Results
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1.
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Receptor occupancy of nonpeptide corticotropin-releasing factor 1 antagonist DMP696: correlation with drug exposure and anxiolytic efficacy. [electronic resource] by
- Li, Yu-Wen
- Hill, Geraldine
- Wong, Harvey
- Kelly, Natasha
- Ward, Kathryn
- Pierdomenico, Marie
- Ren, Shelly
- Gilligan, Paul
- Grossman, Scott
- Trainor, George
- Taub, Rebecca
- McElroy, John
- Zazcek, Robert
Producer: 20030422
In:
The Journal of pharmacology and experimental therapeutics vol. 305
Availability: No items available.
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2.
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An orally active corticotropin releasing factor 1 receptor antagonist from 8-aryl-1,3a,7,8-tetraaza-cyclopenta[a]indenes. [electronic resource] by
- Han, Xiaojun
- Civiello, Rita
- Pin, Sokhom S
- Burris, Kevin
- Balanda, Lynn A
- Knipe, Jay
- Ren, Shelly
- Fiedler, Tracey
- Browman, Kaitlin E
- Macci, Robert
- Taber, Matthew T
- Zhang, Jie
- Dubowchik, Gene M
Producer: 20070725
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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3.
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The synthesis and SAR of calcitonin gene-related peptide (CGRP) receptor antagonists derived from tyrosine surrogates. Part 1. [electronic resource] by
- Han, Xiaojun
- Civiello, Rita L
- Conway, Charles M
- Cook, Deborah A
- Davis, Carl D
- Macci, Robert
- Pin, Sokhom S
- Ren, Shelly X
- Schartman, Richard
- Signor, Laura J
- Thalody, George
- Widmann, Kimberly A
- Xu, Cen
- Chaturvedula, Prasad V
- Macor, John E
- Dubowchik, Gene M
Producer: 20130104
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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4.
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Discovery of (R)-4-(8-fluoro-2-oxo-1,2-dihydroquinazolin-3(4H)-yl)-N-(3-(7-methyl-1H-indazol-5-yl)-1-oxo-1-(4-(piperidin-1-yl)piperidin-1-yl)propan-2-yl)piperidine-1-carboxamide (BMS-694153): a potent antagonist of the human calcitonin gene-related peptide receptor for migraine with rapid and efficient intranasal exposure. [electronic resource] by
- Degnan, Andrew P
- Chaturvedula, Prasad V
- Conway, Charles M
- Cook, Deborah A
- Davis, Carl D
- Denton, Rex
- Han, Xiaojun
- Macci, Robert
- Mathias, Neil R
- Moench, Paul
- Pin, Sokhom S
- Ren, Shelly X
- Schartman, Richard
- Signor, Laura J
- Thalody, George
- Widmann, Kimberly A
- Xu, Cen
- Macor, John E
- Dubowchik, Gene M
Producer: 20080910
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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5.
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Anxiolytic-like effects of the corticotropin-releasing factor1 (CRF1) antagonist DMP904 [4-(3-pentylamino)-2,7-dimethyl-8-(2-methyl-4-methoxyphenyl)-pyrazolo-[1,5-a]-pyrimidine] administered acutely or chronically at doses occupying central CRF1 receptors in rats. [electronic resource] by
- Lelas, Snjezana
- Wong, Harvey
- Li, Yu-Wen
- Heman, Karen L
- Ward, Kathryn A
- Zeller, Kim L
- Sieracki, Kristine K
- Polino, Joseph L
- Godonis, Helen E
- Ren, Shelly X
- Yan, Xiao-Xin
- Arneric, Stephen P
- Robertson, David W
- Hartig, Paul R
- Grossman, Scott
- Trainor, George L
- Taub, Rebecca A
- Zaczek, Robert
- Gilligan, Paul J
- McElroy, John F
Producer: 20040504
In:
The Journal of pharmacology and experimental therapeutics vol. 309
Availability: No items available.
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6.
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N-in-1 dosing pharmacokinetics in drug discovery: experience, theoretical and practical considerations. [electronic resource] by
- He, Kan
- Qian, Mingxin
- Wong, Harvey
- Bai, Stephen A
- He, Bing
- Brogdon, Bernice
- Grace, James E
- Xin, Baomin
- Wu, Jingtao
- Ren, Shelly X
- Zeng, Hang
- Deng, Yuzhong
- Graden, Danielle M
- Olah, Timothy V
- Unger, Steve E
- Luettgen, Joseph M
- Knabb, Robert M
- Pinto, Donald J
- Lam, Patrick Y S
- Duan, James
- Wexler, Ruth R
- Decicco, Carl P
- Christ, David D
- Grossman, Scott J
Producer: 20081009
In:
Journal of pharmaceutical sciences vol. 97
Availability: No items available.
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