Antimalarial activity and mechanisms of action of two novel 4-aminoquinolines against chloroquine-resistant parasites. [electronic resource]
Producer: 20121009Description: e37259 p. digitalISSN:- 1932-6203
- Aminoquinolines -- chemistry
- Animals
- Antimalarials -- chemistry
- Cell Line, Tumor
- Chloroquine
- Dose-Response Relationship, Drug
- Drug Resistance -- physiology
- Enzyme-Linked Immunosorbent Assay
- Hemeproteins -- antagonists & inhibitors
- Humans
- In Vitro Techniques
- L-Lactate Dehydrogenase -- metabolism
- Malaria -- drug therapy
- Mice
- Models, Molecular
- Molecular Structure
- Plasmodium berghei -- drug effects
- Plasmodium falciparum -- drug effects
- Protein Binding
- Protein Conformation
- Tetrazolium Salts
- Thiazoles
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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