspase-1). [electronic resource] by
- Shahripour, Aurash B
- Plummer, Mark S
- Lunney, Elizabeth A
- Albrecht, Hans P
- Hays, Sheryl J
- Kostlan, Catherine R
- Sawyer, Tomi K
- Walker, Nigel P C
- Brady, Kenneth D
- Allen, Hamish J
- Talanian, Robert V
- Wong, Winnie W
- Humblet, Christine
Producer: 20020312
In:
Bioorganic & medicinal chemistry vol. 10
Availability: No items available.
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2.
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Discovery of Selective Small Molecule ROMK Inhibitors as Potential New Mechanism Diuretics. [electronic resource] by
- Tang, Haifeng
- Walsh, Shawn P
- Yan, Yan
- de Jesus, Reynalda K
- Shahripour, Aurash
- Teumelsan, Nardos
- Zhu, Yuping
- Ha, Sookhee
- Owens, Karen A
- Thomas-Fowlkes, Brande S
- Felix, John P
- Liu, Jessica
- Kohler, Martin
- Priest, Birgit T
- Bailey, Timothy
- Brochu, Richard
- Alonso-Galicia, Magdalena
- Kaczorowski, Gregory J
- Roy, Sophie
- Yang, Lihu
- Mills, Sander G
- Garcia, Maria L
- Pasternak, Alexander
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 3
Availability: No items available.
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3.
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Discovery of potent selective bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model. Part II: optimization studies and demonstration of in vivo efficacy. [electronic resource] by
- Plummer, Mark S
- Cornicelli, Joseph
- Roark, Howard
- Skalitzky, Donald J
- Stankovic, Charles J
- Bove, Susan
- Pandit, Jayvardhan
- Goodman, Annise
- Hicks, James
- Shahripour, Aurash
- Beidler, David
- Lu, Xiao Kang
- Sanchez, Brian
- Whitehead, Christopher
- Sarver, Ron
- Braden, Timothy
- Gowan, Richard
- Shen, Xi Qiang
- Welch, Katherine
- Ogden, Adam
- Sadagopan, Nalini
- Baum, Heidi
- Miller, Howard
- Banotai, Craig
- Spessard, Cindy
- Lightle, Sandra
Producer: 20131209
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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4.
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Discovery of potent, selective, bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model, part I: transformation of selective pyrazolodiazepinone phosphodiesterase 4 (PDE4) inhibitors into selective PDE2 inhibitors. [electronic resource] by
- Plummer, Mark S
- Cornicelli, Joseph
- Roark, Howard
- Skalitzky, Donald J
- Stankovic, Charles J
- Bove, Susan
- Pandit, Jayvardhan
- Goodman, Annise
- Hicks, James
- Shahripour, Aurash
- Beidler, David
- Lu, Xiao Kang
- Sanchez, Brian
- Whitehead, Christopher
- Sarver, Ron
- Braden, Timothy
- Gowan, Richard
- Shen, Xi Qiang
- Welch, Katherine
- Ogden, Adam
- Sadagopan, Nalini
- Baum, Heidi
- Miller, Howard
- Banotai, Craig
- Spessard, Cindy
- Lightle, Sandra
Producer: 20131209
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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5.
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Differentiation of ROMK potency from hERG potency in the phenacetyl piperazine series through heterocycle incorporation. [electronic resource] by
- Walsh, Shawn P
- Shahripour, Aurash
- Tang, Haifeng
- de Jesus, Reynalda K
- Teumelsan, Nardos
- Zhu, Yuping
- Frie, Jessica
- Priest, Birgit T
- Swensen, Andrew M
- Alonso-Galicia, Magdalena
- Felix, John P
- Brochu, Richard M
- Bailey, Timothy
- Thomas-Fowlkes, Brande
- Zhou, Xiaoyan
- Pai, Lee-Yuh
- Hampton, Caryn
- Hernandez, Melba
- Owens, Karen
- Ehrhart, Juliann
- Roy, Sophie
- Kaczorowski, Gregory J
- Yang, Lihu
- Garcia, Maria L
- Pasternak, Alexander
Producer: 20161219
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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6.
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Discovery of MK-7145, an Oral Small Molecule ROMK Inhibitor for the Treatment of Hypertension and Heart Failure. [electronic resource] by
- Tang, Haifeng
- Zhu, Yuping
- Teumelsan, Nardos
- Walsh, Shawn P
- Shahripour, Aurash
- Priest, Birgit T
- Swensen, Andrew M
- Felix, John P
- Brochu, Richard M
- Bailey, Timothy
- Thomas-Fowlkes, Brande
- Pai, Lee-Yuh
- Hampton, Caryn
- Corona, Aaron
- Hernandez, Melba
- Metzger, Joseph
- Forrest, Michael
- Zhou, Xiaoyan
- Owens, Karen
- Tong, Vincent
- Parmee, Emma
- Roy, Sophie
- Kaczorowski, Gregory J
- Yang, Lihu
- Alonso-Galicia, Magdalena
- Garcia, Maria L
- Pasternak, Alexander
Producer: 20160720
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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7.
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4-anilino-5-carboxamido-2-pyridone derivatives as noncompetitive inhibitors of mitogen-activated protein kinase kinase. [electronic resource] by
- Spicer, Julie A
- Rewcastle, Gordon W
- Kaufman, Michael D
- Black, Shannon L
- Plummer, Mark S
- Denny, William A
- Quin, John
- Shahripour, Aurash B
- Barrett, Stephen D
- Whitehead, Christopher E
- Milbank, Jared B J
- Ohren, Jeffrey F
- Gowan, Richard C
- Omer, Charles
- Camp, Heidi S
- Esmaeil, Nadia
- Moore, Kelley
- Sebolt-Leopold, Judith S
- Pryzbranowski, Sally
- Merriman, Ronald L
- Ortwine, Daniel F
- Warmus, Joseph S
- Flamme, Cathlin M
- Pavlovsky, Alexander G
- Tecle, Haile
Producer: 20071127
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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8.
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Discovery of a potent and selective ROMK inhibitor with improved pharmacokinetic properties based on an octahydropyrazino[2,1-c][1,4]oxazine scaffold. [electronic resource] by
- Zhu, Yuping
- de Jesus, Reynalda K
- Tang, Haifeng
- Walsh, Shawn P
- Jiang, Jinlong
- Gu, Xin
- Teumelsan, Nardos
- Shahripour, Aurash
- Pio, Barbara
- Ding, Fa-Xiang
- Ha, Sookhee
- Priest, Birgit T
- Swensen, Andrew M
- Alonso-Galicia, Magdalena
- Felix, John P
- Brochu, Richard M
- Bailey, Timothy
- Thomas-Fowlkes, Brande
- Zhou, Xiaoyan
- Pai, Lee-Yuh
- Hampton, Caryn
- Hernandez, Melba
- Owens, Karen
- Ehrhart, Juliann
- Roy, Sophie
- Kaczorowski, Gregory J
- Yang, Lihu
- Parmee, Emma R
- Sullivan, Kathleen
- Garcia, Maria L
- Pasternak, Alexander
Producer: 20170627
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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9.
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Discovery of a Potent and Selective ROMK Inhibitor with Pharmacokinetic Properties Suitable for Preclinical Evaluation. [electronic resource] by
- Walsh, Shawn P
- Shahripour, Aurash
- Tang, Haifeng
- Teumelsan, Nardos
- Frie, Jessica
- Zhu, Yuping
- Priest, Birgit T
- Swensen, Andrew M
- Liu, Jessica
- Margulis, Michael
- Visconti, Richard
- Weinglass, Adam
- Felix, John P
- Brochu, Richard M
- Bailey, Timothy
- Thomas-Fowlkes, Brande
- Alonso-Galicia, Magdalena
- Zhou, Xiaoyan
- Pai, Lee-Yuh
- Corona, Aaron
- Hampton, Caryn
- Hernandez, Melba
- Bentley, Ross
- Chen, Jing
- Shah, Kashmira
- Metzger, Joseph
- Forrest, Michael
- Owens, Karen
- Tong, Vincent
- Ha, Sookhee
- Roy, Sophie
- Kaczorowski, Gregory J
- Yang, Lihu
- Parmee, Emma
- Garcia, Maria L
- Sullivan, Kathleen
- Pasternak, Alexander
Producer: 20150720
In:
ACS medicinal chemistry letters vol. 6
Availability: No items available.
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