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Identification of novel HSP90α/β isoform selective inhibitors using structure-based drug design. demonstration of potential utility in treating CNS disorders such as Huntington's disease. [electronic resource] by
- Ernst, Justin T
- Neubert, Timothy
- Liu, Michael
- Sperry, Samuel
- Zuccola, Harmon
- Turnbull, Amy
- Fleck, Beth
- Kargo, William
- Woody, Lisa
- Chiang, Peggy
- Tran, Dao
- Chen, Weichao
- Snyder, Phillip
- Alcacio, Timothy
- Nezami, Azin
- Reynolds, James
- Alvi, Khisal
- Goulet, Lance
- Stamos, Dean
Producer: 20140706
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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13.
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Preclinical activity of VX-787, a first-in-class, orally bioavailable inhibitor of the influenza virus polymerase PB2 subunit. [electronic resource] by
- Byrn, Randal A
- Jones, Steven M
- Bennett, Hamilton B
- Bral, Chris
- Clark, Michael P
- Jacobs, Marc D
- Kwong, Ann D
- Ledeboer, Mark W
- Leeman, Joshua R
- McNeil, Colleen F
- Murcko, Mark A
- Nezami, Azin
- Perola, Emanuele
- Rijnbrand, Rene
- Saxena, Kumkum
- Tsai, Alice W
- Zhou, Yi
- Charifson, Paul S
Producer: 20151202
In:
Antimicrobial agents and chemotherapy vol. 59
Availability: No items available.
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14.
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Discovery of a novel, first-in-class, orally bioavailable azaindole inhibitor (VX-787) of influenza PB2. [electronic resource] by
- Clark, Michael P
- Ledeboer, Mark W
- Davies, Ioana
- Byrn, Randal A
- Jones, Steven M
- Perola, Emanuele
- Tsai, Alice
- Jacobs, Marc
- Nti-Addae, Kwame
- Bandarage, Upul K
- Boyd, Michael J
- Bethiel, Randy S
- Court, John J
- Deng, Hongbo
- Duffy, John P
- Dorsch, Warren A
- Farmer, Luc J
- Gao, Huai
- Gu, Wenxin
- Jackson, Katrina
- Jacobs, Dylan H
- Kennedy, Joseph M
- Ledford, Brian
- Liang, Jianglin
- Maltais, François
- Murcko, Mark
- Wang, Tiansheng
- Wannamaker, M Woods
- Bennett, Hamilton B
- Leeman, Joshua R
- McNeil, Colleen
- Taylor, William P
- Memmott, Christine
- Jiang, Min
- Rijnbrand, Rene
- Bral, Christopher
- Germann, Ursula
- Nezami, Azin
- Zhang, Yuegang
- Salituro, Francesco G
- Bennani, Youssef L
- Charifson, Paul S
Producer: 20150207
In:
Journal of medicinal chemistry vol. 57
Availability: No items available.
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