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Generation of 3,8-substituted 1,2,4-triazolopyridines as potent inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1). [electronic resource] by
- Wang, Haixia
- Robl, Jeffrey A
- Hamann, Lawrence G
- Simpkins, Ligaya
- Golla, Rajasree
- Li, Yi-Xin
- Seethala, Ramakrishna
- Zvyaga, Tatyana
- Gordon, David A
- Li, James J
Producer: 20111025
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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5.
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Discovery of selective imidazole-based inhibitors of mammalian 15-lipoxygenase: highly potent against human enzyme within a cellular environment. [electronic resource] by
- Weinstein, David S
- Liu, Wen
- Ngu, Khehyong
- Langevine, Charles
- Combs, Donald W
- Zhuang, Shaobin
- Chen, Cindy
- Madsen, Cort S
- Harper, Timothy W
- Robl, Jeffrey A
Producer: 20071227
In:
Bioorganic & medicinal chemistry letters vol. 17
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6.
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Pyrazole-based sulfonamide and sulfamides as potent inhibitors of mammalian 15-lipoxygenase. [electronic resource] by
- Ngu, Khehyong
- Weinstein, David S
- Liu, Wen
- Langevine, Charles
- Combs, Donald W
- Zhuang, Shaobin
- Chen, Xing
- Madsen, Cort S
- Harper, Timothy W
- Ahmad, Saleem
- Robl, Jeffrey A
Producer: 20111025
In:
Bioorganic & medicinal chemistry letters vol. 21
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7.
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A synthesis of N-bridged 5,6-bicylic pyridines via a mild cyclodehydration using the burgess reagent and discovery of a novel carbamylsulfonylation reaction. [electronic resource] by
- Li, Jie Jack
- Li, James J
- Li, Jun
- Trehan, Ashok K
- Wong, Henry S
- Krishnananthan, Subramanian
- Kennedy, Lawrence J
- Gao, Qi
- Ng, Alicia
- Robl, Jeffrey A
- Balasubramanian, Balu
- Chen, Bang-Chi
Producer: 20080916
In:
Organic letters vol. 10
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Synthesis and structure-activity relationship of dihydrobenzofuran derivatives as novel human GPR119 agonists. [electronic resource] by
- Ye, Xiang-Yang
- Morales, Christian L
- Wang, Ying
- Rossi, Karen A
- Malmstrom, Sarah E
- Abousleiman, Mojgan
- Sereda, Larisa
- Apedo, Atsu
- Robl, Jeffrey A
- Miller, Keith J
- Krupinski, John
- Wacker, Dean A
Producer: 20150102
In:
Bioorganic & medicinal chemistry letters vol. 24
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Design, synthesis, and SAR studies of novel polycyclic acids as potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1). [electronic resource] by
- Ye, Xiang-Yang
- Chen, Stephanie Y
- Nayeem, Akbar
- Golla, Rajasree
- Seethala, Ramakrishna
- Wang, Mengmeng
- Harper, Timothy
- Sleczka, Bogdan G
- Li, Yi-Xin
- He, Bin
- Kirby, Mark
- Gordon, David A
- Robl, Jeffrey A
Producer: 20120213
In:
Bioorganic & medicinal chemistry letters vol. 21
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10.
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Diprolyl nitriles as potent dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Zhao, Guohua
- Taunk, Prakash C
- Magnin, David R
- Simpkins, Ligaya M
- Robl, Jeffrey A
- Wang, Aiying
- Robertson, James G
- Marcinkeviciene, Jovita
- Sitkoff, Doree F
- Parker, Rex A
- Kirby, Mark S
- Hamann, Lawrence G
Producer: 20051121
In:
Bioorganic & medicinal chemistry letters vol. 15
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11.
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(D)-2-tert-Butoxycarbonylamino-5,5-difluoro-5-phenyl-pentanoic acid: synthesis and incorporation into the growth hormone secretagogues. [electronic resource] by
- Li, Jun
- Chen, Stephanie Y
- Murphy, Brian J
- Flynn, Neil
- Seethala, Ramakrishna
- Slusarchyk, Dorothy
- Yan, Mujing
- Sleph, Paul
- Zhang, Hongjian
- Humphreys, William G
- Ewing, William R
- Robl, Jeffrey A
- Gordon, David
- Tino, Joseph A
Producer: 20081117
In:
Bioorganic & medicinal chemistry letters vol. 18
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12.
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Treatment of diabetes and atherosclerosis by inhibiting fatty-acid-binding protein aP2. [electronic resource] by
- Furuhashi, Masato
- Tuncman, Gürol
- Görgün, Cem Z
- Makowski, Liza
- Atsumi, Genichi
- Vaillancourt, Eric
- Kono, Keita
- Babaev, Vladimir R
- Fazio, Sergio
- Linton, MacRae F
- Sulsky, Richard
- Robl, Jeffrey A
- Parker, Rex A
- Hotamisligil, Gökhan S
Producer: 20070731
In:
Nature vol. 447
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13.
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Synthesis and structure-activity relationship of 2-adamantylmethyl tetrazoles as potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1). [electronic resource] by
- Ye, Xiang-Yang
- Yoon, David
- Chen, Stephanie Y
- Nayeem, Akbar
- Golla, Rajasree
- Seethala, Ramakrishna
- Wang, Mengmeng
- Harper, Timothy
- Sleczka, Bogdan G
- Apedo, Atsu
- Li, Yi-Xin
- He, Bin
- Kirby, Mark
- Gordon, David A
- Robl, Jeffrey A
Producer: 20140826
In:
Bioorganic & medicinal chemistry letters vol. 24
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Microsomal triglyceride transfer protein inhibitors: discovery and synthesis of alkyl phosphonates as potent MTP inhibitors and cholesterol lowering agents. [electronic resource] by
- Magnin, David R
- Biller, Scott A
- Wetterau, John
- Robl, Jeffrey A
- Dickson, John K
- Taunk, Prakash
- Harrity, Thomas W
- Lawrence, R Michael
- Sun, C-Q
- Wang, Tammy
- Logan, Janette
- Fryszman, Olga
- Connolly, Fergal
- Jolibois, Kern
- Kunselman, Lori
Producer: 20031103
In:
Bioorganic & medicinal chemistry letters vol. 13
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15.
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NMR structure of a potent small molecule inhibitor bound to human keratinocyte fatty acid-binding protein. [electronic resource] by
- McDonnell, Patricia A
- Constantine, Keith L
- Goldfarb, Valentina
- Johnson, Stephen R
- Sulsky, Richard
- Magnin, David R
- Robl, Jeffrey A
- Caulfield, Thomas J
- Parker, Rex A
- Taylor, David S
- Adam, Leonard P
- Metzler, William J
- Mueller, Luciano
- Farmer, Bennett T
Producer: 20060913
In:
Journal of medicinal chemistry vol. 49
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16.
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Tetrazole based amides as growth hormone secretagogues. [electronic resource] by
- Li, James J
- Wang, Haixia
- Li, Jun
- Qu, Fucheng
- Swartz, Stephen G
- Hernández, Andrés S
- Biller, Scott A
- Robl, Jeffrey A
- Tino, Joseph A
- Slusarchyk, Dorothy
- Seethala, Ramakrishna
- Sleph, Paul
- Yan, Mujing
- Grover, Gary
- Flynn, Neil
- Murphy, Brian J
- Gordon, David
Producer: 20080516
In:
Bioorganic & medicinal chemistry letters vol. 18
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17.
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Tetrahydroisoquinoline 1-carboxamides as growth hormone secretagogues. [electronic resource] by
- Li, James J
- Wang, Haixia
- Qu, Fucheng
- Musial, Christa
- Tino, Joseph A
- Robl, Jeffrey A
- Slusarchyk, Dorothy
- Golla, Rajasree
- Seethala, Ramakrishna
- Dickinson, Kenneth
- Giupponi, Leah
- Grover, Gary
- Sleph, Paul
- Flynn, Neil
- Murphy, Brian J
- Gordon, David
- Kung, Melissa
- Stoffel, Robert
Producer: 20050805
In:
Bioorganic & medicinal chemistry letters vol. 15
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18.
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Synthesis and SAR of 2,3,3a,4-tetrahydro-1H-pyrrolo[3,4-c]isoquinolin-5(9bH)-ones as 5-HT2C receptor agonists. [electronic resource] by
- Fevig, John M
- Feng, Jianxin
- Rossi, Karen A
- Miller, Keith J
- Wu, Ginger
- Hung, Chen-Pin
- Ung, Thao
- Malmstrom, Sarah E
- Zhang, Ge
- Keim, William J
- Cullen, Mary Jane
- Rohrbach, Kenneth W
- Qu, Qinling
- Gan, Jinping
- Pelleymounter, Mary Ann
- Robl, Jeffrey A
Producer: 20130528
In:
Bioorganic & medicinal chemistry letters vol. 23
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19.
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Tricyclic dihydroquinazolinones as novel 5-HT2C selective and orally efficacious anti-obesity agents. [electronic resource] by
- Ahmad, Saleem
- Ngu, Khehyong
- Miller, Keith J
- Wu, Ginger
- Hung, Chen-pin
- Malmstrom, Sarah
- Zhang, Ge
- O'Tanyi, Eva
- Keim, William J
- Cullen, Mary Jane
- Rohrbach, Kenneth W
- Thomas, Michael
- Ung, Thao
- Qu, Qinling
- Gan, Jinping
- Narayanan, Rangaraj
- Pelleymounter, Mary Ann
- Robl, Jeffrey A
Producer: 20100920
In:
Bioorganic & medicinal chemistry letters vol. 20
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20.
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Amino(methyl) pyrrolidines as novel scaffolds for factor Xa inhibitors. [electronic resource] by
- Shi, Yan
- Sitkoff, Doree
- Zhang, Jing
- Han, Wei
- Hu, Zilun
- Stein, Philip D
- Wang, Ying
- Kennedy, Lawrence J
- O'Connor, Stephen P
- Ahmad, Saleem
- Liu, Eddie C-K
- Seiler, Steve M
- Lam, Patrick Y S
- Robl, Jeffrey A
- Macor, John E
- Atwal, Karnail S
- Zahler, Robert
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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