Design, synthesis, and optimization of novel epoxide incorporating peptidomimetics as selective calpain inhibitors. [electronic resource]
Producer: 20131111Description: 6054-68 p. digitalISSN:- 1520-4804
- Calpain -- antagonists & inhibitors
- Catalytic Domain
- Click Chemistry
- Computer Simulation
- Drug Design
- Epoxy Compounds -- chemical synthesis
- Kinetics
- Leucine -- analogs & derivatives
- Molecular Docking Simulation
- Papain -- antagonists & inhibitors
- Peptidomimetics -- chemical synthesis
- Stereoisomerism
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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