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Design and Synthesis of P2-P4 Macrocycles Containing a Unique Spirocyclic Proline: A New Class of HCV NS3/4A Inhibitors. [electronic resource] by
- Velázquez, Francisco
- Chelliah, Mariappan
- Clasby, Martin
- Guo, Zhuyan
- Howe, John
- Miller, Randy
- Neelamkavil, Santhosh
- Shah, Unmesh
- Soriano, Aileen
- Xia, Yan
- Venkatraman, Srikanth
- Chackalamannil, Samuel
- Davies, Ian W
Publication details: ACS medicinal chemistry letters Dec 2016
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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7.
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Biaryl and heteroaryl derivatives of SCH 58261 as potent and selective adenosine A2A receptor antagonists. [electronic resource] by
- Shah, Unmesh
- Boyle, Craig D
- Chackalamannil, Samuel
- Neustadt, Bernard R
- Lindo, Neil
- Greenlee, William J
- Foster, Carolyn
- Arik, Leyla
- Zhai, Ying
- Ng, Kwokei
- Wang, Shiyong
- Monopoli, Angela
- Lachowicz, Jean E
Producer: 20081117
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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8.
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Design, synthesis, and evaluation of fused heterocyclic analogs of SCH 58261 as adenosine A2A receptor antagonists. [electronic resource] by
- Shah, Unmesh
- Lankin, Claire M
- Boyle, Craig D
- Chackalamannil, Samuel
- Greenlee, William J
- Neustadt, Bernard R
- Cohen-Williams, Mary E
- Higgins, Guy A
- Ng, Kwokei
- Varty, Geoffrey B
- Zhang, Hongtao
- Lachowicz, Jean E
Producer: 20081117
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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9.
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Discovery of Chromane Propionic Acid Analogues as Selective Agonists of GPR120 with [electronic resource] by
- Adams, Gregory L
- Velazquez, Francisco
- Jayne, Charles
- Shah, Unmesh
- Miao, Shouwu
- Ashley, Eric R
- Madeira, Maria
- Akiyama, Taro E
- Di Salvo, Jerry
- Suzuki, Takao
- Wang, Nengxue
- Truong, Quang
- Gilbert, Eric
- Zhou, Dan
- Verras, Andreas
- Kirkland, Melissa
- Pachanski, Michele
- Powles, Maryann
- Yin, Wu
- Ujjainwalla, Feroze
- Venkatraman, Srikanth
- Edmondson, Scott D
Publication details: ACS medicinal chemistry letters Jan 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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10.
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Novel Quinoline-Based P2-P4 Macrocyclic Derivatives As Pan-Genotypic HCV NS3/4a Protease Inhibitors. [electronic resource] by
- Shah, Unmesh
- Jayne, Charles
- Chackalamannil, Samuel
- Velázquez, Francisco
- Guo, Zhuyan
- Buevich, Alexei
- Howe, John A
- Chase, Robert
- Soriano, Aileen
- Agrawal, Sony
- Rudd, Michael T
- McCauley, John A
- Liverton, Nigel J
- Romano, Joseph
- Bush, Kimberly
- Coleman, Paul J
- Grisé-Bard, Christiane
- Brochu, Marie-Christine
- Charron, Sylvie
- Aulakh, Virender
- Bachand, Benoit
- Beaulieu, Patrick
- Zaghdane, Helmi
- Bhat, Sathesh
- Han, Yongxin
- Vacca, Joseph P
- Davies, Ian W
- Weber, Ann E
- Venkatraman, Srikanth
Producer: 20140606
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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11.
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Discovery of MK-8831, A Novel Spiro-Proline Macrocycle as a Pan-Genotypic HCV-NS3/4a Protease Inhibitor. [electronic resource] by
- Neelamkavil, Santhosh F
- Agrawal, Sony
- Bara, Thomas
- Bennett, Chad
- Bhat, Sathesh
- Biswas, Dipshikha
- Brockunier, Linda
- Buist, Nicole
- Burnette, Duane
- Cartwright, Mark
- Chackalamannil, Samuel
- Chase, Robert
- Chelliah, Mariappan
- Chen, Austin
- Clasby, Martin
- Colandrea, Vincent J
- Davies, Ian W
- Eagen, Keith
- Guo, Zhuyan
- Han, Yongxin
- Howe, John
- Jayne, Charles
- Josien, Hubert
- Kargman, Stacia
- Marcantonio, Karen
- Miao, Shouwu
- Miller, Randy
- Nolting, Andrew
- Pinto, Patrick
- Rajagopalan, Murali
- Ruck, Rebecca T
- Shah, Unmesh
- Soriano, Aileen
- Sperbeck, Donald
- Velazquez, Francisco
- Wu, Jin
- Xia, Yan
- Venkatraman, Srikanth
Producer: 20160128
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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12.
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Design, Synthesis, and Evaluation of Novel and Selective G-protein Coupled Receptor 120 (GPR120) Spirocyclic Agonists. [electronic resource] by
- Cox, Jason M
- Chu, Hong D
- Chelliah, Mariappan V
- Debenham, John S
- Eagen, Keith
- Lan, Ping
- Lombardo, Matthew
- London, Clare
- Plotkin, Michael A
- Shah, Unmesh
- Sun, Zhongxiang
- Vaccaro, Henry M
- Venkatraman, Srikanth
- Suzuki, Takao
- Wang, Nengxue
- Ashley, Eric R
- Crespo, Alejandro
- Madeira, Maria
- Leung, Dennis H
- Alleyne, Candice
- Ogawa, Aimie M
- Souza, Sarah
- Thomas-Fowlkes, Brande
- Di Salvo, Jerry
- Weinglass, Adam
- Kirkland, Melissa
- Pachanski, Michele
- Powles, Mary Ann
- Tozzo, Effie
- Akiyama, Taro E
- Ujjainwalla, Feroze
- Tata, James R
- Sinz, Christopher J
Publication details: ACS medicinal chemistry letters Jan 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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