Pharmacological characterization of 2-methyl-N-((2'-(pyrrolidin-1-ylsulfonyl)biphenyl-4-yl)methyl)propan-1-amine (PF-04455242), a high-affinity antagonist selective for κ-opioid receptors. [electronic resource]
Producer: 20120116Description: 555-66 p. digitalISSN:- 1521-0103
- Animals
- Behavior, Addictive -- drug therapy
- Biomarkers, Pharmacological -- blood
- Biphenyl Compounds -- blood
- Conditioning, Psychological
- Depression -- drug therapy
- Dose-Response Relationship, Drug
- Drug Evaluation, Preclinical
- Extinction, Psychological -- drug effects
- Humans
- Male
- Mice
- Mice, Inbred C57BL
- Mice, Inbred ICR
- Molecular Targeted Therapy
- Motor Activity -- drug effects
- Narcotic Antagonists -- blood
- Narcotics -- blood
- Opioid-Related Disorders -- drug therapy
- Piperazines -- metabolism
- Prolactin -- blood
- Pyrrolidines -- metabolism
- Radioligand Assay
- Rats
- Rats, Sprague-Dawley
- Receptors, Opioid, kappa -- antagonists & inhibitors
- Receptors, Opioid, mu -- metabolism
- Sulfonamides -- blood
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Publication Type: Journal Article
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