A new pyridazinone exhibits potent cytotoxicity on human cancer cells via apoptosis and poly-ubiquitinated protein accumulation. [electronic resource]
Producer: 20200901Description: 503-519 p. digitalISSN:- 1573-6822
- Antineoplastic Agents -- chemical synthesis
- Apoptosis -- drug effects
- Caspase 3 -- metabolism
- Caspases -- metabolism
- Cell Line, Tumor
- Cell Survival
- DNA Fragmentation
- Humans
- Membrane Potential, Mitochondrial -- drug effects
- Mitochondria -- metabolism
- Necrosis -- metabolism
- Neoplasms -- drug therapy
- Proto-Oncogene Proteins c-bcl-2 -- metabolism
- Pyridazines -- pharmacology
- Reactive Oxygen Species -- metabolism
- Signal Transduction
- Ubiquitinated Proteins
- bcl-2-Associated X Protein -- metabolism
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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