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Biochemical characterization of recombinant influenza A polymerase heterotrimer complex: Polymerase activity and mechanisms of action of nucleotide analogs. [electronic resource] by
- Barauskas, Ona
- Xing, Weimei
- Aguayo, Esmeralda
- Willkom, Madeleine
- Sapre, Annapurna
- Clarke, Michael
- Birkus, Gabriel
- Schultz, Brian E
- Sakowicz, Roman
- Kwon, HyockJoo
- Feng, Joy Y
Producer: 20171023
In:
PloS one vol. 12
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Biochemical characterization of recombinant influenza A polymerase heterotrimer complex: Endonuclease activity and evaluation of inhibitors. [electronic resource] by
- Xing, Weimei
- Barauskas, Ona
- Kirschberg, Thorsten
- Niedziela-Majka, Anita
- Clarke, Michael
- Birkus, Gabriel
- Weissburg, Perry
- Liu, Xiaohong
- Schultz, Brian E
- Sakowicz, Roman
- Kwon, HyockJoo
- Feng, Joy Y
Producer: 20171011
In:
PloS one vol. 12
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7.
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Role of Mitochondrial RNA Polymerase in the Toxicity of Nucleotide Inhibitors of Hepatitis C Virus. [electronic resource] by
- Feng, Joy Y
- Xu, Yili
- Barauskas, Ona
- Perry, Jason K
- Ahmadyar, Shekeba
- Stepan, George
- Yu, Helen
- Babusis, Darius
- Park, Yeojin
- McCutcheon, Krista
- Perron, Michel
- Schultz, Brian E
- Sakowicz, Roman
- Ray, Adrian S
Producer: 20161213
In:
Antimicrobial agents and chemotherapy vol. 60
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8.
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Biochemical characterization of tirabrutinib and other irreversible inhibitors of Bruton's tyrosine kinase reveals differences in on - and off - target inhibition. [electronic resource] by
- Liclican, Albert
- Serafini, Loredana
- Xing, Weimei
- Czerwieniec, Gregg
- Steiner, Bart
- Wang, Ting
- Brendza, Katherine M
- Lutz, Justin D
- Keegan, Kathleen S
- Ray, Adrian S
- Schultz, Brian E
- Sakowicz, Roman
- Feng, Joy Y
Producer: 20200914
In:
Biochimica et biophysica acta. General subjects vol. 1864
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Structural, biochemical, and biophysical characterization of idelalisib binding to phosphoinositide 3-kinase δ. [electronic resource] by
- Somoza, John R
- Koditek, David
- Villaseñor, Armando G
- Novikov, Nikolai
- Wong, Melanie H
- Liclican, Albert
- Xing, Weimei
- Lagpacan, Leanna
- Wang, Ruth
- Schultz, Brian E
- Papalia, Giuseppe A
- Samuel, Dharmaraj
- Lad, Latesh
- McGrath, Mary E
Producer: 20150602
In:
The Journal of biological chemistry vol. 290
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Biochemical characterization and structure determination of a potent, selective antibody inhibitor of human MMP9. [electronic resource] by
- Appleby, Todd C
- Greenstein, Andrew E
- Hung, Magdeleine
- Liclican, Albert
- Velasquez, Maile
- Villaseñor, Armando G
- Wang, Ruth
- Wong, Melanie H
- Liu, Xiaohong
- Papalia, Giuseppe A
- Schultz, Brian E
- Sakowicz, Roman
- Smith, Victoria
- Kwon, Hyock Joo
Producer: 20170621
In:
The Journal of biological chemistry vol. 292
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11.
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The KN-93 Molecule Inhibits Calcium/Calmodulin-Dependent Protein Kinase II (CaMKII) Activity by Binding to Ca [electronic resource] by
- Wong, Melanie H
- Samal, Alexandra B
- Lee, Mike
- Vlach, Jiri
- Novikov, Nikolai
- Niedziela-Majka, Anita
- Feng, Joy Y
- Koltun, Dmitry O
- Brendza, Katherine M
- Kwon, Hyock Joo
- Schultz, Brian E
- Sakowicz, Roman
- Saad, Jamil S
- Papalia, Giuseppe A
Producer: 20200402
In:
Journal of molecular biology vol. 431
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Discovery of selective irreversible inhibitors for Bruton's tyrosine kinase. [electronic resource] by
- Pan, Zhengying
- Scheerens, Heleen
- Li, Shyr-Jiann
- Schultz, Brian E
- Sprengeler, Paul A
- Burrill, L Chuck
- Mendonca, Rohan V
- Sweeney, Michael D
- Scott, Keana C K
- Grothaus, Paul G
- Jeffery, Douglas A
- Spoerke, Jill M
- Honigberg, Lee A
- Young, Peter R
- Dalrymple, Stacie A
- Palmer, James T
Producer: 20080715
In:
ChemMedChem vol. 2
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13.
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Discovery of the pan-genotypic hepatitis C virus NS3/4A protease inhibitor voxilaprevir (GS-9857): A component of Vosevi [electronic resource] by
- Taylor, James G
- Zipfel, Sheila
- Ramey, Kyla
- Vivian, Randy
- Schrier, Adam
- Karki, Kapil K
- Katana, Ashley
- Kato, Darryl
- Kobayashi, Tetsuya
- Martinez, Ruben
- Sangi, Michael
- Siegel, Dustin
- Tran, Chinh V
- Yang, Zheng-Yu
- Zablocki, Jeff
- Yang, Cheng Y
- Wang, Yujin
- Wang, Kelly
- Chan, Katie
- Barauskas, Ona
- Cheng, Guofeng
- Jin, Debi
- Schultz, Brian E
- Appleby, Todd
- Villaseñor, Armando G
- Link, John O
Producer: 20200922
In:
Bioorganic & medicinal chemistry letters vol. 29
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14.
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Discovery of Potent and Selective MTH1 Inhibitors for Oncology: Enabling Rapid Target (In)Validation. [electronic resource] by
- Farand, Julie
- Kropf, Jeffrey E
- Blomgren, Peter
- Xu, Jianjun
- Schmitt, Aaron C
- Newby, Zachary E
- Wang, Ting
- Murakami, Eisuke
- Barauskas, Ona
- Sudhamsu, Jawahar
- Feng, Joy Y
- Niedziela-Majka, Anita
- Schultz, Brian E
- Schwartz, Karen
- Viatchenko-Karpinski, Serge
- Kornyeyev, Dmytro
- Kashishian, Adam
- Fan, Peidong
- Chen, Xiaowu
- Lansdon, Eric B
- Ports, Michael O
- Currie, Kevin S
- Watkins, William J
- Notte, Gregory T
Publication details: ACS medicinal chemistry letters Mar 2020
In:
ACS medicinal chemistry letters vol. 11
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15.
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Discovery of Potent Cyclophilin Inhibitors Based on the Structural Simplification of Sanglifehrin A. [electronic resource] by
- Steadman, Victoria A
- Pettit, Simon B
- Poullennec, Karine G
- Lazarides, Linos
- Keats, Andrew J
- Dean, David K
- Stanway, Steven J
- Austin, Carol A
- Sanvoisin, Jonathan A
- Watt, Gregory M
- Fliri, Hans G
- Liclican, Albert C
- Jin, Debi
- Wong, Melanie H
- Leavitt, Stephanie A
- Lee, Yu-Jen
- Tian, Yang
- Frey, Christian R
- Appleby, Todd C
- Schmitz, Uli
- Jansa, Petr
- Mackman, Richard L
- Schultz, Brian E
Producer: 20170706
In:
Journal of medicinal chemistry vol. 60
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16.
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ASK1 contributes to fibrosis and dysfunction in models of kidney disease. [electronic resource] by
- Liles, John T
- Corkey, Britton K
- Notte, Gregory T
- Budas, Grant R
- Lansdon, Eric B
- Hinojosa-Kirschenbaum, Ford
- Badal, Shawn S
- Lee, Michael
- Schultz, Brian E
- Wise, Sarah
- Pendem, Swetha
- Graupe, Michael
- Castonguay, Laurie
- Koch, Keith A
- Wong, Melanie H
- Papalia, Giuseppe A
- French, Dorothy M
- Sullivan, Theodore
- Huntzicker, Erik G
- Ma, Frank Y
- Nikolic-Paterson, David J
- Altuhaifi, Tareq
- Yang, Haichun
- Fogo, Agnes B
- Breckenridge, David G
Producer: 20190911
In:
The Journal of clinical investigation vol. 128
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17.
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Discovery of a Potent and Orally Bioavailable Cyclophilin Inhibitor Derived from the Sanglifehrin Macrocycle. [electronic resource] by
- Mackman, Richard L
- Steadman, Victoria A
- Dean, David K
- Jansa, Petr
- Poullennec, Karine G
- Appleby, Todd
- Austin, Carol
- Blakemore, Caroline A
- Cai, Ruby
- Cannizzaro, Carina
- Chin, Gregory
- Chiva, Jean-Yves C
- Dunbar, Neil A
- Fliri, Hans
- Highton, Adrian J
- Hui, Hon
- Ji, Mingzhe
- Jin, Haolun
- Karki, Kapil
- Keats, Andrew J
- Lazarides, Linos
- Lee, Yu-Jen
- Liclican, Albert
- Mish, Michael
- Murray, Bernard
- Pettit, Simon B
- Pyun, Peter
- Sangi, Michael
- Santos, Rex
- Sanvoisin, Jonathan
- Schmitz, Uli
- Schrier, Adam
- Siegel, Dustin
- Sperandio, David
- Stepan, George
- Tian, Yang
- Watt, Gregory M
- Yang, Hai
- Schultz, Brian E
Producer: 20190919
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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