Results
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2.
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Inhibitors of epidermal growth factor receptor tyrosine kinase: optimisation of potency and in vivo pharmacokinetics. [electronic resource] by
- Ballard, Peter
- Bradbury, Robert H
- Harris, Craig S
- Hennequin, Laurent F A
- Hickinson, Mark
- Kettle, Jason G
- Kendrew, Jane
- Klinowska, Teresa
- Ogilvie, Donald J
- Pearson, Stuart E
- Williams, Emma J
- Wilson, Ingrid
Producer: 20061016
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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3.
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Neutral 5-substituted 4-anilinoquinazolines as potent, orally active inhibitors of erbB2 receptor tyrosine kinase. [electronic resource] by
- Ballard, Peter
- Barlaam, Bernard C
- Bradbury, Robert H
- Dishington, Allan
- Hennequin, Laurent F A
- Hickinson, D Mark
- Hollingsworth, Ian M
- Kettle, Jason G
- Klinowska, Teresa
- Ogilvie, Donald J
- Pearson, Stuart E
- Scott, James S
- Suleman, Abid
- Whittaker, Robin
- Williams, Emma J
- Wood, Robin
- Wright, Lindsay
Producer: 20080623
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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4.
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Discovery of AZD3147: a potent, selective dual inhibitor of mTORC1 and mTORC2. [electronic resource] by
- Pike, Kurt G
- Morris, Jeff
- Ruston, Linette
- Pass, Sarah L
- Greenwood, Ryan
- Williams, Emma J
- Demeritt, Julie
- Culshaw, Janet D
- Gill, Kristy
- Pass, Martin
- Finlay, M Raymond V
- Good, Catherine J
- Roberts, Craig A
- Currie, Gordon S
- Blades, Kevin
- Eden, Jonathan M
- Pearson, Stuart E
Producer: 20150615
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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5.
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A new series of neutral 5-substituted 4-anilinoquinazolines as potent, orally active inhibitors of erbB2 receptor tyrosine kinase. [electronic resource] by
- Barlaam, Bernard
- Ballard, Peter
- Bradbury, Robert H
- Ducray, Richard
- Germain, Hervé
- Hickinson, D Mark
- Hudson, Kevin
- Kettle, Jason G
- Klinowska, Teresa
- Magnien, Françoise
- Ogilvie, Donald J
- Olivier, Annie
- Pearson, Stuart E
- Scott, James S
- Suleman, Abid
- Trigwell, Cath B
- Vautier, Michel
- Whittaker, Robin D
- Wood, Robin
Producer: 20080527
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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6.
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AZD9496: An Oral Estrogen Receptor Inhibitor That Blocks the Growth of ER-Positive and ESR1-Mutant Breast Tumors in Preclinical Models. [electronic resource] by
- Weir, Hazel M
- Bradbury, Robert H
- Lawson, Mandy
- Rabow, Alfred A
- Buttar, David
- Callis, Rowena J
- Curwen, Jon O
- de Almeida, Camila
- Ballard, Peter
- Hulse, Michael
- Donald, Craig S
- Feron, Lyman J L
- Karoutchi, Galith
- MacFaul, Philip
- Moss, Thomas
- Norman, Richard A
- Pearson, Stuart E
- Tonge, Michael
- Davies, Gareth
- Walker, Graeme E
- Wilson, Zena
- Rowlinson, Rachel
- Powell, Steve
- Sadler, Claire
- Richmond, Graham
- Ladd, Brendon
- Pazolli, Ermira
- Mazzola, Anne Marie
- D'Cruz, Celina
- De Savi, Chris
Producer: 20170728
In:
Cancer research vol. 76
Availability: No items available.
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7.
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Optimization of a Novel Binding Motif to (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)phenyl)acrylic Acid (AZD9496), a Potent and Orally Bioavailable Selective Estrogen Receptor Downregulator and Antagonist. [electronic resource] by
- De Savi, Chris
- Bradbury, Robert H
- Rabow, Alfred A
- Norman, Richard A
- de Almeida, Camila
- Andrews, David M
- Ballard, Peter
- Buttar, David
- Callis, Rowena J
- Currie, Gordon S
- Curwen, Jon O
- Davies, Chris D
- Donald, Craig S
- Feron, Lyman J L
- Gingell, Helen
- Glossop, Steven C
- Hayter, Barry R
- Hussain, Syeed
- Karoutchi, Galith
- Lamont, Scott G
- MacFaul, Philip
- Moss, Thomas A
- Pearson, Stuart E
- Tonge, Michael
- Walker, Graeme E
- Weir, Hazel M
- Wilson, Zena
Producer: 20160202
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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