Results
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X-ray Characterization and Structure-Based Optimization of Striatal-Enriched Protein Tyrosine Phosphatase Inhibitors. [electronic resource] by
- Witten, Michael R
- Wissler, Lisa
- Snow, Melanie
- Geschwindner, Stefan
- Read, Jon A
- Brandon, Nicholas J
- Nairn, Angus C
- Lombroso, Paul J
- Käck, Helena
- Ellman, Jonathan A
Producer: 20180123
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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Mapping the sugar dependency for rational generation of a DNA-RNA hybrid-guided Cas9 endonuclease. [electronic resource] by
- Rueda, Fernando Orden
- Bista, Michal
- Newton, Matthew D
- Goeppert, Anne U
- Cuomo, M Emanuela
- Gordon, Euan
- Kröner, Felix
- Read, Jon A
- Wrigley, Jonathan D
- Rueda, David
- Taylor, Benjamin J M
Producer: 20180914
In:
Nature communications vol. 8
Availability: No items available.
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Discovery of 1-methyl-1H-imidazole derivatives as potent Jak2 inhibitors. [electronic resource] by
- Su, Qibin
- Ioannidis, Stephanos
- Chuaqui, Claudio
- Almeida, Lynsie
- Alimzhanov, Marat
- Bebernitz, Geraldine
- Bell, Kirsten
- Block, Michael
- Howard, Tina
- Huang, Shan
- Huszar, Dennis
- Read, Jon A
- Rivard Costa, Caroline
- Shi, Jie
- Su, Mei
- Ye, Minwei
- Zinda, Michael
Producer: 20140310
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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5.
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Rapid Identification of Novel Allosteric PRC2 Inhibitors. [electronic resource] by
- Read, Jon A
- Tart, Jonathan
- Rawlins, Philip B
- Gregson, Clare
- Jones, Karen
- Gao, Ning
- Zhu, Xiahui
- Tomlinson, Ron
- Code, Erin
- Cheung, Tony
- Chen, Huawei
- Kawatkar, Sameer P
- Bloecher, Andy
- Bagal, Sharan
- O'Donovan, Daniel H
- Robinson, James
Producer: 20200407
In:
ACS chemical biology vol. 14
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Adventures in Scaffold Morphing: Discovery of Fused Ring Heterocyclic Checkpoint Kinase 1 (CHK1) Inhibitors. [electronic resource] by
- Yang, Bin
- Vasbinder, Melissa M
- Hird, Alexander W
- Su, Qibin
- Wang, Haixia
- Yu, Yan
- Toader, Dorin
- Lyne, Paul D
- Read, Jon A
- Breed, Jason
- Ioannidis, Stephanos
- Deng, Chun
- Grondine, Michael
- DeGrace, Nancy
- Whitston, David
- Brassil, Patrick
- Janetka, James W
Producer: 20190218
In:
Journal of medicinal chemistry vol. 61
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Methyl-thiazoles: a novel mode of inhibition with the potential to develop novel inhibitors targeting InhA in Mycobacterium tuberculosis. [electronic resource] by
- Shirude, Pravin S
- Madhavapeddi, Prashanti
- Naik, Maruti
- Murugan, Kannan
- Shinde, Vikas
- Nandishaiah, Radha
- Bhat, Jyothi
- Kumar, Anupriya
- Hameed, Shahul
- Holdgate, Geoffrey
- Davies, Gareth
- McMiken, Helen
- Hegde, Naina
- Ambady, Anisha
- Venkatraman, Janani
- Panda, Manoranjan
- Bandodkar, Balachandra
- Sambandamurthy, Vasan K
- Read, Jon A
Producer: 20140318
In:
Journal of medicinal chemistry vol. 56
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Discovery of cofactor-specific, bactericidal Mycobacterium tuberculosis InhA inhibitors using DNA-encoded library technology. [electronic resource] by
- Soutter, Holly H
- Centrella, Paolo
- Clark, Matthew A
- Cuozzo, John W
- Dumelin, Christoph E
- Guie, Marie-Aude
- Habeshian, Sevan
- Keefe, Anthony D
- Kennedy, Kaitlyn M
- Sigel, Eric A
- Troast, Dawn M
- Zhang, Ying
- Ferguson, Andrew D
- Davies, Gareth
- Stead, Eleanor R
- Breed, Jason
- Madhavapeddi, Prashanti
- Read, Jon A
Producer: 20180403
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 113
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Recurrent MLK4 Loss-of-Function Mutations Suppress JNK Signaling to Promote Colon Tumorigenesis. [electronic resource] by
- Marusiak, Anna A
- Stephenson, Natalie L
- Baik, Hayeon
- Trotter, Eleanor W
- Li, Yaoyong
- Blyth, Karen
- Mason, Susan
- Chapman, Phil
- Puto, Lorena A
- Read, Jon A
- Brassington, Claire
- Pollard, Hannah K
- Phillips, Chris
- Green, Isabelle
- Overman, Ross
- Collier, Matthew
- Testoni, Ewelina
- Miller, Crispin J
- Hunter, Tony
- Sansom, Owen J
- Brognard, John
Producer: 20160628
In:
Cancer research vol. 76
Availability: No items available.
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AMPK activation protects against diet induced obesity through Ucp1-independent thermogenesis in subcutaneous white adipose tissue. [electronic resource] by
- Pollard, Alice E
- Martins, Luís
- Muckett, Phillip J
- Khadayate, Sanjay
- Bornot, Aurélie
- Clausen, Maryam
- Admyre, Therese
- Bjursell, Mikael
- Fiadeiro, Rebeca
- Wilson, Laura
- Whilding, Chad
- Kotiadis, Vassilios N
- Duchen, Michael R
- Sutton, Daniel
- Penfold, Lucy
- Sardini, Alessandro
- Bohlooly-Y, Mohammad
- Smith, David M
- Read, Jon A
- Snowden, Michael A
- Woods, Angela
- Carling, David
Producer: 20210119
In:
Nature metabolism vol. 1
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Discovery of AZ0108, an orally bioavailable phthalazinone PARP inhibitor that blocks centrosome clustering. [electronic resource] by
- Johannes, Jeffrey W
- Almeida, Lynsie
- Daly, Kevin
- Ferguson, Andrew D
- Grosskurth, Shaun E
- Guan, Huiping
- Howard, Tina
- Ioannidis, Stephanos
- Kazmirski, Steven
- Lamb, Michelle L
- Larsen, Nicholas A
- Lyne, Paul D
- Mikule, Keith
- Ogoe, Claude
- Peng, Bo
- Petteruti, Philip
- Read, Jon A
- Su, Nancy
- Sylvester, Mark
- Throner, Scott
- Wang, Wenxian
- Wang, Xin
- Wu, Jiaquan
- Ye, Qing
- Yu, Yan
- Zheng, Xiaolan
- Scott, David A
Producer: 20160829
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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12.
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Discovery of (2 [electronic resource] by
- Su, Qibin
- Banks, Erica
- Bebernitz, Geraldine
- Bell, Kirsten
- Borenstein, Cassandra F
- Chen, Huawei
- Chuaqui, Claudio E
- Deng, Nanhua
- Ferguson, Andrew D
- Kawatkar, Sameer
- Grimster, Neil P
- Ruston, Linette
- Lyne, Paul D
- Read, Jon A
- Peng, Xianyou
- Pei, Xiaohui
- Fawell, Stephen
- Tang, Zhanlei
- Throner, Scott
- Vasbinder, Melissa M
- Wang, Haoyu
- Winter-Holt, Jon
- Woessner, Richard
- Wu, Allan
- Yang, Wenzhan
- Zinda, Michael
- Kettle, Jason G
Producer: 20201102
In:
Journal of medicinal chemistry vol. 63
Availability: No items available.
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13.
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Discovery and Optimization of a Novel Series of Highly Selective JAK1 Kinase Inhibitors. [electronic resource] by
- Grimster, Neil P
- Anderson, Erica
- Alimzhanov, Marat
- Bebernitz, Geraldine
- Bell, Kirsten
- Chuaqui, Claudio
- Deegan, Tracy
- Ferguson, Andrew D
- Gero, Thomas
- Harsch, Andreas
- Huszar, Dennis
- Kawatkar, Aarti
- Kettle, Jason G
- Lyne, Paul
- Read, Jon A
- Rivard Costa, Caroline
- Ruston, Linette
- Schroeder, Patricia
- Shi, Jie
- Su, Qibin
- Throner, Scott
- Toader, Dorin
- Vasbinder, Melissa
- Woessner, Richard
- Wang, Haixia
- Wu, Allan
- Ye, Minwei
- Zheng, Weijia
- Zinda, Michael
Producer: 20190618
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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