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Anthracene-polyamine conjugates inhibit in vitro proliferation of intraerythrocytic Plasmodium falciparum parasites. [electronic resource] by
- Niemand, Jandeli
- Burger, Pieter
- Verlinden, Bianca K
- Reader, Janette
- Joubert, Annie M
- Kaiser, Annette
- Louw, Abraham I
- Kirk, Kiaran
- Phanstiel, Otto
- Birkholtz, Lyn-Marie
Producer: 20131025
In:
Antimicrobial agents and chemotherapy vol. 57
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4.
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Nowhere to hide: interrogating different metabolic parameters of Plasmodium falciparum gametocytes in a transmission blocking drug discovery pipeline towards malaria elimination. [electronic resource] by
- Reader, Janette
- Botha, Mariëtte
- Theron, Anjo
- Lauterbach, Sonja B
- Rossouw, Claire
- Engelbrecht, Dewaldt
- Wepener, Melanie
- Smit, Annél
- Leroy, Didier
- Mancama, Dalu
- Coetzer, Theresa L
- Birkholtz, Lyn-Marie
Producer: 20160216
In:
Malaria journal vol. 14
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Activities of 11-Azaartemisinin and N-Sulfonyl Derivatives against Asexual and Transmissible Malaria Parasites. [electronic resource] by
- Harmse, Rozanne
- Coertzen, Dina
- Wong, Ho Ning
- Smit, Frans J
- van der Watt, Mariette E
- Reader, Janette
- Nondaba, Sindiswe H
- Birkholtz, Lyn-Marie
- Haynes, Richard K
- N'Da, David D
Producer: 20171225
In:
ChemMedChem vol. 12
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6.
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Interrogating alkyl and arylalkylpolyamino (bis)urea and (bis)thiourea isosteres as potent antimalarial chemotypes against multiple lifecycle forms of Plasmodium falciparum parasites. [electronic resource] by
- Verlinden, Bianca K
- de Beer, Marna
- Pachaiyappan, Boobalan
- Besaans, Ethan
- Andayi, Warren A
- Reader, Janette
- Niemand, Jandeli
- van Biljon, Riette
- Guy, Kiplin
- Egan, Timothy
- Woster, Patrick M
- Birkholtz, Lyn-Marie
Producer: 20160512
In:
Bioorganic & medicinal chemistry vol. 23
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Inducing controlled cell cycle arrest and re-entry during asexual proliferation of Plasmodium falciparum malaria parasites. [electronic resource] by
- van Biljon, Riëtte
- Niemand, Jandeli
- van Wyk, Roelof
- Clark, Katherine
- Verlinden, Bianca
- Abrie, Clarissa
- von Grüning, Hilde
- Smidt, Werner
- Smit, Annél
- Reader, Janette
- Painter, Heather
- Llinás, Manuel
- Doerig, Christian
- Birkholtz, Lyn-Marié
Producer: 20191028
In:
Scientific reports vol. 8
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8.
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Optimal 10-Aminoartemisinins With Potent Transmission-Blocking Capabilities for New Artemisinin Combination Therapies-Activities Against Blood Stage [electronic resource] by
- Wong, Ho Ning
- Padín-Irizarry, Vivian
- van der Watt, Mariëtte E
- Reader, Janette
- Liebenberg, Wilna
- Wiesner, Lubbe
- Smith, Peter
- Eribez, Korina
- Winzeler, Elizabeth A
- Kyle, Dennis E
- Birkholtz, Lyn-Marie
- Coertzen, Dina
- Haynes, Richard K
Publication details: Frontiers in chemistry 2019
In:
Frontiers in chemistry vol. 7
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9.
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Artemisone and Artemiside Are Potent Panreactive Antimalarial Agents That Also Synergize Redox Imbalance in Plasmodium falciparum Transmissible Gametocyte Stages. [electronic resource] by
- Coertzen, Dina
- Reader, Janette
- van der Watt, Mariëtte
- Nondaba, Sindisiwe H
- Gibhard, Liezl
- Wiesner, Lubbe
- Smith, Peter
- D'Alessandro, Sarah
- Taramelli, Donatella
- Wong, Ho Ning
- du Preez, Jan L
- Wu, Ronald Wai Keung
- Birkholtz, Lyn-Marie
- Haynes, Richard K
Producer: 20190923
In:
Antimicrobial agents and chemotherapy vol. 62
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Discovery of compounds blocking the proliferation of Toxoplasma gondii and Plasmodium falciparum in a chemical space based on piperidinyl-benzimidazolone analogs. [electronic resource] by
- Saïdani, Nadia
- Botté, Cyrille Y
- Deligny, Michael
- Bonneau, Anne-Laure
- Reader, Janette
- Lasselin, Ronald
- Merer, Goulven
- Niepceron, Alisson
- Brossier, Fabien
- Cintrat, Jean-Christophe
- Rousseau, Bernard
- Birkholtz, Lyn-Marie
- Cesbron-Delauw, Marie-France
- Dubremetz, Jean-François
- Mercier, Corinne
- Vial, Henri
- Lopez, Roman
- Maréchal, Eric
Producer: 20150515
In:
Antimicrobial agents and chemotherapy vol. 58
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11.
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Structure-Activity Relationship Studies and Plasmodium Life Cycle Profiling Identifies Pan-Active N-Aryl-3-trifluoromethyl Pyrido[1,2- a]benzimidazoles Which Are Efficacious in an in Vivo Mouse Model of Malaria. [electronic resource] by
- Mayoka, Godfrey
- Njoroge, Mathew
- Okombo, John
- Gibhard, Liezl
- Sanches-Vaz, Margarida
- Fontinha, Diana
- Birkholtz, Lyn-Marie
- Reader, Janette
- van der Watt, Mariëtte
- Coetzer, Theresa L
- Lauterbach, Sonja
- Churchyard, Alisje
- Bezuidenhout, Belinda
- Egan, Timothy J
- Yeates, Clive
- Wittlin, Sergio
- Prudêncio, Miguel
- Chibale, Kelly
Producer: 20191017
In:
Journal of medicinal chemistry vol. 62
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Multistage Antiplasmodium Activity of Astemizole Analogues and Inhibition of Hemozoin Formation as a Contributor to Their Mode of Action. [electronic resource] by
- Kumar, Malkeet
- Okombo, John
- Mambwe, Dickson
- Taylor, Dale
- Lawrence, Nina
- Reader, Janette
- van der Watt, Mariëtte
- Fontinha, Diana
- Sanches-Vaz, Margarida
- Bezuidenhout, Belinda C
- Lauterbach, Sonja B
- Liebenberg, Dale
- Birkholtz, Lyn-Marie
- Coetzer, Theresa L
- Prudêncio, Miguel
- Egan, Timothy J
- Wittlin, Sergio
- Chibale, Kelly
Producer: 20191212
In:
ACS infectious diseases vol. 5
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13.
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Antimalarial Pyrido[1,2-a]benzimidazoles: Lead Optimization, Parasite Life Cycle Stage Profile, Mechanistic Evaluation, Killing Kinetics, and in Vivo Oral Efficacy in a Mouse Model. [electronic resource] by
- Singh, Kawaljit
- Okombo, John
- Brunschwig, Christel
- Ndubi, Ferdinand
- Barnard, Linley
- Wilkinson, Chad
- Njogu, Peter M
- Njoroge, Mathew
- Laing, Lizahn
- Machado, Marta
- Prudêncio, Miguel
- Reader, Janette
- Botha, Mariette
- Nondaba, Sindisiwe
- Birkholtz, Lyn-Marie
- Lauterbach, Sonja
- Churchyard, Alisje
- Coetzer, Theresa L
- Burrows, Jeremy N
- Yeates, Clive
- Denti, Paolo
- Wiesner, Lubbe
- Egan, Timothy J
- Wittlin, Sergio
- Chibale, Kelly
Producer: 20170616
In:
Journal of medicinal chemistry vol. 60
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14.
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A Novel Pyrazolopyridine with in Vivo Activity in Plasmodium berghei- and Plasmodium falciparum-Infected Mouse Models from Structure-Activity Relationship Studies around the Core of Recently Identified Antimalarial Imidazopyridazines. [electronic resource] by
- Le Manach, Claire
- Paquet, Tanya
- Brunschwig, Christel
- Njoroge, Mathew
- Han, Ze
- Gonzàlez Cabrera, Diego
- Bashyam, Sridevi
- Dhinakaran, Rajkumar
- Taylor, Dale
- Reader, Janette
- Botha, Mariette
- Churchyard, Alisje
- Lauterbach, Sonja
- Coetzer, Theresa L
- Birkholtz, Lyn-Marie
- Meister, Stephan
- Winzeler, Elizabeth A
- Waterson, David
- Witty, Michael J
- Wittlin, Sergio
- Jiménez-Díaz, María-Belén
- Santos Martínez, María
- Ferrer, Santiago
- Angulo-Barturen, Iñigo
- Street, Leslie J
- Chibale, Kelly
Producer: 20160225
In:
Journal of medicinal chemistry vol. 58
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15.
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Potent Plasmodium falciparum gametocytocidal compounds identified by exploring the kinase inhibitor chemical space for dual active antimalarials. [electronic resource] by
- van der Watt, Mariëtte E
- Reader, Janette
- Churchyard, Alisje
- Nondaba, Sindisiwe H
- Lauterbach, Sonja B
- Niemand, Jandeli
- Abayomi, Sijuade
- van Biljon, Riëtte A
- Connacher, Jessica I
- van Wyk, Roelof D J
- Le Manach, Claire
- Paquet, Tanya
- González Cabrera, Diego
- Brunschwig, Christel
- Theron, Anjo
- Lozano-Arias, Sonia
- Rodrigues, Janneth F I
- Herreros, Esperanza
- Leroy, Didier
- Duffy, James
- Street, Leslie J
- Chibale, Kelly
- Mancama, Dalu
- Coetzer, Theresa L
- Birkholtz, Lyn-Marie
Producer: 20190626
In:
The Journal of antimicrobial chemotherapy vol. 73
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16.
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Identification of a Potential Antimalarial Drug Candidate from a Series of 2-Aminopyrazines by Optimization of Aqueous Solubility and Potency across the Parasite Life Cycle. [electronic resource] by
- Le Manach, Claire
- Nchinda, Aloysius T
- Paquet, Tanya
- Gonzàlez Cabrera, Diego
- Younis, Yassir
- Han, Ze
- Bashyam, Sridevi
- Zabiulla, Mohammed
- Taylor, Dale
- Lawrence, Nina
- White, Karen L
- Charman, Susan A
- Waterson, David
- Witty, Michael J
- Wittlin, Sergio
- Botha, Mariëtte E
- Nondaba, Sindisiswe H
- Reader, Janette
- Birkholtz, Lyn-Marie
- Jiménez-Díaz, María Belén
- Martínez, María Santos
- Ferrer, Santiago
- Angulo-Barturen, Iñigo
- Meister, Stephan
- Antonova-Koch, Yevgeniya
- Winzeler, Elizabeth A
- Street, Leslie J
- Chibale, Kelly
Producer: 20170608
In:
Journal of medicinal chemistry vol. 59
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17.
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Erratum for Brunschwig et al., "UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of Malaria". [electronic resource] by
- Brunschwig, Christel
- Lawrence, Nina
- Taylor, Dale
- Abay, Efrem
- Njoroge, Mathew
- Basarab, Gregory S
- Le Manach, Claire
- Paquet, Tanya
- Gonzàlez Cabrera, Diego
- Nchinda, Aloysius T
- de Kock, Carmen
- Wiesner, Lubbe
- Denti, Paolo
- Waterson, David
- Blasco, Benjamin
- Leroy, Didier
- Witty, Michael J
- Donini, Cristina
- Duffy, James
- Wittlin, Sergio
- White, Karen L
- Charman, Susan A
- Jiménez-Díaz, Maria Belén
- Angulo-Barturen, Iñigo
- Herreros, Esperanza
- Gamo, Francisco Javier
- Rochford, Rosemary
- Mancama, Dalu
- Coetzer, Theresa L
- van der Watt, Mariëtte E
- Reader, Janette
- Birkholtz, Lyn-Marie
- Marsh, Kennan C
- Solapure, Suresh M
- Burke, John E
- McPhail, Jacob A
- Vanaerschot, Manu
- Fidock, David A
- Fish, Paul V
- Siegl, Peter
- Smith, Dennis A
- Wirjanata, Grennady
- Noviyanti, Rintis
- Price, Ric N
- Marfurt, Jutta
- Silue, Kigbafori D
- Street, Leslie J
- Chibale, Kelly
Publication details: Antimicrobial agents and chemotherapy 11 2018
In:
Antimicrobial agents and chemotherapy vol. 62
Availability: No items available.
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18.
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UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of Malaria. [electronic resource] by
- Brunschwig, Christel
- Lawrence, Nina
- Taylor, Dale
- Abay, Efrem
- Njoroge, Mathew
- Basarab, Gregory S
- Le Manach, Claire
- Paquet, Tanya
- Cabrera, Diego Gonzàlez
- Nchinda, Aloysius T
- de Kock, Carmen
- Wiesner, Lubbe
- Denti, Paolo
- Waterson, David
- Blasco, Benjamin
- Leroy, Didier
- Witty, Michael J
- Donini, Cristina
- Duffy, James
- Wittlin, Sergio
- White, Karen L
- Charman, Susan A
- Jiménez-Díaz, Maria Belén
- Angulo-Barturen, Iñigo
- Herreros, Esperanza
- Gamo, Francisco Javier
- Rochford, Rosemary
- Mancama, Dalu
- Coetzer, Theresa L
- van der Watt, Mariëtte E
- Reader, Janette
- Birkholtz, Lyn-Marie
- Marsh, Kennan C
- Solapure, Suresh M
- Burke, John E
- McPhail, Jacob A
- Vanaerschot, Manu
- Fidock, David A
- Fish, Paul V
- Siegl, Peter
- Smith, Dennis A
- Wirjanata, Grennady
- Noviyanti, Rintis
- Price, Ric N
- Marfurt, Jutta
- Silue, Kigbafori D
- Street, Leslie J
- Chibale, Kelly
Producer: 20190926
In:
Antimicrobial agents and chemotherapy vol. 62
Availability: No items available.
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19.
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Antimalarial efficacy of MMV390048, an inhibitor of [electronic resource] by
- Paquet, Tanya
- Le Manach, Claire
- Cabrera, Diego González
- Younis, Yassir
- Henrich, Philipp P
- Abraham, Tara S
- Lee, Marcus C S
- Basak, Rajshekhar
- Ghidelli-Disse, Sonja
- Lafuente-Monasterio, María José
- Bantscheff, Marcus
- Ruecker, Andrea
- Blagborough, Andrew M
- Zakutansky, Sara E
- Zeeman, Anne-Marie
- White, Karen L
- Shackleford, David M
- Mannila, Janne
- Morizzi, Julia
- Scheurer, Christian
- Angulo-Barturen, Iñigo
- Martínez, María Santos
- Ferrer, Santiago
- Sanz, Laura María
- Gamo, Francisco Javier
- Reader, Janette
- Botha, Mariette
- Dechering, Koen J
- Sauerwein, Robert W
- Tungtaeng, Anchalee
- Vanachayangkul, Pattaraporn
- Lim, Chek Shik
- Burrows, Jeremy
- Witty, Michael J
- Marsh, Kennan C
- Bodenreider, Christophe
- Rochford, Rosemary
- Solapure, Suresh M
- Jiménez-Díaz, María Belén
- Wittlin, Sergio
- Charman, Susan A
- Donini, Cristina
- Campo, Brice
- Birkholtz, Lyn-Marie
- Hanson, Kirsten K
- Drewes, Gerard
- Kocken, Clemens H M
- Delves, Michael J
- Leroy, Didier
- Fidock, David A
- Waterson, David
- Street, Leslie J
- Chibale, Kelly
Producer: 20180212
In:
Science translational medicine vol. 9
Availability: No items available.
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