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4,5-dihydroxypyrimidine carboxamides and N-alkyl-5-hydroxypyrimidinone carboxamides are potent, selective HIV integrase inhibitors with good pharmacokinetic profiles in preclinical species. [electronic resource] by
- Summa, Vincenzo
- Petrocchi, Alessia
- Matassa, Victor G
- Gardelli, Cristina
- Muraglia, Ester
- Rowley, Michael
- Paz, Odalys Gonzalez
- Laufer, Ralph
- Monteagudo, Edith
- Pace, Paola
Producer: 20070119
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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A novel series of potent and selective ketone histone deacetylase inhibitors with antitumor activity in vivo. [electronic resource] by
- Jones, Philip
- Altamura, Sergio
- De Francesco, Raffaele
- Paz, Odalys Gonzalez
- Kinzel, Olaf
- Mesiti, Giuseppe
- Monteagudo, Edith
- Pescatore, Giovanna
- Rowley, Michael
- Verdirame, Maria
- Steinkühler, Christian
Producer: 20080602
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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Discovery and synthesis of HIV integrase inhibitors: development of potent and orally bioavailable N-methyl pyrimidones. [electronic resource] by
- Gardelli, Cristina
- Nizi, Emanuela
- Muraglia, Ester
- Crescenzi, Benedetta
- Ferrara, Marco
- Orvieto, Federica
- Pace, Paola
- Pescatore, Giovanna
- Poma, Marco
- Ferreira, Maria Del Rosario Rico
- Scarpelli, Rita
- Homnick, Carl F
- Ikemoto, Norihiro
- Alfieri, Anna
- Verdirame, Maria
- Bonelli, Fabio
- Paz, Odalys Gonzalez
- Taliani, Marina
- Monteagudo, Edith
- Pesci, Silvia
- Laufer, Ralph
- Felock, Peter
- Stillmock, Kara A
- Hazuda, Daria
- Rowley, Michael
- Summa, Vincenzo
Producer: 20071121
In:
Journal of medicinal chemistry vol. 50
Availability: No items available.
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