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Compelling P1 substituent affect on metalloprotease binding profile enables the design of a novel cyclohexyl core scaffold with excellent MMP selectivity and HER-2 sheddase inhibition. [electronic resource] by
- Burns, David M
- Li, Yun-Long
- Shi, Eric
- He, Chunhong
- Xu, Meizhong
- Zhuo, Jincong
- Zhang, Colin
- Qian, Ding-Quan
- Li, Yanlong
- Wynn, Richard
- Covington, Maryanne B
- Katiyar, Kamna
- Marando, Cindy A
- Fridman, Jordan S
- Scherle, Peggy
- Friedman, Steve
- Metcalf, Brian
- Yao, Wenqing
Producer: 20090901
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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4.
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INCB38579, a novel and potent histamine H₄ receptor small molecule antagonist with anti-inflammatory pain and anti-pruritic functions. [electronic resource] by
- Shin, Niu
- Covington, Maryanne
- Bian, Di
- Zhuo, Jincong
- Bowman, Kevin
- Li, Yanlong
- Soloviev, Maxim
- Qian, Ding-Quan
- Feldman, Patricia
- Leffet, Lynn
- He, Xin
- He Wang, Kathy
- Krug, Kristin
- Bell, Dan
- Czerniak, Philip
- Hu, Zhijing
- Zhao, Hui
- Zhang, Jing
- Yeleswaram, Swamy
- Yao, Wenqing
- Newton, Robert
- Scherle, Peggy
Producer: 20120504
In:
European journal of pharmacology vol. 675
Availability: No items available.
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5.
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Design and identification of selective HER-2 sheddase inhibitors via P1' manipulation and unconventional P2' perturbations to induce a molecular metamorphosis. [electronic resource] by
- Yao, Wenqing
- Zhuo, Jincong
- Burns, David M
- Li, Yun-Long
- Qian, Ding-Quan
- Zhang, Colin
- He, Chunhong
- Xu, Meizhong
- Shi, Eric
- Li, Yanlong
- Marando, Cindy A
- Covington, Maryanne B
- Yang, Gengjie
- Liu, Xiangdong
- Pan, Max
- Fridman, Jordan S
- Scherle, Peggy
- Wasserman, Zelda R
- Hollis, Gregory
- Vaddi, Kris
- Yeleswaram, Swamy
- Newton, Robert
- Friedman, Steve
- Metcalf, Brian
Producer: 20080212
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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6.
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Identification of ADAM10 as a major source of HER2 ectodomain sheddase activity in HER2 overexpressing breast cancer cells. [electronic resource] by
- Liu, Phillip C C
- Liu, Xiangdong
- Li, Yanlong
- Covington, Maryanne
- Wynn, Richard
- Huber, Reid
- Hillman, Milton
- Yang, Gengjie
- Ellis, Dawn
- Marando, Cindy
- Katiyar, Kamna
- Bradley, Jodi
- Abremski, Kenneth
- Stow, Mark
- Rupar, Mark
- Zhuo, Jincong
- Li, Yun-Long
- Lin, Qiyan
- Burns, David
- Xu, Meizhong
- Zhang, Colin
- Qian, Ding-Quan
- He, Chunhong
- Sharief, Vaqar
- Weng, Lingkai
- Agrios, Costas
- Shi, Eric
- Metcalf, Brian
- Newton, Robert
- Friedman, Steven
- Yao, Wenqing
- Scherle, Peggy
- Hollis, Gregory
- Burn, Timothy C
Producer: 20070129
In:
Cancer biology & therapy vol. 5
Availability: No items available.
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7.
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Discovery of a potent, selective, and orally active human epidermal growth factor receptor-2 sheddase inhibitor for the treatment of cancer. [electronic resource] by
- Yao, Wenqing
- Zhuo, Jincong
- Burns, David M
- Xu, Meizhong
- Zhang, Colin
- Li, Yun-Long
- Qian, Ding-Quan
- He, Chunhong
- Weng, Lingkai
- Shi, Eric
- Lin, Qiyan
- Agrios, Costas
- Burn, Timothy C
- Caulder, Eian
- Covington, Maryanne B
- Fridman, Jordan S
- Friedman, Steven
- Katiyar, Kamna
- Hollis, Gregory
- Li, Yanlong
- Liu, Changnian
- Liu, Xiangdong
- Marando, Cindy A
- Newton, Robert
- Pan, Max
- Scherle, Peggy
- Taylor, Nancy
- Vaddi, Kris
- Wasserman, Zelda R
- Wynn, Richard
- Yeleswaram, Swamy
- Jalluri, Ravi
- Bower, Michael
- Zhou, Bing-Bing
- Metcalf, Brian
Producer: 20070327
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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