Structural basis for GPR40 allosteric agonism and incretin stimulation. [electronic resource]
Producer: 20181212Description: 1645 p. digitalISSN:- 2041-1723
- Allosteric Site -- genetics
- Animals
- Benzofurans -- pharmacology
- Crystallography, X-Ray
- Diabetes Mellitus, Type 2 -- drug therapy
- Drug Synergism
- HEK293 Cells
- Humans
- Hypoglycemic Agents -- pharmacology
- Incretins -- metabolism
- Insulin -- metabolism
- Insulin Secretion
- Male
- Mice
- Mice, Inbred C57BL
- Mice, Inbred ICR
- Mice, Knockout
- Molecular Docking Simulation
- Mutagenesis, Site-Directed
- Receptors, G-Protein-Coupled -- agonists
- Recombinant Proteins -- chemistry
- Sulfones -- pharmacology
- gamma-Linolenic Acid -- metabolism
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
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