In vitro and in vivo metabolism of a novel cannabinoid-1 receptor inverse agonist, taranabant, in rats and monkeys. [electronic resource]
Producer: 20110602Description: 650-62 p. digitalISSN:- 1366-5928
- Amides -- blood
- Animals
- Antibodies, Monoclonal -- pharmacology
- Body Fluids -- metabolism
- Brain -- drug effects
- Drug Inverse Agonism
- Female
- Haplorhini
- Humans
- Ketoconazole -- pharmacology
- Magnetic Resonance Spectroscopy
- Male
- Mass Spectrometry
- Microsomes, Liver -- drug effects
- Pyridines -- blood
- Radioactivity
- Rats
- Receptor, Cannabinoid, CB1 -- agonists
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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