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Retro-binding thrombin active site inhibitors: identification of an orally active inhibitor of thrombin catalytic activity. [electronic resource] by
- Iwanowicz, Edwin J
- Kimball, S David
- Lin, James
- Lau, Wan
- Han, W-C
- Wang, Tammy C
- Roberts, Daniel G M
- Schumacher, W A
- Ogletree, Martin L
- Seiler, Steven M
Producer: 20030318
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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6.
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Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors. [electronic resource] by
- Sutton, James C
- Bolton, Scott A
- Davis, Malcolm E
- Hartl, Karen S
- Jacobson, Bruce
- Mathur, Arvind
- Ogletree, Martin L
- Slusarchyk, William A
- Zahler, Robert
- Seiler, Steven M
- Bisacchi, Gregory S
Producer: 20041222
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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7.
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Synthesis of potent and highly selective nonguanidine azetidinone inhibitors of human tryptase. [electronic resource] by
- Bisacchi, Gregory S
- Slusarchyk, William A
- Bolton, Scott A
- Hartl, Karen S
- Jacobs, Glenn
- Mathur, Arvind
- Meng, Wei
- Ogletree, Martin L
- Pi, Zulan
- Sutton, James C
- Treuner, Uwe
- Zahler, Robert
- Zhao, Guohua
- Seiler, Steven M
Producer: 20041222
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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8.
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Synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors. [electronic resource] by
- Sutton, James C
- Bolton, Scott A
- Hartl, Karen S
- Huang, Ming-Hsing
- Jacobs, Glenn
- Meng, Wei
- Ogletree, Martin L
- Pi, Zulan
- Schumacher, William A
- Seiler, Steven M
- Slusarchyk, William A
- Treuner, Uwe
- Zahler, Robert
- Zhao, Guohua
- Bisacchi, Gregory S
Producer: 20030318
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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9.
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Synthesis of potent and highly selective inhibitors of human tryptase. [electronic resource] by
- Slusarchyk, William A
- Bolton, Scott A
- Hartl, Karen S
- Huang, Ming-Hsing
- Jacobs, Glenn
- Meng, Wei
- Ogletree, Martin L
- Pi, Zulan
- Schumacher, William A
- Seiler, Steven M
- Sutton, James C
- Treuner, Uwe
- Zahler, Robert
- Zhao, Guohua
- Bisacchi, Gregory S
Producer: 20030318
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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10.
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Molecular design and structure--activity relationships leading to the potent, selective, and orally active thrombin active site inhibitor BMS-189664. [electronic resource] by
- Das, Jagabandhu
- Kimball, S David
- Hall, Steven E
- Han, Wen Ching
- Iwanowicz, Edwin
- Lin, James
- Moquin, Robert V
- Reid, Joyce A
- Sack, John S
- Malley, Mary F
- Chang, Chiehying Y
- Chong, Saeho
- Wang-Iverson, David B
- Roberts, Daniel G M
- Seiler, Steven M
- Schumacher, William A
- Ogletree, Martin L
Producer: 20021004
In:
Bioorganic & medicinal chemistry letters vol. 12
Availability: No items available.
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11.
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Discovery of nonbenzamidine factor VIIa inhibitors using a biaryl acid scaffold. [electronic resource] by
- Bolton, Scott A
- Sutton, James C
- Anumula, Rushith
- Bisacchi, Gregory S
- Jacobson, Bruce
- Slusarchyk, William A
- Treuner, Uwe D
- Wu, Shung C
- Zhao, Guohua
- Pi, Zulan
- Sheriff, Steven
- Smirk, Rebecca A
- Bisaha, Sharon
- Cheney, Daniel L
- Wei, Anzhi
- Schumacher, William A
- Hartl, Karen S
- Liu, Eddie
- Zahler, Robert
- Seiler, Steven M
Producer: 20140331
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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12.
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Ketene aminal-based lactam derivatives as a novel class of orally active FXa inhibitors. [electronic resource] by
- Shi, Yan
- Zhang, Jing
- Stein, Philip D
- Shi, Mengxiao
- O'Connor, Stephen P
- Bisaha, Sharon N
- Li, Chi
- Atwal, Karnail S
- Bisacchi, Gregory S
- Sitkoff, Doree
- Pudzianowski, Andrew T
- Liu, Eddie C
- Hartl, Karen S
- Seiler, Steven M
- Youssef, Sonia
- Steinbacher, Thomas E
- Schumacher, William A
- Rendina, Alan R
- Bozarth, Jeffrey M
- Peterson, Tara L
- Zhang, Ge
- Zahler, Robert
Producer: 20060627
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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