Results
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Design of selective PI3Kα inhibitors starting from a promiscuous pan kinase scaffold. [electronic resource] by
- Barlaam, Bernard
- Cosulich, Sabina
- Fitzek, Martina
- Green, Stephen
- Harris, Craig S
- Hudson, Kevin
- Lambert-van der Brempt, Christine
- Ouvry, Gilles
- Page, Ken
- Ruston, Linette
- Ward, Lara
- Delouvrié, Bénédicte
Producer: 20160422
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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4.
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Optimization of potent and selective dual mTORC1 and mTORC2 inhibitors: the discovery of AZD8055 and AZD2014. [electronic resource] by
- Pike, Kurt G
- Malagu, Karine
- Hummersone, Marc G
- Menear, Keith A
- Duggan, Heather M E
- Gomez, Sylvie
- Martin, Niall M B
- Ruston, Linette
- Pass, Sarah L
- Pass, Martin
Producer: 20140113
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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5.
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Discovery of a novel aminopyrazine series as selective PI3Kα inhibitors. [electronic resource] by
- Barlaam, Bernard
- Cosulich, Sabina
- Fitzek, Martina
- Germain, Hervé
- Green, Stephen
- Hanson, Lyndsey L
- Harris, Craig S
- Hancox, Urs
- Hudson, Kevin
- Lambert-van der Brempt, Christine
- Lamorlette, Maryannick
- Magnien, Françoise
- Ouvry, Gilles
- Page, Ken
- Ruston, Linette
- Ward, Lara
- Delouvrié, Bénédicte
Producer: 20170818
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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6.
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Discovery of AZD3147: a potent, selective dual inhibitor of mTORC1 and mTORC2. [electronic resource] by
- Pike, Kurt G
- Morris, Jeff
- Ruston, Linette
- Pass, Sarah L
- Greenwood, Ryan
- Williams, Emma J
- Demeritt, Julie
- Culshaw, Janet D
- Gill, Kristy
- Pass, Martin
- Finlay, M Raymond V
- Good, Catherine J
- Roberts, Craig A
- Currie, Gordon S
- Blades, Kevin
- Eden, Jonathan M
- Pearson, Stuart E
Producer: 20150615
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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7.
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Discovery of 4-amino-N-[(1S)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide (AZD5363), an orally bioavailable, potent inhibitor of Akt kinases. [electronic resource] by
- Addie, Matt
- Ballard, Peter
- Buttar, David
- Crafter, Claire
- Currie, Gordon
- Davies, Barry R
- Debreczeni, Judit
- Dry, Hannah
- Dudley, Philippa
- Greenwood, Ryan
- Johnson, Paul D
- Kettle, Jason G
- Lane, Clare
- Lamont, Gillian
- Leach, Andrew
- Luke, Richard W A
- Morris, Jeff
- Ogilvie, Donald
- Page, Ken
- Pass, Martin
- Pearson, Stuart
- Ruston, Linette
Producer: 20130514
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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8.
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Discovery of 1-(4-(5-(5-amino-6-(5-tert-butyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1,2,4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-one (AZD8835): A potent and selective inhibitor of PI3Kα and PI3Kδ for the treatment of cancers. [electronic resource] by
- Barlaam, Bernard
- Cosulich, Sabina
- Delouvrié, Bénédicte
- Ellston, Rebecca
- Fitzek, Martina
- Germain, Hervé
- Green, Stephen
- Hancox, Urs
- Harris, Craig S
- Hudson, Kevin
- Lambert-van der Brempt, Christine
- Lebraud, Honorine
- Magnien, Françoise
- Lamorlette, Maryannick
- Le Griffon, Antoine
- Morgentin, Rémy
- Ouvry, Gilles
- Page, Ken
- Pasquet, Georges
- Polanska, Urszula
- Ruston, Linette
- Saleh, Twana
- Vautier, Michel
- Ward, Lara
Producer: 20160718
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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9.
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Discovery and Optimization of a Novel Series of Highly Selective JAK1 Kinase Inhibitors. [electronic resource] by
- Grimster, Neil P
- Anderson, Erica
- Alimzhanov, Marat
- Bebernitz, Geraldine
- Bell, Kirsten
- Chuaqui, Claudio
- Deegan, Tracy
- Ferguson, Andrew D
- Gero, Thomas
- Harsch, Andreas
- Huszar, Dennis
- Kawatkar, Aarti
- Kettle, Jason G
- Lyne, Paul
- Read, Jon A
- Rivard Costa, Caroline
- Ruston, Linette
- Schroeder, Patricia
- Shi, Jie
- Su, Qibin
- Throner, Scott
- Toader, Dorin
- Vasbinder, Melissa
- Woessner, Richard
- Wang, Haixia
- Wu, Allan
- Ye, Minwei
- Zheng, Weijia
- Zinda, Michael
Producer: 20190618
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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10.
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Discovery of (2 [electronic resource] by
- Su, Qibin
- Banks, Erica
- Bebernitz, Geraldine
- Bell, Kirsten
- Borenstein, Cassandra F
- Chen, Huawei
- Chuaqui, Claudio E
- Deng, Nanhua
- Ferguson, Andrew D
- Kawatkar, Sameer
- Grimster, Neil P
- Ruston, Linette
- Lyne, Paul D
- Read, Jon A
- Peng, Xianyou
- Pei, Xiaohui
- Fawell, Stephen
- Tang, Zhanlei
- Throner, Scott
- Vasbinder, Melissa M
- Wang, Haoyu
- Winter-Holt, Jon
- Woessner, Richard
- Wu, Allan
- Yang, Wenzhan
- Zinda, Michael
- Kettle, Jason G
Producer: 20201102
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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