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Beyond Traditional Structure-Based Drug Design: The Role of Iron Complexation, Strain, and Water in the Binding of Inhibitors for Hypoxia-Inducible Factor Prolyl Hydroxylase 2. [electronic resource] by
- Bembenek, Scott D
- Venkatesan, Hariharan
- Peltier, Hillary M
- Rosen, Mark D
- Barrett, Terrance D
- Kanelakis, Kimon C
- Palomino, Heather L
- Brondstetter, Theresa I
- Mirzadegan, Taraneh
- Rabinowitz, Michael H
Publication details: ACS omega Apr 2019
In:
ACS omega vol. 4
Availability: No items available.
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Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective hypoxia-inducible factor prolyl hydroxylase inhibitor. [electronic resource] by
- Barrett, Terrance D
- Palomino, Heather L
- Brondstetter, Theresa I
- Kanelakis, Kimon C
- Wu, Xiaodong
- Haug, Peter V
- Yan, Wen
- Young, Andrew
- Hua, Hong
- Hart, Juliet C
- Tran, Da-Thao
- Venkatesan, Hariharan
- Rosen, Mark D
- Peltier, Hillary M
- Sepassi, Kia
- Rizzolio, Michele C
- Bembenek, Scott D
- Mirzadegan, Tara
- Rabinowitz, Michael H
- Shankley, Nigel P
Producer: 20110801
In:
Molecular pharmacology vol. 79
Availability: No items available.
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10.
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Benzimidazole-2-pyrazole HIF Prolyl 4-Hydroxylase Inhibitors as Oral Erythropoietin Secretagogues. [electronic resource] by
- Rosen, Mark D
- Venkatesan, Hariharan
- Peltier, Hillary M
- Bembenek, Scott D
- Kanelakis, Kimon C
- Zhao, Lucy X
- Leonard, Barry E
- Hocutt, Frances M
- Wu, Xiaodong
- Palomino, Heather L
- Brondstetter, Theresa I
- Haugh, Peter V
- Cagnon, Laurence
- Yan, Wen
- Liotta, Lisa A
- Young, Andrew
- Mirzadegan, Tara
- Shankley, Nigel P
- Barrett, Terrance D
- Rabinowitz, Michael H
Producer: 20140605
In:
ACS medicinal chemistry letters vol. 1
Availability: No items available.
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