Results
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1.
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Comparative structure-activity relationship studies of 1-(5-methylsulfonylpyrid-2-yl)-5-alkyl and (hetero)aryl triazoles and pyrazoles in canine COX inhibition. [electronic resource] by
- Sakya, Subas M
- Shavnya, Andrei
- Cheng, Hengmiao
- Li, Chao
- Rast, Bryson
- Li, Jin
- Koss, David A
- Jaynes, Burton H
- Mann, Donald W
- Petras, Carol F
- Seibel, Scott B
- Haven, Michelle L
- Lynch, Michael P
Producer: 20080324
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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2.
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5-Heteroatom substituted pyrazoles as canine COX-2 inhibitors. Part III: molecular modeling studies on binding contribution of 1-(5-methylsulfonyl)pyrid-2-yl and 4-nitrile. [electronic resource] by
- Sakya, Subas M
- Hou, Xinjun
- Minich, Martha L
- Rast, Bryson
- Shavnya, Andrei
- DeMello, Kristin M L
- Cheng, Hengmiao
- Li, Jin
- Jaynes, Burton H
- Mann, Donald W
- Petras, Carol F
- Seibel, Scott B
- Haven, Michelle L
Producer: 20070413
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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3.
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The discovery of furo[2,3-c]pyridine-based indanone oximes as potent and selective B-Raf inhibitors. [electronic resource] by
- Buckmelter, Alex J
- Ren, Li
- Laird, Ellen R
- Rast, Bryson
- Miknis, Greg
- Wenglowsky, Steve
- Schlachter, Stephen
- Welch, Mike
- Tarlton, Eugene
- Grina, Jonas
- Lyssikatos, Joseph
- Brandhuber, Barbara J
- Morales, Tony
- Randolph, Nikole
- Vigers, Guy
- Martinson, Matthew
- Callejo, Michele
Producer: 20110523
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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4.
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Non-oxime inhibitors of B-Raf(V600E) kinase. [electronic resource] by
- Ren, Li
- Wenglowsky, Steve
- Miknis, Greg
- Rast, Bryson
- Buckmelter, Alex J
- Ely, Robert J
- Schlachter, Stephen
- Laird, Ellen R
- Randolph, Nikole
- Callejo, Michele
- Martinson, Matthew
- Galbraith, Sarah
- Brandhuber, Barbara J
- Vigers, Guy
- Morales, Tony
- Voegtli, Walter C
- Lyssikatos, Joseph
Producer: 20110523
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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5.
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5-Heteroatom-substituted pyrazoles as canine COX-2 inhibitors: Part 2. Structure-activity relationship studies of 5-alkylethers and 5-thioethers. [electronic resource] by
- Sakya, Subas M
- Cheng, Hengmiao
- Lundy Demello, Kristin M
- Shavnya, Andrei
- Minich, Martha L
- Rast, Bryson
- Dutra, Jason
- Li, Chao
- Rafka, Robert J
- Koss, David A
- Li, Jin
- Jaynes, Burton H
- Ziegler, Carl B
- Mann, Donald W
- Petras, Carol F
- Seibel, Scott B
- Silvia, Annette M
- George, David M
- Hickman, Anne
- Haven, Michelle L
- Lynch, Michael P
Producer: 20060323
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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6.
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5-heteroatom substituted pyrazoles as canine COX-2 inhibitors. Part 1: Structure-activity relationship studies of 5-alkylamino pyrazoles and discovery of a potent, selective, and orally active analog. [electronic resource] by
- Sakya, Subas M
- DeMello, Kristin M Lundy
- Minich, Martha L
- Rast, Bryson
- Shavnya, Andrei
- Rafka, Robert J
- Koss, David A
- Cheng, Hengmiao
- Li, Jin
- Jaynes, Burton H
- Ziegler, Carl B
- Mann, Donald W
- Petras, Carol F
- Seibel, Scott B
- Silvia, Annette M
- George, David M
- Lund, Lisa A
- St Denis, Suzanne
- Hickman, Anne
- Haven, Michelle L
- Lynch, Michael P
Producer: 20060302
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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7.
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Discovery of a potent, selective and orally active canine COX-2 inhibitor, 2-(3-difluoromethyl-5-phenyl-pyrazol-1-yl)-5-methanesulfonyl-pyridine. [electronic resource] by
- Li, Jin
- DeMello, Kristin M Lundy
- Cheng, Henry
- Sakya, Subas M
- Bronk, Brian S
- Rafka, Robert J
- Jaynes, Burton H
- Ziegler, Carl B
- Kilroy, Carolyn
- Mann, Donald W
- Nimz, Eric L
- Lynch, Michael P
- Haven, Michelle L
- Kolosko, Nicole L
- Minich, Martha L
- Li, Chao
- Dutra, Jason K
- Rast, Bryson
- Crosson, Rhonda M
- Morton, Barry J
- Kirk, Glen W
- Callaghan, Kathleen M
- Koss, David A
- Shavnya, Andrei
- Lund, Lisa A
- Seibel, Scott B
- Petras, Carol F
- Silvia, Annette
Producer: 20040827
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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