Results
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Diastereoselective synthesis and configuration-dependent activity of (3-substituted-cycloalkyl)glycine pyrrolidides and thiazolidides as dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Ashton, Wallace T
- Dong, Hong
- Sisco, Rosemary M
- Doss, George A
- Leiting, Barbara
- Patel, Reshma A
- Wu, Joseph K
- Marsilio, Frank
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20040928
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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3.
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Imidazopiperidine amides as dipeptidyl peptidase IV inhibitors for the treatment of diabetes. [electronic resource] by
- Chen, Ping
- Caldwell, Charles G
- Mathvink, Robert J
- Leiting, Barbara
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- He, Huaibing
- Lyons, Kathryn A
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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4.
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Dipeptidyl peptidase IV inhibitors derived from beta-aminoacylpiperidines bearing a fused thiazole, oxazole, isoxazole, or pyrazole. [electronic resource] by
- Ashton, Wallace T
- Sisco, Rosemary M
- Dong, Hong
- Lyons, Kathryn A
- He, Huaibing
- Doss, George A
- Leiting, Barbara
- Patel, Reshma A
- Wu, Joseph K
- Marsilio, Frank
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20050930
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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5.
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Discovery of potent and selective phenylalanine based dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Xu, Jinyou
- Wei, Lan
- Mathvink, Robert
- He, Jiafang
- Park, You-Jung
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20051011
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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6.
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Design, synthesis, and biological evaluation of triazolopiperazine-based beta-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitors. [electronic resource] by
- Kowalchick, Jennifer E
- Leiting, Barbara
- Pryor, KellyAnn D
- Marsilio, Frank
- Wu, Joseph K
- He, Huaibing
- Lyons, Kathryn A
- Eiermann, George J
- Petrov, Aleksandr
- Scapin, Giovanna
- Patel, Reshma A
- Thornberry, Nancy A
- Weber, Ann E
- Kim, Dooseop
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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7.
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Substituted piperazines as novel dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Brockunier, Linda L
- He, Jiafang
- Colwell, Lawrence F
- Habulihaz, Bahanu
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Marsilio, Frank
- Patel, Reshma A
- Teffera, Yohannes
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
- Parmee, Emma R
Producer: 20050307
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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8.
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Fluoropyrrolidine amides as dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Caldwell, Charles G
- Chen, Ping
- He, Jiafang
- Parmee, Emma R
- Leiting, Barbara
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- Eiermann, George J
- Petrov, Aleksandr
- He, Huaibing
- Lyons, Kathryn A
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20041012
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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9.
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Discovery of 3-aminopiperidines as potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Cox, Jason M
- Harper, Bart
- Mastracchio, Anthony
- Leiting, Barbara
- Sinha Roy, Ranabir
- Patel, Reshma A
- Wu, Joseph K
- Lyons, Kathryn A
- He, Huaibing
- Xu, Shiyao
- Zhu, Bing
- Thornberry, Nancy A
- Weber, Ann E
- Edmondson, Scott D
Producer: 20071121
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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10.
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Triazolopiperazine-amides as dipeptidyl peptidase IV inhibitors: close analogs of JANUVIA (sitagliptin phosphate). [electronic resource] by
- Kim, Dooseop
- Kowalchick, Jennifer E
- Edmondson, Scott D
- Mastracchio, Anthony
- Xu, Jinyou
- Eiermann, George J
- Leiting, Barbara
- Wu, Joseph K
- Pryor, KellyAnn D
- Patel, Reshma A
- He, Huaibing
- Lyons, Kathryn A
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20070830
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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11.
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Discovery of potent and selective beta-homophenylalanine based dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Xu, Jinyou
- Ok, Hyun O
- Gonzalez, Edward J
- Colwell, Lawrence F
- Habulihaz, Bahanu
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
- Parmee, Emma R
Producer: 20050307
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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12.
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4-aminophenylalanine and 4-aminocyclohexylalanine derivatives as potent, selective, and orally bioavailable inhibitors of dipeptidyl peptidase IV. [electronic resource] by
- Duffy, Joseph L
- Kirk, Brian A
- Wang, Liping
- Eiermann, George J
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Patel, Reshma A
- Patel, Sangita B
- Petrov, Alexsandr
- Scapin, Giovanna
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20070730
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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13.
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4-arylcyclohexylalanine analogs as potent, selective, and orally active inhibitors of dipeptidyl peptidase IV. [electronic resource] by
- Kaelin, David E
- Smenton, Abigail L
- Eiermann, George J
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Patel, Reshma A
- Patel, Sangita B
- Petrov, Alexsandr
- Scapin, Giovanna
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
- Duffy, Joseph L
Producer: 20080205
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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14.
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Discovery of potent, selective, and orally bioavailable pyridone-based dipeptidyl peptidase-4 inhibitors. [electronic resource] by
- Xu, Jinyou
- Wei, Lan
- Mathvink, Robert
- Edmondson, Scott D
- Mastracchio, Anthony
- Eiermann, George J
- He, Huaibing
- Leone, Joseph F
- Leiting, Barbara
- Lyons, Kathryn A
- Marsilio, Frank
- Patel, Reshma A
- Petrov, Aleksandr
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20060323
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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15.
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Discovery of potent and selective orally bioavailable beta-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Edmondson, Scott D
- Mastracchio, Anthony
- Duffy, Joseph L
- Eiermann, George J
- He, Huaibing
- Ita, Ida
- Leiting, Barbara
- Leone, Joseph F
- Lyons, Kathryn A
- Makarewicz, Amanda M
- Patel, Reshma A
- Petrov, Aleksandr
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20050919
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
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16.
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Aminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors. [electronic resource] by
- Edmondson, Scott D
- Mastracchio, Anthony
- Cox, Jason M
- Eiermann, George J
- He, Huaibing
- Lyons, Kathryn A
- Patel, Reshma A
- Patel, Sangita B
- Petrov, Aleksandr
- Scapin, Giovanna
- Wu, Joseph K
- Xu, Shiyao
- Zhu, Bing
- Thornberry, Nancy A
- Roy, Ranabir Sinha
- Weber, Ann E
Producer: 20091207
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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17.
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Potent and selective proline derived dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Edmondson, Scott D
- Mastracchio, Anthony
- Beconi, Maria
- Colwell, Lawrence F
- Habulihaz, Bahanu
- He, Huaibing
- Kumar, Sanjeev
- Leiting, Barbara
- Lyons, Kathryn A
- Mao, Ann
- Marsilio, Frank
- Patel, Reshma A
- Wu, Joseph K
- Zhu, Lan
- Thornberry, Nancy A
- Weber, Ann E
- Parmee, Emma R
Producer: 20050404
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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18.
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Discovery of potent, selective, and orally bioavailable oxadiazole-based dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Xu, Jinyou
- Wei, Lan
- Mathvink, Robert J
- Edmondson, Scott D
- Eiermann, George J
- He, Huaibing
- Leone, Joseph F
- Leiting, Barbara
- Lyons, Kathryn A
- Marsilio, Frank
- Patel, Reshma A
- Patel, Sangita B
- Petrov, Aleksandr
- Scapin, Giovanna
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20061204
In:
Bioorganic & medicinal chemistry letters vol. 16
Availability: No items available.
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19.
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Fluoroolefins as amide bond mimics in dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Edmondson, Scott D
- Wei, Lan
- Xu, Jinyou
- Shang, Jackie
- Xu, Shiyao
- Pang, Jianmei
- Chaudhary, Ashok
- Dean, Dennis C
- He, Huaibing
- Leiting, Barbara
- Lyons, Kathryn A
- Patel, Reshma A
- Patel, Sangita B
- Scapin, Giovanna
- Wu, Joseph K
- Beconi, Maria G
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20080708
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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20.
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4-Amino cyclohexylglycine analogues as potent dipeptidyl peptidase IV inhibitors. [electronic resource] by
- Parmee, Emma R
- He, Jiafang
- Mastracchio, Anthony
- Edmondson, Scott D
- Colwell, Larry
- Eiermann, George
- Feeney, William P
- Habulihaz, Bahanu
- He, Huaibing
- Kilburn, Ruth
- Leiting, Barbara
- Lyons, Kathryn
- Marsilio, Frank
- Patel, Reshma A
- Petrov, Aleksandr
- Di Salvo, Jerry
- Wu, Joseph K
- Thornberry, Nancy A
- Weber, Ann E
Producer: 20040827
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
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