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2-Aryl-3-methyloctahydrophenanthrene-2,3,7-triols as potent dissociated glucocorticoid receptor agonists. [electronic resource] by
- Chantigny, Yves A
- Murray, John C
- Kleinman, Edward F
- Robinson, Ralph P
- Plotkin, Michael A
- Reese, Matthew R
- Buckbinder, Leonard
- McNiff, Patricia A
- Millham, Michele L
- Schaefer, Jean F
- Abramov, Yuriy A
- Bordner, Jon
Producer: 20150526
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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Optimization of Preclinical Metabolism for Somatostatin Receptor Subtype 5-Selective Antagonists. [electronic resource] by
- Liu, Weiguo
- Hussain, Zahid
- Zang, Yi
- Sweis, Ramzi F
- Romero, F Anthony
- Finke, Paul E
- Moningka, Remond
- Bao, Jianming
- Plotkin, Michael A
- Shang, Jin
- Dingley, Karen H
- Salituro, Gino
- Murphy, Beth Ann
- Howard, Andrew D
- Ujjainwalla, Feroze
- Wood, Harold B
- Duffy, Joseph L
Publication details: ACS medicinal chemistry letters Nov 2018
In:
ACS medicinal chemistry letters vol. 9
Availability: No items available.
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Corrigendum to "Discovery of benzofuran propanoic acid GPR120 agonists: From uHTS hit to mechanism-based pharmacodynamic effects" [Bioorg. Med. Chem. Lett. 26 (2016) 5724-5728]. [electronic resource] by
- Lombardo, Matthew
- Bender, Kate
- London, Clare
- Plotkin, Michael A
- Kirkland, Melissa
- Mane, Joel
- Pachanski, Michele
- Geissler, Wayne
- Cummings, John
- Habulihaz, Bahanu
- Akiyama, Taro E
- Di Salvo, Jerry
- Madeira, Maria
- Pols, Joanna
- Powles, Mary Ann
- Finley, Michael F
- Johnson, Eric
- Roussel, Thomas
- Uebele, Victor N
- Crespo, Alejandro
- Leung, Dennis
- Alleyne, Candice
- Trusca, Dorina
- Lei, Ying
- Howard, Andrew D
- Ujjainwalla, Feroze
- Tata, James R
- Sinz, Christopher J
Publication details: Bioorganic & medicinal chemistry letters 03 2017
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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5.
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Discovery of benzofuran propanoic acid GPR120 agonists: From uHTS hit to mechanism-based pharmacodynamic effects. [electronic resource] by
- Lombardo, Matthew
- Bender, Kate
- London, Clare
- Plotkin, Michael A
- Kirkland, Melissa
- Mane, Joel
- Pachanski, Michele
- Geissler, Wayne
- Cummings, John
- Habulihaz, Bahanu
- Akiyama, Taro E
- Di Salvo, Jerry
- Madeira, Maria
- Pols, Joanna
- Powles, Mary Ann
- Finley, Michael F
- Johnson, Eric
- Roussel, Thomas
- Uebele, Victor N
- Crespo, Alejandro
- Leung, Dennis
- Alleyne, Candice
- Trusca, Dorina
- Lei, Ying
- Howard, Andrew D
- Ujjainwalla, Feroze
- Tata, James R
- Sinz, Christopher J
Producer: 20170627
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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Selective small-molecule inhibition of an RNA structural element. [electronic resource] by
- Howe, John A
- Wang, Hao
- Fischmann, Thierry O
- Balibar, Carl J
- Xiao, Li
- Galgoci, Andrew M
- Malinverni, Juliana C
- Mayhood, Todd
- Villafania, Artjohn
- Nahvi, Ali
- Murgolo, Nicholas
- Barbieri, Christopher M
- Mann, Paul A
- Carr, Donna
- Xia, Ellen
- Zuck, Paul
- Riley, Dan
- Painter, Ronald E
- Walker, Scott S
- Sherborne, Brad
- de Jesus, Reynalda
- Pan, Weidong
- Plotkin, Michael A
- Wu, Jin
- Rindgen, Diane
- Cummings, John
- Garlisi, Charles G
- Zhang, Rumin
- Sheth, Payal R
- Gill, Charles J
- Tang, Haifeng
- Roemer, Terry
Producer: 20160426
In:
Nature vol. 526
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Design, Synthesis, and Evaluation of Novel and Selective G-protein Coupled Receptor 120 (GPR120) Spirocyclic Agonists. [electronic resource] by
- Cox, Jason M
- Chu, Hong D
- Chelliah, Mariappan V
- Debenham, John S
- Eagen, Keith
- Lan, Ping
- Lombardo, Matthew
- London, Clare
- Plotkin, Michael A
- Shah, Unmesh
- Sun, Zhongxiang
- Vaccaro, Henry M
- Venkatraman, Srikanth
- Suzuki, Takao
- Wang, Nengxue
- Ashley, Eric R
- Crespo, Alejandro
- Madeira, Maria
- Leung, Dennis H
- Alleyne, Candice
- Ogawa, Aimie M
- Souza, Sarah
- Thomas-Fowlkes, Brande
- Di Salvo, Jerry
- Weinglass, Adam
- Kirkland, Melissa
- Pachanski, Michele
- Powles, Mary Ann
- Tozzo, Effie
- Akiyama, Taro E
- Ujjainwalla, Feroze
- Tata, James R
- Sinz, Christopher J
Publication details: ACS medicinal chemistry letters Jan 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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