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	1.	Collagen and aggrecan degradation is blocked in interleukin-1-treated cartilage explants by an inhibitor of IkappaB kinase through suppression of metalloproteinase expression. [electronic resource] by Pattoli, Mark A MacMaster, John F Gregor, Kurt R Burke, James R Producer: 20051128 In: The Journal of pharmacology and experimental therapeutics vol. 315 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	2.	Conversion of carbazole carboxamide based reversible inhibitors of Bruton's tyrosine kinase (BTK) into potent, selective irreversible inhibitors in the carbazole, tetrahydrocarbazole, and a new 2,3-dimethylindole series. [electronic resource] by Liu, Qingjie Batt, Douglas G Chaudhry, Charu Lippy, Jonathan S Pattoli, Mark A Surti, Neha Xu, Songmei Carter, Percy H Burke, James R Tino, Joseph A Producer: 20190321 In: Bioorganic & medicinal chemistry letters vol. 28 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	3.	A highly selective inhibitor of I kappa B kinase, BMS-345541, blocks both joint inflammation and destruction in collagen-induced arthritis in mice. [electronic resource] by McIntyre, Kim W Shuster, David J Gillooly, Kathleen M Dambach, Donna M Pattoli, Mark A Lu, Pin Zhou, Xia-Di Qiu, Yuping Zusi, F Christopher Burke, James R Producer: 20031017 In: Arthritis and rheumatism vol. 48 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	4.	BMS-345541 is a highly selective inhibitor of I kappa B kinase that binds at an allosteric site of the enzyme and blocks NF-kappa B-dependent transcription in mice. [electronic resource] by Burke, James R Pattoli, Mark A Gregor, Kurt R Brassil, Patrick J MacMaster, John F McIntyre, Kim W Yang, Xiaoxia Iotzova, Violetta S Clarke, Wendy Strnad, Joann Qiu, Yuping Zusi, F Christopher Producer: 20030214 In: The Journal of biological chemistry vol. 278 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	5.	Determination of Real Time in Vivo Drug Receptor Occupancy for a Covalent Binding Drug as a Clinical Pharmacodynamic Biomarker by Immunocapture-LC-MS/MS. [electronic resource] by Zheng, Naiyu Catlett, Ian M Taylor, Kristin Gu, Huidong Pattoli, Mark A Neely, Robert J Li, Wenying Allentoff, Alban Yuan, Xiling Ciccimaro, Eugene Yao, Ming Warrack, Bethanne M Burke, James R Zhang, Yan J Pillutla, Renuka Zeng, Jianing Producer: 20200918 In: Analytical chemistry vol. 91 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	6.	Synthesis and biological evaluation of 4-amino derivatives of benzimidazoquinoxaline, benzimidazoquinoline, and benzopyrazoloquinazoline as potent IKK inhibitors. [electronic resource] by Beaulieu, Francis Ouellet, Carl Ruediger, Edward H Belema, Makonen Qiu, Yuping Yang, Xuejie Banville, Jacques Burke, James R Gregor, Kurt R MacMaster, John F Martel, Alain McIntyre, Kim W Pattoli, Mark A Zusi, F Christopher Vyas, Dolatrai Producer: 20070515 In: Bioorganic & medicinal chemistry letters vol. 17 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	7.	Bruton's tyrosine kinase inhibitor BMS-986142 in experimental models of rheumatoid arthritis enhances efficacy of agents representing clinical standard-of-care. [electronic resource] by Gillooly, Kathleen M Pulicicchio, Claudine Pattoli, Mark A Cheng, Lihong Skala, Stacey Heimrich, Elizabeth M McIntyre, Kim W Taylor, Tracy L Kukral, Daniel W Dudhgaonkar, Shailesh Nagar, Jignesh Banas, Dana Watterson, Scott H Tino, Joseph A Fura, Aberra Burke, James R Producer: 20170929 In: PloS one vol. 12 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	8.	Synthesis and structure-activity relationship of imidazo(1,2-a)thieno(3,2-e)pyrazines as IKK-beta inhibitors. [electronic resource] by Belema, Makonen Bunker, Amy Nguyen, Van N Beaulieu, Francis Ouellet, Carl Qiu, Yuping Zhang, Yunhui Martel, Alain Burke, James R McIntyre, Kim W Pattoli, Mark A Daloisio, Connie Gillooly, Kathleen M Clarke, Wendy J Brassil, Patrick J Zusi, F Chris Vyas, Dolatrai M Producer: 20071001 In: Bioorganic & medicinal chemistry letters vol. 17 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	9.	Imidazo[4,5-d]thiazolo[5,4-b]pyridine based inhibitors of IKK2: synthesis, SAR, PK/PD and activity in a preclinical model of rheumatoid arthritis. [electronic resource] by Dyckman, Alaric J Langevine, Charles M Quesnelle, Claude Kempson, James Guo, Junqing Gill, Patrice Spergel, Steven H Watterson, Scott H Li, Tianle Nirschl, David S Gillooly, Kathleen M Pattoli, Mark A McIntyre, Kim W Chen, Laishun McKinnon, Murray Dodd, John H Barrish, Joel C Burke, James R Pitts, William J Producer: 20110414 In: Bioorganic & medicinal chemistry letters vol. 21 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	10.	Periodic, partial inhibition of IkappaB Kinase beta-mediated signaling yields therapeutic benefit in preclinical models of rheumatoid arthritis. [electronic resource] by Gillooly, Kathleen M Pattoli, Mark A Taylor, Tracy L Chen, Laishun Cheng, Lihong Gregor, Kurt R Whitney, Gena S Susulic, Vojkan Watterson, Scott H Kempson, James Pitts, William J Booth-Lute, Hollie Yang, Guchen Davies, Paul Kukral, Daniel W Strnad, Joann McIntyre, Kim W Darienzo, Celia J Salter-Cid, Luisa Yang, Zheng Wang-Iverson, David B Burke, James R Producer: 20091130 In: The Journal of pharmacology and experimental therapeutics vol. 331 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	11.	Novel tricyclic inhibitors of IKK2: discovery and SAR leading to the identification of 2-methoxy-N-((6-(1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl)pyridin-2-yl)methyl)acetamide (BMS-066). [electronic resource] by Watterson, Scott H Langevine, Charles M Van Kirk, Katy Kempson, James Guo, Junquing Spergel, Steven H Das, Jagabandhu Moquin, Robert V Dyckman, Alaric J Nirschl, David Gregor, Kurt Pattoli, Mark A Yang, XiaoXia McIntyre, Kim W Yang, Guchen Galella, Michael A Booth-Lute, Hollie Chen, Laishun Yang, Zheng Wang-Iverson, David McKinnon, Murray Dodd, John H Barrish, Joel C Burke, James R Pitts, William J Producer: 20120418 In: Bioorganic & medicinal chemistry letters vol. 21 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	12.	Novel tricyclic inhibitors of IkappaB kinase. [electronic resource] by Kempson, James Spergel, Steven H Guo, Junqing Quesnelle, Claude Gill, Patrice Belanger, Dominique Dyckman, Alaric J Li, Tianle Watterson, Scott H Langevine, Charles M Das, Jagabandhu Moquin, Robert V Furch, Joseph A Marinier, Anne Dodier, Marco Martel, Alain Nirschl, David Van Kirk, Katy Burke, James R Pattoli, Mark A Gillooly, Kathleen McIntyre, Kim W Chen, Laishun Yang, Zheng Marathe, Punit H Wang-Iverson, David Dodd, John H McKinnon, Murray Barrish, Joel C Pitts, William J Producer: 20090428 In: Journal of medicinal chemistry vol. 52 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	13.	Small Molecule Reversible Inhibitors of Bruton's Tyrosine Kinase (BTK): Structure-Activity Relationships Leading to the Identification of 7-(2-Hydroxypropan-2-yl)-4-[2-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)phenyl]-9H-carbazole-1-carboxamide (BMS-935177). [electronic resource] by De Lucca, George V Shi, Qing Liu, Qingjie Batt, Douglas G Beaudoin Bertrand, Myra Rampulla, Rick Mathur, Arvind Discenza, Lorell D'Arienzo, Celia Dai, Jun Obermeier, Mary Vickery, Rodney Zhang, Yingru Yang, Zheng Marathe, Punit Tebben, Andrew J Muckelbauer, Jodi K Chang, ChiehYing J Zhang, Huiping Gillooly, Kathleen Taylor, Tracy Pattoli, Mark A Skala, Stacey Kukral, Daniel W McIntyre, Kim W Salter-Cid, Luisa Fura, Aberra Burke, James R Barrish, Joel C Carter, Percy H Tino, Joseph A Producer: 20170710 In: Journal of medicinal chemistry vol. 59 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	14.	Discovery of 6-Fluoro-5-(R)-(3-(S)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4H)-yl)-2-methylphenyl)-2-(S)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1H-carbazole-8-carboxamide (BMS-986142): A Reversible Inhibitor of Bruton's Tyrosine Kinase (BTK) Conformationally Constrained by Two Locked Atropisomers. [electronic resource] by Watterson, Scott H De Lucca, George V Shi, Qing Langevine, Charles M Liu, Qingjie Batt, Douglas G Beaudoin Bertrand, Myra Gong, Hua Dai, Jun Yip, Shiuhang Li, Peng Sun, Dawn Wu, Dauh-Rurng Wang, Chunlei Zhang, Yingru Traeger, Sarah C Pattoli, Mark A Skala, Stacey Cheng, Lihong Obermeier, Mary T Vickery, Rodney Discenza, Lorell N D'Arienzo, Celia J Zhang, Yifan Heimrich, Elizabeth Gillooly, Kathleen M Taylor, Tracy L Pulicicchio, Claudine McIntyre, Kim W Galella, Michael A Tebben, Andy J Muckelbauer, Jodi K Chang, ChiehYing Rampulla, Richard Mathur, Arvind Salter-Cid, Luisa Barrish, Joel C Carter, Percy H Fura, Aberra Burke, James R Tino, Joseph A Producer: 20170619 In: Journal of medicinal chemistry vol. 59 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)
	15.	Discovery of Branebrutinib (BMS-986195): A Strategy for Identifying a Highly Potent and Selective Covalent Inhibitor Providing Rapid in Vivo Inactivation of Bruton's Tyrosine Kinase (BTK). [electronic resource] by Watterson, Scott H Liu, Qingjie Beaudoin Bertrand, Myra Batt, Douglas G Li, Ling Pattoli, Mark A Skala, Stacey Cheng, Lihong Obermeier, Mary T Moore, Robin Yang, Zheng Vickery, Rodney Elzinga, Paul A Discenza, Lorell D'Arienzo, Celia Gillooly, Kathleen M Taylor, Tracy L Pulicicchio, Claudine Zhang, Yifan Heimrich, Elizabeth McIntyre, Kim W Ruan, Qian Westhouse, Richard A Catlett, Ian M Zheng, Naiyu Chaudhry, Charu Dai, Jun Galella, Michael A Tebben, Andrew J Pokross, Matt Li, Jianqing Zhao, Rulin Smith, Daniel Rampulla, Richard Allentoff, Alban Wallace, Michael A Mathur, Arvind Salter-Cid, Luisa Macor, John E Carter, Percy H Fura, Aberra Burke, James R Tino, Joseph A Producer: 20200914 In: Journal of medicinal chemistry vol. 62 Online resources: Available from publisher's website Availability: No items available. Save to lists Add to cart (remove)