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Novel peroxisome proliferator-activated receptor alpha agonists lower low-density lipoprotein and triglycerides, raise high-density lipoprotein, and synergistically increase cholesterol excretion with a liver X receptor agonist. [electronic resource] by
- Mukherjee, Ranjan
- Locke, Kenneth T
- Miao, Bowman
- Meyers, Daniel
- Monshizadegan, Hossain
- Zhang, Rongan
- Search, Debra
- Grimm, Denise
- Flynn, Michael
- O'Malley, Kevin M
- Zhang, Litao
- Li, Jun
- Shi, Yan
- Kennedy, Lawrence J
- Blanar, Michael
- Cheng, Peter T
- Tino, Joseph
- Srivastava, Rai Ajit
Producer: 20090105
In:
The Journal of pharmacology and experimental therapeutics vol. 327
Availability: No items available.
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P2Y6 receptor potentiates pro-inflammatory responses in macrophages and exhibits differential roles in atherosclerotic lesion development. [electronic resource] by
- Garcia, Ricardo A
- Yan, Mujing
- Search, Debra
- Zhang, Rongan
- Carson, Nancy L
- Ryan, Carol S
- Smith-Monroy, Constance
- Zheng, Joanna
- Chen, Jian
- Kong, Yan
- Tang, Huaping
- Hellings, Samuel E
- Wardwell-Swanson, Judith
- Dinchuk, Joseph E
- Psaltis, George C
- Gordon, David A
- Glunz, Peter W
- Gargalovic, Peter S
Producer: 20150625
In:
PloS one vol. 9
Availability: No items available.
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Synthesis and structure-activity relationships of 2-aryl-4-oxazolylmethoxy benzylglycines and 2-aryl-4-thiazolylmethoxy benzylglycines as novel, potent PPARalpha selective activators- PPARalpha and PPARgamma selectivity modulation. [electronic resource] by
- Ye, Xiang-Yang
- Chen, Stephanie
- Zhang, Hao
- Locke, Kenneth T
- O'Malley, Kevin
- Zhang, Litao
- Srivastava, Raijit
- Miao, Bowman
- Meyers, Daniel
- Monshizadegan, Hossain
- Search, Debra
- Grimm, Denise
- Zhang, Rongan
- Lippy, Jonathan
- Twamley, Celeste
- Muckelbauer, Jodi K
- Chang, Chiehying
- An, Yongmi
- Hosagrahara, Vinayak
- Zhang, Lisa
- Yang, T-J
- Mukherjee, Ranjan
- Cheng, Peter T W
- Tino, Joseph A
Producer: 20100727
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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The Guinea pig as a preclinical model for demonstrating the efficacy and safety of statins. [electronic resource] by
- Madsen, Cort S
- Janovitz, Evan
- Zhang, Rongan
- Nguyen-Tran, Van
- Ryan, Carol S
- Yin, Xiaohong
- Monshizadegan, Hossain
- Chang, Ming
- D'Arienzo, Celia
- Scheer, Susan
- Setters, Robert
- Search, Debra
- Chen, Xing
- Zhuang, Shaobin
- Kunselman, Lori
- Peters, Andrew
- Harrity, Thomas
- Apedo, Atsu
- Huang, Christine
- Cuff, Carolyn A
- Kowala, Mark C
- Blanar, Michael A
- Sun, Chong-Qing
- Robl, Jeffrey A
- Stein, Philip D
Producer: 20080219
In:
The Journal of pharmacology and experimental therapeutics vol. 324
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11β-hydroxysteroid dehydrogenase type 1 gene knockout attenuates atherosclerosis and in vivo foam cell formation in hyperlipidemic apoE⁻/⁻ mice. [electronic resource] by
- García, Ricardo A
- Search, Debra J
- Lupisella, John A
- Ostrowski, Jacek
- Guan, Bo
- Chen, Jian
- Yang, Wen-Pin
- Truong, Amy
- He, Aiqing
- Zhang, Rongan
- Yan, Mujing
- Hellings, Samuel E
- Gargalovic, Peter S
- Ryan, Carol S
- Watson, Linda M
- Langish, Robert A
- Shipkova, Petia A
- Carson, Nancy L
- Taylor, Joseph R
- Yang, Richard
- Psaltis, George C
- Harrity, Thomas W
- Robl, Jeffrey A
- Gordon, David A
Producer: 20130715
In:
PloS one vol. 8
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(3R,5S,E)-7-(4-(4-fluorophenyl)-6-isopropyl-2-(methyl(1-methyl-1h-1,2,4-triazol-5-yl)amino)pyrimidin-5-yl)-3,5-dihydroxyhept-6-enoic acid (BMS-644950): a rationally designed orally efficacious 3-hydroxy-3-methylglutaryl coenzyme-a reductase inhibitor with reduced myotoxicity potential. [electronic resource] by
- Ahmad, Saleem
- Madsen, Cort S
- Stein, Philip D
- Janovitz, Evan
- Huang, Christine
- Ngu, Khehyong
- Bisaha, Sharon
- Kennedy, Lawrence J
- Chen, Bang-Chi
- Zhao, Rulin
- Sitkoff, Doree
- Monshizadegan, Hossain
- Yin, Xiaohong
- Ryan, Carol S
- Zhang, Rongan
- Giancarli, Mary
- Bird, Eileen
- Chang, Ming
- Chen, Xing
- Setters, Robert
- Search, Debra
- Zhuang, Shaobin
- Nguyen-Tran, Van
- Cuff, Carolyn A
- Harrity, Thomas
- Darienzo, Celia J
- Li, Tong
- Reeves, Richard A
- Blanar, Michael A
- Barrish, Joel C
- Zahler, Robert
- Robl, Jeffrey A
Producer: 20080709
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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8.
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Discovery and Preclinical Evaluation of BMS-711939, an Oxybenzylglycine Based PPARα Selective Agonist. [electronic resource] by
- Shi, Yan
- Li, Jun
- Kennedy, Lawrence J
- Tao, Shiwei
- Hernández, Andrés S
- Lai, Zhi
- Chen, Sean
- Wong, Henry
- Zhu, Juliang
- Trehan, Ashok
- Lim, Ngiap-Kie
- Zhang, Huiping
- Chen, Bang-Chi
- Locke, Kenneth T
- O'Malley, Kevin M
- Zhang, Litao
- Srivastava, Rai Ajit
- Miao, Bowman
- Meyers, Daniel S
- Monshizadegan, Hossain
- Search, Debra
- Grimm, Denise
- Zhang, Rongan
- Harrity, Thomas
- Kunselman, Lori K
- Cap, Michael
- Muckelbauer, Jodi
- Chang, Chiehying
- Krystek, Stanley R
- Li, Yi-Xin
- Hosagrahara, Vinayak
- Zhang, Lisa
- Kadiyala, Pathanjali
- Xu, Carrie
- Blanar, Michael A
- Zahler, Robert
- Mukherjee, Ranjan
- Cheng, Peter T W
- Tino, Joseph A
Producer: 20160621
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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9.
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Discovery of an oxybenzylglycine based peroxisome proliferator activated receptor alpha selective agonist 2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid (BMS-687453). [electronic resource] by
- Li, Jun
- Kennedy, Lawrence J
- Shi, Yan
- Tao, Shiwei
- Ye, Xiang-Yang
- Chen, Stephanie Y
- Wang, Ying
- Hernández, Andrés S
- Wang, Wei
- Devasthale, Pratik V
- Chen, Sean
- Lai, Zhi
- Zhang, Hao
- Wu, Shung
- Smirk, Rebecca A
- Bolton, Scott A
- Ryono, Denis E
- Zhang, Huiping
- Lim, Ngiap-Kie
- Chen, Bang-Chi
- Locke, Kenneth T
- O'Malley, Kevin M
- Zhang, Litao
- Srivastava, Rai Ajit
- Miao, Bowman
- Meyers, Daniel S
- Monshizadegan, Hossain
- Search, Debra
- Grimm, Denise
- Zhang, Rongan
- Harrity, Thomas
- Kunselman, Lori K
- Cap, Michael
- Kadiyala, Pathanjali
- Hosagrahara, Vinayak
- Zhang, Lisa
- Xu, Carrie
- Li, Yi-Xin
- Muckelbauer, Jodi K
- Chang, Chiehying
- An, Yongmi
- Krystek, Stanley R
- Blanar, Michael A
- Zahler, Robert
- Mukherjee, Ranjan
- Cheng, Peter T W
- Tino, Joseph A
Producer: 20100510
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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