Results
|
1.
|
|
|
2.
|
|
|
3.
|
Estrogen receptor ligands. Part 5: The SAR of dihydrobenzoxathiins containing modified basic side chains. [electronic resource] by
- Tan, Qiang
- Birzin, Elizabeth T
- Chan, Wanda
- Tien Yang, Yi
- Pai, Lee-Yuh
- Hayes, Edward C
- DaSilva, Carolyn A
- DiNinno, Frank
- Rohrer, Susan P
- Schaeffer, James M
- Hammond, Milton L
Producer: 20050207
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
|
|
4.
|
Estrogen receptor ligands. Part 6: Synthesis and binding affinity of dihydrobenzodithiins. [electronic resource] by
- Tan, Qiang
- Birzin, Elizabeth T
- Chan, Wanda
- Yang, Yi Tien
- Pai, Lee-Yuh
- Hayes, Edward C
- DaSilva, Carolyn A
- DiNinno, Frank
- Rohrer, Susan P
- Schaeffer, James M
- Hammond, Milton L
Producer: 20050207
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
|
|
5.
|
Estrogen receptor ligands. Part 11: Synthesis and activity of isochromans and isothiochromans. [electronic resource] by
- Liu, Jian
- Birzin, Elizabeth T
- Chan, Wanda
- Yang, Yi Tien
- Pai, Lee-Yuh
- Dasilva, Carolyn
- Hayes, Edward C
- Mosley, Ralph T
- Dininno, Frank
- Rohrer, Susan P
- Schaeffer, James M
- Hammond, Milton L
Producer: 20050607
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
|
|
6.
|
Estrogen receptor ligands. Part 14: application of novel antagonist side chains to existing platforms. [electronic resource] by
- Blizzard, Timothy A
- Morgan, Jerry D
- Chan, Wanda
- Birzin, Elizabeth T
- Pai, Lee-Yuh
- Hayes, Edward C
- DaSilva, Carolyn A
- Mosley, Ralph T
- Yang, Yi Tien
- Rohrer, Susan P
- Dininno, Frank
- Hammond, Milton L
Producer: 20060123
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
|
|
7.
|
A strategy of employing aminoheterocycles as amide mimics to identify novel, potent and bioavailable soluble epoxide hydrolase inhibitors. [electronic resource] by
- Shen, Hong C
- Ding, Fa-Xiang
- Deng, Qiaolin
- Xu, Suoyu
- Tong, Xinchun
- Zhang, Xiaoping
- Chen, Yuli
- Zhou, Gaochao
- Pai, Lee-Yuh
- Alonso-Galicia, Magdalena
- Roy, Sophie
- Zhang, Bei
- Tata, James R
- Berger, Joel P
- Colletti, Steven L
Producer: 20091130
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
|
|
8.
|
Estrogen receptor ligands. Part 13: Dihydrobenzoxathiin SERAMs with an optimized antagonist side chain. [electronic resource] by
- Blizzard, Timothy A
- DiNinno, Frank
- Chen, Helen Y
- Kim, Seongkon
- Wu, Jane Y
- Chan, Wanda
- Birzin, Elizabeth T
- Yang, Yi Tien
- Pai, Lee-Yuh
- Hayes, Edward C
- DaSilva, Carolyn A
- Rohrer, Susan P
- Schaeffer, James M
- Hammond, Milton L
Producer: 20051018
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
|
|
9.
|
Evaluation of selective inhibitors of 11β-HSD1 for the treatment of hypertension. [electronic resource] by
- Bauman, David R
- Whitehead, Alan
- Contino, Lisa C
- Cui, Jisong
- Garcia-Calvo, Margarita
- Gu, Xin
- Kevin, Nancy
- Ma, Xiuying
- Pai, Lee-yuh
- Shah, Kashmira
- Shen, Xiaolan
- Stribling, Sloan
- Zokian, Hratch J
- Metzger, Joe
- Shevell, Diane E
- Waddell, Sherman T
Producer: 20140424
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
|
|
10.
|
Estrogen receptor ligands. Part 16: 2-Aryl indoles as highly subtype selective ligands for ERalpha. [electronic resource] by
- Dykstra, Kevin D
- Guo, Liangqin
- Birzin, Elizabeth T
- Chan, Wanda
- Yang, Yi Tien
- Hayes, Edward C
- DaSilva, Carolyn A
- Pai, Lee-Yuh
- Mosley, Ralph T
- Kraker, Bryan
- Fitzgerald, Paula M D
- DiNinno, Frank
- Rohrer, Susan P
- Schaeffer, James M
- Hammond, Milton L
Producer: 20070530
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
|
|
11.
|
Discovery of 3,3-disubstituted piperidine-derived trisubstituted ureas as highly potent soluble epoxide hydrolase inhibitors. [electronic resource] by
- Shen, Hong C
- Ding, Fa-Xiang
- Deng, Qiaolin
- Xu, Suoyu
- Chen, Hsuan-Shen
- Tong, Xinchun
- Tong, Vincent
- Zhang, Xiaoping
- Chen, Yuli
- Zhou, Gaochao
- Pai, Lee-Yuh
- Alonso-Galicia, Magdalena
- Zhang, Bei
- Roy, Sophie
- Tata, James R
- Berger, Joel P
- Colletti, Steven L
Producer: 20091123
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
|
|
12.
|
Estrogen receptor ligands. II. Discovery of benzoxathiins as potent, selective estrogen receptor alpha modulators. [electronic resource] by
- Kim, Seongkon
- Wu, Jane Y
- Birzin, Elizabeth T
- Frisch, Katalin
- Chan, Wanda
- Pai, Lee-Yuh
- Yang, Yi Tien
- Mosley, Ralph T
- Fitzgerald, Paula M D
- Sharma, Nandini
- Dahllund, Johanna
- Thorsell, Ann-Gerd
- DiNinno, Frank
- Rohrer, Susan P
- Schaeffer, James M
- Hammond, Milton L
Producer: 20040520
In:
Journal of medicinal chemistry vol. 47
Availability: No items available.
|
|
13.
|
Discovery of spirocyclic secondary amine-derived tertiary ureas as highly potent, selective and bioavailable soluble epoxide hydrolase inhibitors. [electronic resource] by
- Shen, Hong C
- Ding, Fa-Xiang
- Wang, Siyi
- Xu, Suoyu
- Chen, Hsuan-shen
- Tong, Xinchun
- Tong, Vincent
- Mitra, Kaushik
- Kumar, Sanjeev
- Zhang, Xiaoping
- Chen, Yuli
- Zhou, Gaochao
- Pai, Lee-Yuh
- Alonso-Galicia, Magdalena
- Chen, Xiaoli
- Zhang, Bei
- Tata, James R
- Berger, Joel P
- Colletti, Steven L
Producer: 20090901
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
|
|
14.
|
Estrogen receptor ligands. Part 8: Dihydrobenzoxathiin SERAMs with heteroatom-substituted side chains. [electronic resource] by
- Blizzard, Timothy A
- DiNinno, Frank
- Morgan, Jerry D
- Wu, Jane Y
- Chen, Helen Y
- Kim, Seongkon
- Chan, Wanda
- Birzin, Elizabeth T
- Yang, Yi Tien
- Pai, Lee-Yuh
- Zhang, Zhoupeng
- Hayes, Edward C
- DaSilva, Carolyn A
- Tang, Wei
- Rohrer, Susan P
- Schaeffer, James M
- Hammond, Milton L
Producer: 20050412
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
|
|
15.
|
Estrogen receptor ligands. Part 7: Dihydrobenzoxathiin SERAMs with bicyclic amine side chains. [electronic resource] by
- Blizzard, Timothy A
- DiNinno, Frank
- Morgan, Jerry D
- Chen, Helen Y
- Wu, Jane Y
- Gude, Candido
- Kim, Seongkon
- Chan, Wanda
- Birzin, Elizabeth T
- Tien Yang, Yi
- Pai, Lee-Yuh
- Zhang, Zhoupeng
- Hayes, Edward C
- DaSilva, Carolyn A
- Tang, Wei
- Rohrer, Susan P
- Schaeffer, James M
- Hammond, Milton L
Producer: 20050412
In:
Bioorganic & medicinal chemistry letters vol. 14
Availability: No items available.
|
|
16.
|
Pharmacologic inhibition of the renal outer medullary potassium channel causes diuresis and natriuresis in the absence of kaliuresis. [electronic resource] by
- Garcia, Maria L
- Priest, Birgit T
- Alonso-Galicia, Magdalena
- Zhou, Xiaoyan
- Felix, John P
- Brochu, Richard M
- Bailey, Timothy
- Thomas-Fowlkes, Brande
- Liu, Jessica
- Swensen, Andrew
- Pai, Lee-Yuh
- Xiao, Jianying
- Hernandez, Melba
- Hoagland, Kimberly
- Owens, Karen
- Tang, Haifeng
- de Jesus, Reynalda K
- Roy, Sophie
- Kaczorowski, Gregory J
- Pasternak, Alexander
Producer: 20140210
In:
The Journal of pharmacology and experimental therapeutics vol. 348
Availability: No items available.
|
|
17.
|
Estrogen receptor ligands. Part 9: Dihydrobenzoxathiin SERAMs with alkyl substituted pyrrolidine side chains and linkers. [electronic resource] by
- Blizzard, Timothy A
- Dininno, Frank
- Morgan, Jerry D
- Chen, Helen Y
- Wu, Jane Y
- Kim, Seongkon
- Chan, Wanda
- Birzin, Elizabeth T
- Yang, Yi Tien
- Pai, Lee-Yuh
- Fitzgerald, Paula M D
- Sharma, Nandini
- Li, Ying
- Zhang, Zhoupeng
- Hayes, Edward C
- Dasilva, Carolyn A
- Tang, Wei
- Rohrer, Susan P
- Schaeffer, James M
- Hammond, Milton L
Producer: 20050502
In:
Bioorganic & medicinal chemistry letters vol. 15
Availability: No items available.
|
|
18.
|
The Renal Outer Medullary Potassium Channel Inhibitor, MK-7145, Lowers Blood Pressure, and Manifests Features of Bartter's Syndrome Type II Phenotype. [electronic resource] by
- Hampton, Caryn
- Zhou, Xiaoyan
- Priest, Birgit T
- Pai, Lee-Yuh
- Felix, John P
- Thomas-Fowlkes, Brande
- Liu, Jessica
- Kohler, Martin
- Xiao, Jianying
- Corona, Aaron
- Price, Olga
- Gill, Charles
- Shah, Kashmira
- Rasa, Cordelia
- Tong, Vince
- Owens, Karen
- Ormes, James
- Tang, Haifeng
- Roy, Sophie
- Sullivan, Kathleen A
- Metzger, Joseph M
- Alonso-Galicia, Magdalena
- Kaczorowski, Gregory J
- Pasternak, Alexander
- Garcia, Maria L
Producer: 20170526
In:
The Journal of pharmacology and experimental therapeutics vol. 359
Availability: No items available.
|
|
19.
|
Discovery of a highly potent, selective, and bioavailable soluble epoxide hydrolase inhibitor with excellent ex vivo target engagement. [electronic resource] by
- Shen, Hong C
- Ding, Fa-Xiang
- Wang, Siyi
- Deng, Qiaolin
- Zhang, Xiaoping
- Chen, Yuli
- Zhou, Gaochao
- Xu, Suoyu
- Chen, Hsuan-Shen
- Tong, Xinchun
- Tong, Vincent
- Mitra, Kaushik
- Kumar, Sanjeev
- Tsai, Christine
- Stevenson, Andra S
- Pai, Lee-Yuh
- Alonso-Galicia, Magdalena
- Chen, Xiaoli
- Soisson, Stephen M
- Roy, Sophie
- Zhang, Bei
- Tata, James R
- Berger, Joel P
- Colletti, Steven L
Producer: 20100701
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
|
|
20.
|
The design and synthesis of novel spirocyclic heterocyclic sulfone ROMK inhibitors as diuretics. [electronic resource] by
- Chobanian, Harry R
- Guo, Yan
- Pio, Barbara
- Tang, Haifeng
- Teumelsan, Nardos
- Clements, Matthew
- Frie, Jessica
- Ferguson, Ronald
- Guo, Zach
- Thomas-Fowlkes, Brande S
- Felix, John P
- Liu, Jessica
- Kohler, Martin
- Priest, Birgit
- Hampton, Caryn
- Pai, Lee-Yuh
- Corona, Aaron
- Metzger, Joseph
- Tong, Vincent
- Joshi, Elizabeth M
- Xu, Ling
- Owens, Karen
- Maloney, Kevin
- Sullivan, Kathleen
- Pasternak, Alexander
Producer: 20170818
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
|