Structure-based design and synthesis of pyrazinones containing novel P1 'side pocket' moieties as inhibitors of TF/VIIa. [electronic resource]
Producer: 20050919Description: 3006-11 p. digitalISSN:- 0960-894X
- Benzamidines -- chemistry
- Binding Sites
- Drug Design
- Factor VIIa -- antagonists & inhibitors
- Fibrinolytic Agents -- chemical synthesis
- Inhibitory Concentration 50
- Models, Molecular
- Protein Binding
- Pyrazines -- chemical synthesis
- Serine Proteinase Inhibitors -- chemical synthesis
- Structure-Activity Relationship
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
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