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Integrated strategies for identifying leads that target the NS3 helicase of the hepatitis C virus. [electronic resource] by
- LaPlante, Steven R
- Padyana, Anil K
- Abeywardane, Asitha
- Bonneau, Pierre
- Cartier, Mireille
- Coulombe, René
- Jakalian, Araz
- Wildeson-Jones, Jessi
- Li, Xiang
- Liang, Shuang
- McKercher, Ginette
- White, Peter
- Zhang, Qiang
- Taylor, Steven J
Producer: 20140515
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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7.
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Discovery of potent, selective chymase inhibitors via fragment linking strategies. [electronic resource] by
- Taylor, Steven J
- Padyana, Anil K
- Abeywardane, Asitha
- Liang, Shuang
- Hao, Ming-Hong
- De Lombaert, Stéphane
- Proudfoot, John
- Farmer, Bennett S
- Li, Xiang
- Collins, Brandon
- Martin, Leslie
- Albaugh, Daniel R
- Hill-Drzewi, Melissa
- Pullen, Steven S
- Takahashi, Hidenori
Producer: 20130820
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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8.
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Structure and inhibition mechanism of the catalytic domain of human squalene epoxidase. [electronic resource] by
- Padyana, Anil K
- Gross, Stefan
- Jin, Lei
- Cianchetta, Giovanni
- Narayanaswamy, Rohini
- Wang, Feng
- Wang, Rui
- Fang, Cheng
- Lv, Xiaobing
- Biller, Scott A
- Dang, Lenny
- Mahoney, Christopher E
- Nagaraja, Nelamangala
- Pirman, David
- Sui, Zhihua
- Popovici-Muller, Janeta
- Smolen, Gromoslaw A
Producer: 20190205
In:
Nature communications vol. 10
Availability: No items available.
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9.
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Indole RSK inhibitors. Part 1: discovery and initial SAR. [electronic resource] by
- Boyer, Stephen J
- Burke, Jennifer
- Guo, Xin
- Kirrane, Thomas M
- Snow, Roger J
- Zhang, Yunlong
- Sarko, Chris
- Soleymanzadeh, Lida
- Swinamer, Alan
- Westbrook, John
- Dicapua, Frank
- Padyana, Anil
- Cogan, Derek
- Gao, Amy
- Xiong, Zhaoming
- Madwed, Jeffrey B
- Kashem, Mohammed
- Kugler, Stanley
- O'Neill, Margaret M
Producer: 20120803
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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10.
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Correction to Fragment-Based Discovery of Indole Inhibitors of Matrix Metalloproteinase-13. [electronic resource] by
- Taylor, Steven J
- Abeywardane, Asitha
- Liang, Shuang
- Muegge, Ingo
- Padyana, Anil K
- Xiong, Zhaoming
- Hill-Drzewi, Melissa
- Farmer, Bennett
- Li, Xiang
- Collins, Brandon
- Li, John Xiang
- Heim-Riether, Alexander
- Proudfoot, John
- Zhang, Qiang
- Goldberg, Daniel
- Zuvela-Jelaska, Ljiljana
- Zaher, Hani
- Li, Jun
- Farrow, Neil A
Producer: 20151028
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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11.
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Distinct Hepatic PKA and CDK Signaling Pathways Control Activity-Independent Pyruvate Kinase Phosphorylation and Hepatic Glucose Production. [electronic resource] by
- Gassaway, Brandon M
- Cardone, Rebecca L
- Padyana, Anil K
- Petersen, Max C
- Judd, Evan T
- Hayes, Sebastian
- Tong, Shuilong
- Barber, Karl W
- Apostolidi, Maria
- Abulizi, Abudukadier
- Sheetz, Joshua B
- Aerni, Hans R
- Gross, Stefan
- Kung, Charles
- Samuel, Varman T
- Shulman, Gerald I
- Kibbey, Richard G
- Rinehart, Jesse
Producer: 20200923
In:
Cell reports vol. 29
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12.
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Fragment-based discovery of indole inhibitors of matrix metalloproteinase-13. [electronic resource] by
- Taylor, Steven J
- Abeywardane, Asitha
- Liang, Shuang
- Muegge, Ingo
- Padyana, Anil K
- Xiong, Zhaoming
- Hill-Drzewi, Melissa
- Farmer, Bennett
- Li, Xiang
- Collins, Brandon
- Li, John Xiang
- Heim-Riether, Alexander
- Proudfoot, John
- Zhang, Qiang
- Goldberg, Daniel
- Zuvela-Jelaska, Ljiljana
- Zaher, Hani
- Li, Jun
- Farrow, Neil A
Producer: 20120305
In:
Journal of medicinal chemistry vol. 54
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13.
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Vorasidenib (AG-881): A First-in-Class, Brain-Penetrant Dual Inhibitor of Mutant IDH1 and 2 for Treatment of Glioma. [electronic resource] by
- Konteatis, Zenon
- Artin, Erin
- Nicolay, Brandon
- Straley, Kimberly
- Padyana, Anil K
- Jin, Lei
- Chen, Yue
- Narayaraswamy, Rohini
- Tong, Shuilong
- Wang, Feng
- Zhou, Ding
- Cui, Dawei
- Cai, Zhenwei
- Luo, Zhiyong
- Fang, Cheng
- Tang, Huachun
- Lv, Xiaobing
- Nagaraja, Raj
- Yang, Hua
- Su, Shin-San M
- Sui, Zhihua
- Dang, Lenny
- Yen, Katharine
- Popovici-Muller, Janeta
- Codega, Paolo
- Campos, Carl
- Mellinghoff, Ingo K
- Biller, Scott A
Publication details: ACS medicinal chemistry letters Feb 2020
In:
ACS medicinal chemistry letters vol. 11
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14.
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A chemical biology screen identifies a vulnerability of neuroendocrine cancer cells to SQLE inhibition. [electronic resource] by
- Mahoney, Christopher E
- Pirman, David
- Chubukov, Victor
- Sleger, Taryn
- Hayes, Sebastian
- Fan, Zi Peng
- Allen, Eric L
- Chen, Ying
- Huang, Lingling
- Liu, Meina
- Zhang, Yingjia
- McDonald, Gabrielle
- Narayanaswamy, Rohini
- Choe, Sung
- Chen, Yue
- Gross, Stefan
- Cianchetta, Giovanni
- Padyana, Anil K
- Murray, Stuart
- Liu, Wei
- Marks, Kevin M
- Murtie, Joshua
- Dorsch, Marion
- Jin, Shengfang
- Nagaraja, Nelamangala
- Biller, Scott A
- Roddy, Thomas
- Popovici-Muller, Janeta
- Smolen, Gromoslaw A
Producer: 20190205
In:
Nature communications vol. 10
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15.
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Synthesis, SAR, and series evolution of novel oxadiazole-containing 5-lipoxygenase activating protein inhibitors: discovery of 2-[4-(3-{(r)-1-[4-(2-amino-pyrimidin-5-yl)-phenyl]-1-cyclopropyl-ethyl}-[1,2,4]oxadiazol-5-yl)-pyrazol-1-yl]-N,N-dimethyl-acetamide (BI 665915). [electronic resource] by
- Takahashi, Hidenori
- Riether, Doris
- Bartolozzi, Alessandra
- Bosanac, Todd
- Berger, Valentina
- Binetti, Ralph
- Broadwater, John
- Chen, Zhidong
- Crux, Rebecca
- De Lombaert, Stéphane
- Dave, Rajvee
- Dines, Jonathon A
- Fadra-Khan, Tazmeen
- Flegg, Adam
- Garrigou, Michael
- Hao, Ming-Hong
- Huber, John
- Hutzler, J Matthew
- Kerr, Steven
- Kotey, Adrian
- Liu, Weimin
- Lo, Ho Yin
- Loke, Pui Leng
- Mahaney, Paige E
- Morwick, Tina M
- Napier, Spencer
- Olague, Alan
- Pack, Edward
- Padyana, Anil K
- Thomson, David S
- Tye, Heather
- Wu, Lifen
- Zindell, Renee M
- Abeywardane, Asitha
- Simpson, Thomas
Producer: 20150507
In:
Journal of medicinal chemistry vol. 58
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16.
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AG-221, a First-in-Class Therapy Targeting Acute Myeloid Leukemia Harboring Oncogenic [electronic resource] by
- Yen, Katharine
- Travins, Jeremy
- Wang, Fang
- David, Muriel D
- Artin, Erin
- Straley, Kimberly
- Padyana, Anil
- Gross, Stefan
- DeLaBarre, Byron
- Tobin, Erica
- Chen, Yue
- Nagaraja, Raj
- Choe, Sung
- Jin, Lei
- Konteatis, Zenon
- Cianchetta, Giovanni
- Saunders, Jeffrey O
- Salituro, Francesco G
- Quivoron, Cyril
- Opolon, Paule
- Bawa, Olivia
- Saada, Véronique
- Paci, Angelo
- Broutin, Sophie
- Bernard, Olivier A
- de Botton, Stéphane
- Marteyn, Benoît S
- Pilichowska, Monika
- Xu, YingXia
- Fang, Cheng
- Jiang, Fan
- Wei, Wentao
- Jin, Shengfang
- Silverman, Lee
- Liu, Wei
- Yang, Hua
- Dang, Lenny
- Dorsch, Marion
- Penard-Lacronique, Virginie
- Biller, Scott A
- Su, Shin-San Michael
Producer: 20180102
In:
Cancer discovery vol. 7
Availability: No items available.
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17.
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Outcome of the First wwPDB/CCDC/D3R Ligand Validation Workshop. [electronic resource] by
- Adams, Paul D
- Aertgeerts, Kathleen
- Bauer, Cary
- Bell, Jeffrey A
- Berman, Helen M
- Bhat, Talapady N
- Blaney, Jeff M
- Bolton, Evan
- Bricogne, Gerard
- Brown, David
- Burley, Stephen K
- Case, David A
- Clark, Kirk L
- Darden, Tom
- Emsley, Paul
- Feher, Victoria A
- Feng, Zukang
- Groom, Colin R
- Harris, Seth F
- Hendle, Jorg
- Holder, Thomas
- Joachimiak, Andrzej
- Kleywegt, Gerard J
- Krojer, Tobias
- Marcotrigiano, Joseph
- Mark, Alan E
- Markley, John L
- Miller, Matthew
- Minor, Wladek
- Montelione, Gaetano T
- Murshudov, Garib
- Nakagawa, Atsushi
- Nakamura, Haruki
- Nicholls, Anthony
- Nicklaus, Marc
- Nolte, Robert T
- Padyana, Anil K
- Peishoff, Catherine E
- Pieniazek, Susan
- Read, Randy J
- Shao, Chenghua
- Sheriff, Steven
- Smart, Oliver
- Soisson, Stephen
- Spurlino, John
- Stouch, Terry
- Svobodova, Radka
- Tempel, Wolfram
- Terwilliger, Thomas C
- Tronrud, Dale
- Velankar, Sameer
- Ward, Suzanna C
- Warren, Gregory L
- Westbrook, John D
- Williams, Pamela
- Yang, Huanwang
- Young, Jasmine
Producer: 20161216
In:
Structure (London, England : 1993) vol. 24
Availability: No items available.
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