Expression of drug transporters and drug metabolizing enzymes in the bladder urothelium in man and affinity of the bladder spasmolytic trospium chloride to transporters likely involved in its pharmacokinetics. [electronic resource]
Producer: 20151110Description: 171-8 p. digitalISSN:- 1543-8392
- ATP Binding Cassette Transporter, Subfamily B, Member 1 -- metabolism
- Administration, Intravesical
- Administration, Oral
- Animals
- Benzilates -- pharmacokinetics
- Binding, Competitive
- Blood-Brain Barrier -- drug effects
- Dogs
- Gene Expression Regulation
- HEK293 Cells
- Humans
- Madin Darby Canine Kidney Cells
- Nortropanes -- pharmacokinetics
- Parasympatholytics -- pharmacokinetics
- Urinary Bladder -- drug effects
- Urothelium -- drug effects
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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